Wolfgang Haap

2.1k total citations
36 papers, 1.6k citations indexed

About

Wolfgang Haap is a scholar working on Molecular Biology, Organic Chemistry and Computational Theory and Mathematics. According to data from OpenAlex, Wolfgang Haap has authored 36 papers receiving a total of 1.6k indexed citations (citations by other indexed papers that have themselves been cited), including 19 papers in Molecular Biology, 11 papers in Organic Chemistry and 6 papers in Computational Theory and Mathematics. Recurrent topics in Wolfgang Haap's work include Chemical Synthesis and Analysis (11 papers), Computational Drug Discovery Methods (6 papers) and Crystallography and molecular interactions (6 papers). Wolfgang Haap is often cited by papers focused on Chemical Synthesis and Analysis (11 papers), Computational Drug Discovery Methods (6 papers) and Crystallography and molecular interactions (6 papers). Wolfgang Haap collaborates with scholars based in Switzerland, Germany and United States. Wolfgang Haap's co-authors include François Diederich, David W. Banner, Jörg Benz, Bernd Kuhn, Guido Hartmann, Lilli Anselm, Ralf Thoma, Bernard Gsell, M. Stihle and Jean‐Marc Plancher and has published in prestigious journals such as Science, Angewandte Chemie International Edition and Nature Immunology.

In The Last Decade

Wolfgang Haap

36 papers receiving 1.6k citations

Peers

Wolfgang Haap
Bernard Gsell Switzerland
M. Stihle Switzerland
Carlos H. Faerman United States
David Hangauer United States
Ken A. Brameld United States
Joachim Diez Switzerland
Peter J. Dandliker United States
Bernard Gsell Switzerland
Wolfgang Haap
Citations per year, relative to Wolfgang Haap Wolfgang Haap (= 1×) peers Bernard Gsell

Countries citing papers authored by Wolfgang Haap

Since Specialization
Citations

This map shows the geographic impact of Wolfgang Haap's research. It shows the number of citations coming from papers published by authors working in each country. You can also color the map by specialization and compare the number of citations received by Wolfgang Haap with the expected number of citations based on a country's size and research output (numbers larger than one mean the country cites Wolfgang Haap more than expected).

Fields of papers citing papers by Wolfgang Haap

Since Specialization
Physical SciencesHealth SciencesLife SciencesSocial Sciences

This network shows the impact of papers produced by Wolfgang Haap. Nodes represent research fields, and links connect fields that are likely to share authors. Colored nodes show fields that tend to cite the papers produced by Wolfgang Haap. The network helps show where Wolfgang Haap may publish in the future.

Co-authorship network of co-authors of Wolfgang Haap

This figure shows the co-authorship network connecting the top 25 collaborators of Wolfgang Haap. A scholar is included among the top collaborators of Wolfgang Haap based on the total number of citations received by their joint publications. Widths of edges represent the number of papers authors have co-authored together. Node borders signify the number of papers an author published with Wolfgang Haap. Wolfgang Haap is excluded from the visualization to improve readability, since they are connected to all nodes in the network.

All Works

20 of 20 papers shown
1.
Dragovich, Peter S., Wolfgang Haap, Melinda M. Mulvihill, Jean‐Marc Plancher, & Antonia F. Stepan. (2022). Small-Molecule Lead-Finding Trends across the Roche and Genentech Research Organizations. Journal of Medicinal Chemistry. 65(4). 3606–3615. 11 indexed citations
2.
Kuhn, Bernd, Wolfgang Haap, U. Obst-Sander, Christian Krämer, & Martin Ståhl. (2021). What We Learned in 25 Years of Interactive Molecular Design Sessions. ChemMedChem. 16(18). 2760–2763. 4 indexed citations
3.
Giroud, Maude, Bernd Kuhn, Rainer E. Martin, et al.. (2018). 2H-1,2,3-Triazole-Based Dipeptidyl Nitriles: Potent, Selective, and Trypanocidal Rhodesain Inhibitors by Structure-Based Design. Journal of Medicinal Chemistry. 61(8). 3370–3388. 44 indexed citations
4.
Kim, Sun Jung, Sebastian Schätzle, Sohail Ahmed, et al.. (2017). Increased cathepsin S in Prdm1−/− dendritic cells alters the TFH cell repertoire and contributes to lupus. Nature Immunology. 18(9). 1016–1024. 58 indexed citations
5.
Theron, Michel, Ana Patrícia Silva, Bernhard Reis, et al.. (2017). Cathepsin S inhibition suppresses autoimmune-triggered inflammatory responses in macrophages. Biochemical Pharmacology. 146. 151–164. 33 indexed citations
6.
Kumar, Santhosh V., Yajuan Liu, Shrikant R. Mulay, et al.. (2017). Cathepsin S inhibition combines control of systemic and peripheral pathomechanisms of autoimmune tissue injury. Scientific Reports. 7(1). 2775–2775. 47 indexed citations
7.
Qiu, Zongxing, Bernd Kuhn, Johannes D. Aebi, et al.. (2016). Discovery of Fluoromethylketone-Based Peptidomimetics as Covalent ATG4B (Autophagin-1) Inhibitors. ACS Medicinal Chemistry Letters. 7(8). 802–806. 55 indexed citations
8.
Figueiredo, Jose‐Luiz, Masanori Aikawa, Chunyu Zheng, et al.. (2015). Selective Cathepsin S Inhibition Attenuates Atherosclerosis in Apolipoprotein E–Deficient Mice with Chronic Renal Disease. American Journal Of Pathology. 185(4). 1156–1166. 63 indexed citations
9.
Rupanagudi, Khader Valli, Onkar P. Kulkarni, Julia Lichtnekert, et al.. (2013). Cathepsin S inhibition suppresses systemic lupus erythematosus and lupus nephritis because cathepsin S is essential for MHC class II-mediated CD4 T cell and B cell priming. Annals of the Rheumatic Diseases. 74(2). 452–463. 82 indexed citations
11.
Hardegger, Leo A., Bernd Kuhn, Lilli Anselm, et al.. (2011). Halogen Bonding at the Active Sites of Human Cathepsin L and MEK1 Kinase: Efficient Interactions in Different Environments. ChemMedChem. 6(11). 2048–2054. 105 indexed citations
12.
Hebeisen, Paul, Wolfgang Haap, Bernd Kuhn, et al.. (2011). Orally active aminopyridines as inhibitors of tetrameric fructose-1,6-bisphosphatase. Bioorganic & Medicinal Chemistry Letters. 21(11). 3237–3242. 14 indexed citations
13.
Salonen, Laura M., Mareike C. Holland, Philip S. J. Kaib, et al.. (2011). Molecular Recognition at the Active Site of Factor Xa: Cation–π Interactions, Stacking on Planar Peptide Surfaces, and Replacement of Structural Water. Chemistry - A European Journal. 18(1). 213–222. 48 indexed citations
14.
Hardegger, Leo A., Bernd Kuhn, Lilli Anselm, et al.. (2010). Systematic Investigation of Halogen Bonding in Protein–Ligand Interactions. Angewandte Chemie International Edition. 50(1). 314–318. 423 indexed citations
15.
Anselm, Lilli, David W. Banner, Jörg Benz, et al.. (2010). Discovery of a factor Xa inhibitor (3R,4R)-1-(2,2-difluoro-ethyl)-pyrrolidine-3,4-dicarboxylic acid 3-[(5-chloro-pyridin-2-yl)-amide] 4-{[2-fluoro-4-(2-oxo-2H-pyridin-1-yl)-phenyl]-amide} as a clinical candidate. Bioorganic & Medicinal Chemistry Letters. 20(17). 5313–5319. 31 indexed citations
16.
Kitas, Eric, Peter J. Mohr, Bernd Kuhn, et al.. (2009). Sulfonylureido thiazoles as fructose-1,6-bisphosphatase inhibitors for the treatment of Type-2 diabetes. Bioorganic & Medicinal Chemistry Letters. 20(2). 594–599. 25 indexed citations
17.
Salonen, Laura M., C. Bucher, David W. Banner, et al.. (2008). Cation–π Interactions at the Active Site of Factor Xa: Dramatic Enhancement upon Stepwise N‐Alkylation of Ammonium Ions. Angewandte Chemie International Edition. 48(4). 811–814. 71 indexed citations
18.
Goodnow, Robert A., Wolfgang Guba, & Wolfgang Haap. (2003). Library Design Practices for Success in Lead Generation With Small Molecule Libraries. Combinatorial Chemistry & High Throughput Screening. 6(7). 649–660. 22 indexed citations
19.
Haap, Wolfgang, Tilmann Walk, & Günther Jung. (1998). FT-IR Mapping—A New Tool for Spatially Resolved Characterization of Polymer-Bound Combinatorial Compound Libraries with IR Microscopy. Angewandte Chemie International Edition. 37(23). 3311–3314. 20 indexed citations
20.
Haap, Wolfgang, Jörg W. Metzger, Christoph Kempter, & Günther Jung. (1997). Composition and Purity of Combinatorial Aryl Ether Collections Analyzed by Electrospray Mass Spectrometry. Molecular Diversity. 3(1). 29–41. 8 indexed citations

Rankless uses publication and citation data sourced from OpenAlex, an open and comprehensive bibliographic database. While OpenAlex provides broad and valuable coverage of the global research landscape, it—like all bibliographic datasets—has inherent limitations. These include incomplete records, variations in author disambiguation, differences in journal indexing, and delays in data updates. As a result, some metrics and network relationships displayed in Rankless may not fully capture the entirety of a scholar's output or impact.

Explore authors with similar magnitude of impact

Rankless by CCL
2026