William Tieu

SuFEx-enabled, agnostic discovery of covalent inhibitors of human neutrophil elastase

Directed Evolution Mimics Allosteric Activation by Stepwise Tuning of the Conformational Ensemble

Reaction site-driven regioselective synthesis of AChE inhibitors

Speculative strategies for new antibacterials: all roads should not lead to Rome

Two-dimensional Zr/Hf-hydroxamate metal–organic frameworks

Role of Biocatalysis in Sustainable Chemistry

Steric and Dynamic Parameters Influencing In Situ Cycloadditions to Form Triazole Inhibitors with Crystalline Acetylcholinesterase

New insights into the kinetic target-guided synthesis of protein ligands

Antibiotics and Bacterial Resistance in the 21st Century

Metal‐Organic Frameworks with Rod Yttrium Secondary Building Units

<i>In Situ</i> Click Chemistry for the Identification of a Potent D-Amino Acid Oxidase Inhibitor

Kinetic Target-Guided Synthesis in Drug Discovery and Chemical Biology: A Comprehensive Facts and Figures Survey

Protein-Catalyzed Capture Agents

Selective inhibition of Biotin Protein Ligase from Staphylococcus aureus

Biotin Analogues with Antibacterial Activity Are Potent Inhibitors of Biotin Protein Ligase

Optimising in situ click chemistry: the screening and identification of biotin protein ligase inhibitors

Reverse Biosynthesis: Generating Combinatorial Pools of Drug Leads from Enzyme‐Mediated Fragmentation of Natural Products

Octadentate Zirconium(IV)-Loaded Macrocycles with Varied Stoichiometry Assembled From Hydroxamic Acid Monomers using Metal-Templated Synthesis