Tomoyuki Kitazaki

1.6k citations

33 papers · 1.4k · h-index 16

Impact in

Immunology top 5%
- Immune Response and Inflammation
- Immune cells in cancer
Virology top 5%
- HIV Research and Treatment

Papers in

Organic Chemistry 15
- Synthesis and biological activity 8
- Synthesis of Tetrazole Derivatives 7
- Synthesis and Characterization of Heterocyclic Compounds 5
- Synthesis and Biological Evaluation 5
- Click Chemistry and Applications 4
Molecular Biology 7

Co-authors: Masayuki Ii (7 shared papers)Yuji Iizawa (8 shared papers)Tomohiro Kawamoto (1 shared paper)Hiroyuki Kimura (1 shared paper)Katsumi Itoh (13 shared papers)Mie Sunamoto (5 shared papers)Kazuyo Nakamura (2 shared papers)Naoko Matsunaga (2 shared papers)
Journals: Chemical and Pharmaceutical Bulletin (12 papers)Journal of Medicinal Chemistry (4 papers)Bioorganic & Medicinal Chemistry (3 papers)Antimicrobial Agents and Chemotherapy (2 papers)Critical Care Medicine (2 papers)
Partner nations: Japan United States

In The Last Decade

Tomoyuki Kitazaki

33 papers receiving 1.3k citations

Peers

Countries citing papers authored by Tomoyuki Kitazaki

Since Specialization

Citations

This map shows the geographic impact of Tomoyuki Kitazaki's research. It shows the number of citations coming from papers published by authors working in each country. You can also color the map by specialization and compare the number of citations received by Tomoyuki Kitazaki with the expected number of citations based on a country's size and research output (numbers larger than one mean the country cites Tomoyuki Kitazaki more than expected).

Fields of papers citing papers by Tomoyuki Kitazaki

Since Specialization

Physical SciencesHealth SciencesLife SciencesSocial Sciences

This network shows the impact of papers produced by Tomoyuki Kitazaki. Nodes represent research fields, and links connect fields that are likely to share authors. Colored nodes show fields that tend to cite the papers produced by Tomoyuki Kitazaki. The network helps show where Tomoyuki Kitazaki may publish in the future.

Co-authors

The 25 scholars most cited alongside Tomoyuki Kitazaki, linked wherever they have co-authored with each other. Click a name or a connecting line to browse the papers they share.

Border = papers with Tomoyuki Kitazaki Line = papers co-authored together Tomoyuki Kitazaki links everyone, so they are left out of the graph.

All Works

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20 of 20 papers shown

Showing the 20 most-cited of 33 papers — load more, or switch the sort, to bring in the rest.

#	Work
1	A Novel Cyclohexene Derivative, Ethyl (6R)-6-[N-(2-Chloro-4-fluorophenyl)sulfamoyl]cyclohex-1-ene-1-carboxylate (TAK-242), Selectively Inhibits Toll-Like Receptor 4-Mediated Cytokine Production through Suppression of Intracellular Signaling Molecular Pharmacology ·Masayuki Ii, Naoko Matsunaga, Kaoru Hazeki, Kazuyo Nakamura, Katsunori Takashima, Tsukasa Seya, Osamu Hazeki, Tomoyuki Kitazaki, Yuji Iizawa	2005	318
2	TAK-242 selectively suppresses Toll-like receptor 4-signaling mediated by the intracellular domain European Journal of Pharmacology ·Tomohiro Kawamoto, Masayuki Ii, Tomoyuki Kitazaki, Yuji Iizawa, Hiroyuki Kimura	2008	270
3	Therapeutic effects of TAK-242, a novel selective Toll-like receptor 4 signal transduction inhibitor, in mouse endotoxin shock model European Journal of Pharmacology ·Takukyu Sha, Mie Sunamoto, Tomoyuki Kitazaki, Jun Sato, Masayuki Ii, Yuji Iizawa	2007	154
4	Discovery of Novel and Potent Small-Molecule Inhibitors of NO and Cytokine Production as Antisepsis Agents: Synthesis and Biological Activity of Alkyl 6-(N-Substituted sulfamoyl)cyclohex-1-ene-1-carboxylate Journal of Medicinal Chemistry ·Masami Yamada, Takashi Ichikawa, Masayuki Ii, Mie Sunamoto, Katsumi Itoh, Norikazu Tamura, Tomoyuki Kitazaki	2005	96
5	Discovery of 1-{4-[1-(2,6-Difluorobenzyl)-5-[(dimethylamino)methyl]-3-(6-methoxypyridazin-3-yl)-2,4-dioxo-1,2,3,4-tetrahydrothieno[2,3- d ]pyrimidin-6-yl]phenyl}-3-methoxyurea (TAK-385) as a Potent, Orally Active, Non-Peptide Antagonist of the Human Gonadotropin-Releasing Hormone Receptor Journal of Medicinal Chemistry ·Kazuhiro Miwa, Takenori Hitaka, Takashi Imada, Satoshi Sasaki, Mie Yoshimatsu, Masami Kusaka, Akira Tanaka, Daisuke Nakata, Shuichi Furuya, Satoshi Endo, Kazumasa Hamamura, Tomoyuki Kitazaki	2011	86
6	Generation and characterization of a human immunodeficiency virus type 1 (HIV-1) mutant resistant to an HIV-1 protease inhibitor Journal of Virology ·Mohamed A. El‐Farrash, Marcelo J. Kuroda, Tomoyuki Kitazaki, Takao Masuda, Koichi Kato, Masakazu Hatanaka, Shinji Harada	1994	85
7	Novel cyclohexene derivatives as anti-sepsis agents: Synthetic studies and inhibition of NO and cytokine production Bioorganic & Medicinal Chemistry ·Masami Yamada, Takashi Ichikawa, Masayuki Ii, Katsumi Itoh, Norikazu Tamura, Tomoyuki Kitazaki	2008	34
8	Optically Active Antifungal Azoles. VI. Synthesis and Antifungal Activity of N-((1R,2R)-2-(2,4-Difluorophenyl)-2-hydroxy-1-methyl-3-(1H-1,2,4-triazol-1-yl)propyl)-N'-(4-substituted phenyl)-3(2H,4H)-1,2,4-triazolones and 5(1H,4H)-tetrazolones. Chemical and Pharmaceutical Bulletin ·Tomoyuki Kitazaki, Norikazu Tamura, Akihiro Tasaka, Yoshihiro Matsushita, Ryogo HAYASHI, Kenji Okonogi, Katsumi Itoh	1996	25
9	Optically Active Antifungal Azoles. XIII. Synthesis of Stereoisomers and Metabolites of 1-[(1R,2R)-2-(2,4-Difluorophenyl)-2-hydroxy-1-methyl-3-(1H-1,2,4-triazol-1-yl)propyl]-3-[4-(1H-1-tetrazolyl)phenyl]-2-imidazolidinone (TAK-456). Chemical and Pharmaceutical Bulletin ·Takashi Ichikawa, Masami Yamada, Masashi Yamaguchi, Tomoyuki Kitazaki, Yoshihiro Matsushita, Keiko Higashikawa, Katsumi Itoh	2001	25
10	Discovery of a Novel Series ofN-Phenylindoline-5-sulfonamide Derivatives as Potent, Selective, and Orally Bioavailable Acyl CoA:Monoacylglycerol Acyltransferase-2 Inhibitors Journal of Medicinal Chemistry ·Kenjiro Sato, Hiroki Takahagi, Takeshi Yoshikawa, Shinji Morimoto, Takafumi Takai, Kousuke Hidaka, Masahiro Kamaura, Osamu Kubo, Ryutaro Adachi, Tsuyoshi Ishii, Toshiyuki Maki, Taisuke Mochida, Shiro Takekawa, Masanori Nakakariya, Nobuyuki Amano, Tomoyuki Kitazaki	2015	25
11	Optically Active Antifungal Azoles. XII. Synthesis and Antifungal Activity of the Water-Soluble Prodrugs of 1-[(1R,2R)-2-(2,4-Difluorophenyl)-2-hydroxy-1-methyl-3-(1H-1,2,4-triazol-1-yl)propyl]-3-[4-(1H-1-tetrazolyl)phenyl]-2-imidazolidinone. Chemical and Pharmaceutical Bulletin ·Takashi Ichikawa, Tomoyuki Kitazaki, Yoshihiro Matsushita, Masami Yamada, Ryogo HAYASHI, Masashi Yamaguchi, Yutaka Kiyota, Kenji Okonogi, Katsumi Itoh	2001	25
12	Pharmacological Inhibition of Monoacylglycerol O-Acyltransferase 2 Improves Hyperlipidemia, Obesity, and Diabetes by Change in Intestinal Fat Utilization PLoS ONE ·Kazumi Take, Taisuke Mochida, Toshiyuki Maki, Yoshinori Satomi, Megumi Hirayama, Masanori Nakakariya, Nobuyuki Amano, Ryutaro Adachi, Kenjiro Sato, Tomoyuki Kitazaki, Shiro Takekawa	2016	24
13	Optically Active Antifungal Azoles. X. Synthesis and Antifungal Activity of N-[4-(Azolyl)phenyl]- and N-[4-(Azolylmethyl)phenyl]-N'-[(1R,2R)-2-(2,4-difluorophenyl)-2-hydroxy-1-methyl-3-(1H-1,2,4-triazol-1-yl)propyl]-azolones. Chemical and Pharmaceutical Bulletin ·Tomoyuki Kitazaki, Takashi Ichikawa, (unknown), (unknown), (unknown), R Hayashi, Kenji Okonogi, (unknown)	2000	23
14	Optically Active Antifungal Azoles. XI. An Alternative Synthetic Route for 1-[(1R,2R)-2-(2,4-Difluorophenyl)-2-hydroxy-1-methyl-3-(1H-1,2,4-triazol-1-yl)propyl]-3-[4-(1H-1-tetrazolyl)phenyl]-2-imidazolidinone (TAK-456) and Its Analog. Chemical and Pharmaceutical Bulletin ·Takashi Ichikawa, Tomoyuki Kitazaki, Yoshihiro Matsushita, Hiroshi Hosono, Masami Yamada, Masahiro Mizuno, Katsumi Itoh	2000	18
15	Optically Active Antifungal Azoles. VII. Synthesis and Antifungal Activity of Stereoisomers of 2-((1R,2R)-2-(2,4-Difluorophenyl)-2-hydroxy-1-methyl-3-(1H-1,2,4-triazol-1-yl)propyl)-4-(4-(2,2,3,3-tetrafluoropropoxy)phenyl)-3(2H,4H)-1,2,4-triazolone (TAK-187). Chemical and Pharmaceutical Bulletin ·Akihiro Tasaka, Tomoyuki Kitazaki, Noboru Tsuchimori, Yoshihiro Matsushita, (unknown), Kenji Okonogi, Katsumi Itoh	1997	16
16	Optically Active Antifungal Azoles. IV. Synthesis and Antifungal Activity of (2R,3R)-3-Azolyl-2-(substituted phenyl)-1-(1H-1,2,4-triazol-1-yl)-2-butanols. Chemical and Pharmaceutical Bulletin ·Akihiro Tasaka, Norikazu Tamura, Yoshihiro Matsushita, Tomoyuki Kitazaki, Ryogo HAYASHI, Kenji Okonogi, Katsumi Itoh	1995	16
17	Discovery of a novel series of GPR119 agonists: Design, synthesis, and biological evaluation of N-(Piperidin-4-yl)-N-(trifluoromethyl)pyrimidin-4-amine derivatives Bioorganic & Medicinal Chemistry ·Osamu Kubo, Kazuaki Takami, Masahiro Kamaura, Koji Watanabe, Hirohisa Miyashita, Shinichi Abe, Kae Matsuda, Yoshiyuki Tsujihata, Tomoyuki Odani, Shinji Iwasaki, Tomoyuki Kitazaki, Toshiki Murata, Kenjiro Sato	2021	15
18	Functionalized Bilayer Membranes as Artificial Tryptophan Synthase. Characterization of Catalytic Efficiency, Substrate Specificity, and Reaction Selectivity Bulletin of the Chemical Society of Japan ·Yukito Murakami, Jun-ichi Kikuchi, Yoshio Hisaeda, Koichiro Nakamura, Tomoyuki Kitazaki, Hidenori Kaya	1990	13
19	In Vitro and In Vivo Antifungal Activities of TAK-456, a Novel Oral Triazole with a Broad Antifungal Spectrum Antimicrobial Agents and Chemotherapy ·Noboru Tsuchimori, Ryogo HAYASHI, Naomi Kitamoto, Kentaro Asai, Tomoyuki Kitazaki, Yuji Iizawa, Katsumi Itoh, Kenji Okonogi	2002	13
20	Optically Active Cyclohexene Derivative as a New Antisepsis Agent: An Efficient Synthesis of Ethyl (6R)-6-[N-(2-Chloro-4-fluorophenyl)sulfamoyl]cyclohex-1-ene-1-carboxylate (TAK-242) Chemical and Pharmaceutical Bulletin ·Masami Yamada, Takashi Ichikawa, Toru Yamano, Fumio Kikumoto, Yuji Nishikimi, Norikazu Tamura, Tomoyuki Kitazaki	2006	12

About Tomoyuki Kitazaki

Tomoyuki Kitazaki is a scholar working on Organic Chemistry, Molecular Biology, Biochemistry, Immunology and Infectious Diseases, having authored 33 papers that have together received 1.4k indexed citations. Recurring topics across this work include Synthesis and biological activity (8 papers), Synthesis of Tetrazole Derivatives (7 papers), Synthesis and Characterization of Heterocyclic Compounds (5 papers), Synthesis and Biological Evaluation (5 papers), Click Chemistry and Applications (4 papers), Lipid metabolism and biosynthesis (4 papers), Antifungal resistance and susceptibility (3 papers) and Immune Response and Inflammation (3 papers). The work is most often cited by research in Immunology (463 citations), Virology (76 citations), Organic Chemistry (261 citations), Infectious Diseases (150 citations) and Cancer Research (103 citations). Tomoyuki Kitazaki has collaborated with scholars based in Japan and United States. Frequent co-authors include Masayuki Ii, Yuji Iizawa, Tomohiro Kawamoto, Hiroyuki Kimura, Katsumi Itoh, Mie Sunamoto, Kazuyo Nakamura, Naoko Matsunaga, Katsunori Takashima and Kaoru Hazeki. Their work appears in journals such as Chemical and Pharmaceutical Bulletin, Journal of Medicinal Chemistry, Bioorganic & Medicinal Chemistry, Antimicrobial Agents and Chemotherapy and Critical Care Medicine.

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Tomoyuki Kitazaki

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