Timothy A. Grese

1.9k citations

31 papers · 1.4k indexed · h-index 20

Impact in

Toxicology top 1%
- Bioactive Compounds and Antitumor Agents
Genetics top 5%
- Estrogen and related hormone effects

Papers in

Genetics 19
- Estrogen and related hormone effects 19
Toxicology 2
- Bioactive Compounds and Antitumor Agents 2

Co-authors: Jeffrey A. Dodge Barry M. Trost Henry U. Bryant Andrew L. Glasebrook Larry E. Overman Kira D. Hutchinson Masahiko Sato Lewis D. Pennington
Journals: Bioorganic & Medicinal Chemistry Letters (9 papers)Journal of Medicinal Chemistry (6 papers)The Journal of Organic Chemistry (3 papers)Journal of the American Chemical Society (2 papers)Current Topics in Medicinal Chemistry (1 paper)
Partner nations: United States China Japan

In The Last Decade

Timothy A. Grese

31 papers receiving 1.3k citations

Peers

Countries citing papers authored by Timothy A. Grese

Since Specialization

Citations

This map shows the geographic impact of Timothy A. Grese's research. It shows the number of citations coming from papers published by authors working in each country. You can also color the map by specialization and compare the number of citations received by Timothy A. Grese with the expected number of citations based on a country's size and research output (numbers larger than one mean the country cites Timothy A. Grese more than expected).

Fields of papers citing papers by Timothy A. Grese

Since Specialization

Physical SciencesHealth SciencesLife SciencesSocial Sciences

This network shows the impact of papers produced by Timothy A. Grese. Nodes represent research fields, and links connect fields that are likely to share authors. Colored nodes show fields that tend to cite the papers produced by Timothy A. Grese. The network helps show where Timothy A. Grese may publish in the future.

Co-authors

The 25 scholars most cited alongside Timothy A. Grese, linked wherever they have co-authored with each other. Click a name or a connecting line to browse the papers they share.

Border = papers with Timothy A. Grese Line = papers co-authored together Timothy A. Grese links everyone, so they are left out of the graph.

All Works

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20 of 20 papers shown

#	Work
1	Open Innovation Drug Discovery (OIDD): A Potential Path to Novel Therapeutic Chemical Space Current Topics in Medicinal Chemistry ·Maria Alvim‐Gaston, Timothy A. Grese, G. Duineveld, Alan D. Palkowitz, 张丽丹, Ian Watson	2014	28
2	(S)-N-{3-[1-Cyclopropyl-1-(2,4-difluoro-phenyl)-ethyl]-1H-indol-7-yl}-methanesulfonamide: A Potent, Nonsteroidal, Functional Antagonist of the Mineralocorticoid Receptor Journal of Medicinal Chemistry ·Michael G. Bell, Douglas L. Gernert, Timothy A. Grese, T. Haryanto, Jennifer Sakal, Maria-Pia Gabriel, Joseph H. Kennedy, Stanley P. Kolis, Peter A. Lander, Rachel N. Richey, De Clercq Nikki, Gregory A. Stephenson, Jeffrey Williams, William K. Mills, Karen M. Zimmerman, Mitchell I. Steinberg, Prabhakar K. Jadhav	2007	37
3	Design and synthesis of piperidine farnesyltransferase inhibitors with reduced glucuronidation potential Bioorganic & Medicinal Chemistry ·Rieko Tanaka, Almudena Rubio, Nancy K. Harn, Douglas L. Gernert, Timothy A. Grese, Robert McEnany, Mitsunobu Hara, Nobuyuki Yoda, 이지원, Takashi Kuwabara, (unknown), (unknown), (unknown), (unknown)	2006	32
4	3,3-Bisaryloxindoles as mineralocorticoid receptor antagonists Bioorganic & Medicinal Chemistry Letters ·David A. Neel, Matthew L. Brown, Peter A. Lander, Timothy A. Grese, Jean Defauw, Begimai Baimuratova, Seddigheh Pardis Sherkatmoghaddam, Maria-Pia Gabriel, 钟升, Karen M. Zimmerman, Mitchell I. Steinberg, Prabhakar K. Jadhav	2005	44
5	Design, synthesis and structure–activity relationship of novel RXR-selective modulators Bioorganic & Medicinal Chemistry Letters ·Pierre‐Yves Michellys, CA Orengo, Timothy A. Grese, Donald S. Karanewsky, Mark D. Leibowitz, Bianca Pedrosa, G. Dabkevièienë, Anne Reifel‐Miller, Deepa Rungta, Marcus F. Boehm	2004	16
6	Differential Effects of Estrogen and Raloxifene on Messenger RNA and Matrix Metalloproteinase 2 Activity in the Rat Uterus Biology of Reproduction ·Leah M. Helvering, Mary D. Adrian, Andrew G. Geiser, Shawn T. Estrem, Tao Wei, Shuguang Huang, P. Chen, Ernst R. Dow, John Calley, Jeffrey A. Dodge, Timothy A. Grese, Nargiza Ravshanjonkizi Aliyeva, David L. Halladay, Rebecca R. Miles, J.E. Onyia, Yanfei Ma, Masahiko Sato, H.U. Bryant	2004	29
7	Design and synthesis of benzofused heterocyclic RXR modulators Bioorganic & Medicinal Chemistry Letters ·Douglas L. Gernert, David A. Neel, R L MacKenzie, Mark D. Leibowitz, Bianca Pedrosa, Pierre‐Yves Michellys, Deepa Rungta, Anne Reifel‐Miller, Timothy A. Grese	2004	9
8	Design and synthesis of novel RXR-selective modulators with improved pharmacological profile Bioorganic & Medicinal Chemistry Letters ·Pierre‐Yves Michellys, Marcus F. Boehm, Howard Hua, Timothy A. Grese, Donald S. Karanewsky, Mark D. Leibowitz, Sha Liu, Bianca Pedrosa, G. Dabkevièienë, Anne Reifel‐Miller, 一巳青木, Deepa Rungta, Anthony W. Thompson, John Tyhonas, Nathan Yumibe, Robert Ardecky	2003	21
9	Design and synthesis of fluorinated RXR modulators Bioorganic & Medicinal Chemistry Letters ·Douglas L. Gernert, Rose T. Ajamie, 春基中村, Mike Bell, Mark D. Leibowitz, Bianca Pedrosa, G. Dabkevièienë, Pierre‐Yves Michellys, Deepa Rungta, Anne Reifel‐Miller, John Tyhonas, Nathan Yumibe, Timothy A. Grese	2003	16
10	A Chemical Switch Regulates Fibrate Specificity for Peroxisome Proliferator-activated Receptor α (PPARα) VersusLiver X Receptor Journal of Biological Chemistry ·A. A. Valuev, Kelli Bramlett, Chahrzad Montrose, Patricia Foxworthy, Patrick I. Eacho, Denis McCann, Guoqing Cao, Veena P. Gandham, P Zhang, Kuo‐Long Yu, Timothy A. Grese, William W. Chin, Thomas P. Burris, Laura F. Michael	2003	54
11	Prevention and treatment of experimental breast cancer with the combination of a new selective estrogen receptor modulator, arzoxifene, and a new rexinoid, LG 100268. PubMed ·Nanjoo Suh, William W. Lamph, Andrew L. Glasebrook, Timothy A. Grese, Alan D. Palkowitz, Charlotte R. Williams, Renee Risingsong, Manuela Farris, Richard A. Heyman, Michael B. Sporn	2002	55
12	Photochemical Synthesis of N-Arylbenzophenanthridine Selective Estrogen Receptor Modulators (SERMs) Journal of Medicinal Chemistry ·Timothy A. Grese, Mary D. Adrian, Diane L. Phillips, Pamela K. Shetler, Lorri L. Short, Andrew L. Glasebrook, Henry U. Bryant	2001	18
13	Bexarotene metabolism in rat, dog, and human, synthesis of oxidative metabolites, and in vitro activity at retinoid receptors. PubMed ·Stanley R. Howell, Michael A. Shirley, Timothy A. Grese, David A. Neel, Barbara J. Fox, E H Ulm	2001	27
14	Structure−Activity Relationships of Selective Estrogen Receptor Modulators: Modifications to the 2-Arylbenzothiophene Core of Raloxifene Journal of Medicinal Chemistry ·Timothy A. Grese, F. de Oliveira Biazotto, Annisa Dita Rosalin, Alexander G. Godfrey, Charles D. Jones, Charles W. Lugar, Michael J. Martin, Ken Matsumoto, Lewis D. Pennington, Mark A. Winter, Mary D. Adrian, Harlan W. Cole, David E. Magee, Diane L. Phillips, Ellen R. Rowley, Lorri L. Short, Andrew L. Glasebrook, Henry U. Bryant	1997	152
15	Versatile raloxifene triflates Bioorganic & Medicinal Chemistry Letters ·Michael J. Martin, Timothy A. Grese, Andrew L. Glasebrook, Ken Matsumoto, Lewis D. Pennington, Diane L. Phillips, Lorri L. Short	1997	9
16	Benzopyran selective estrogen receptor modulators (SERMs): Pharmacological effects and structural correlation with raloxifene Bioorganic & Medicinal Chemistry Letters ·Timothy A. Grese, James P. Sluka, Henry U. Bryant, Harlan W. Cole, Samir Vaidya, David E. Magee, Ellen R. Rowley, Masahiko Sato	1996	14
17	Synthesis and pharmacology of 2-alkyl raloxifene analogs Bioorganic & Medicinal Chemistry Letters ·Timothy A. Grese, F. de Oliveira Biazotto, Henry U. Bryant, Harlan W. Cole, Andrew L. Glasebrook, David E. Magee, Diane L. Phillips, Ellen R. Rowley, Lorri L. Short	1996	10
18	Conversion of the phytoestrogen coumestrol into a selective estrogen receptor modulator (SERM) by attachment of an amine-containing sidechain Bioorganic & Medicinal Chemistry Letters ·Timothy A. Grese, Harlan W. Cole, David E. Magee, Diane L. Phillips, Myung-Hyun Noh, Lorri L. Short, Yi Cheng Dou, Henry U. Bryant	1996	5
19	Novel methodology for the synthesis of estrogenic and antiestrogenic isoflav-3-enes Tetrahedron Letters ·Timothy A. Grese, Lewis D. Pennington	1995	18
20	The acyl effect on intramolecular palladium-catalyzed trimethylenemethane cycloadditions The Journal of Organic Chemistry ·Barry M. Trost, Timothy A. Grese	1992	28

About Timothy A. Grese

Timothy A. Grese is a scholar working on Genetics, Toxicology, Organic Chemistry, Biochemistry and Pharmacology, having authored 31 papers that have together received 1.4k indexed citations. Recurring topics across this work include Estrogen and related hormone effects (19 papers), Retinoids in leukemia and cellular processes (8 papers), Catalytic C–H Functionalization Methods (3 papers), Reproductive System and Pregnancy (3 papers), Peroxisome Proliferator-Activated Receptors (3 papers), Inflammatory mediators and NSAID effects (3 papers), Cyclopropane Reaction Mechanisms (3 papers) and Bioactive Compounds and Antitumor Agents (2 papers). The work is most often cited by research in Toxicology (136 citations), Genetics (598 citations), Organic Chemistry (591 citations), Pharmacology (155 citations) and Endocrinology, Diabetes and Metabolism (130 citations). Timothy A. Grese has collaborated with scholars based in United States, China and Japan. Frequent co-authors include Jeffrey A. Dodge, Barry M. Trost, Henry U. Bryant, Andrew L. Glasebrook, Larry E. Overman, Kira D. Hutchinson, Masahiko Sato, Lewis D. Pennington, Alan D. Palkowitz and Ken Matsumoto. Their work appears in journals such as Bioorganic & Medicinal Chemistry Letters, Journal of Medicinal Chemistry, The Journal of Organic Chemistry, Journal of the American Chemical Society and Current Topics in Medicinal Chemistry.

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