Citation Impact
Citing Papers
In situ click chemistry generation of cyclooxygenase-2 inhibitors
2017 Standout
Recent Researches in Triazole Compounds as Medicinal Drugs
2012
Bioorthogonal Chemistry: Fishing for Selectivity in a Sea of Functionality
2009 StandoutNobel
Imaging beyond the proteome
2012 StandoutNobel
Understanding organofluorine chemistry. An introduction to the C–F bond
2007 Standout
Microwave Assisted Synthesis: A New Technology in Drug Discovery
2009
Rethinking amide bond synthesis
2011 StandoutNature
The crystal structure of human muscle glycogen phosphorylase a with bound glucose and AMP: An intermediate conformation with T‐state and R‐state features
2006
Open Babel: An open chemical toolbox
2011 Standout
Design strategies for bioorthogonal smart probes
2014 StandoutNobel
Marine natural products
1990 Standout
Systemic Fluorescence Imaging of Zebrafish Glycans with Bioorthogonal Chemistry
2015 StandoutNobel
Macrophages in immunoregulation and therapeutics
2023 Standout
Introduction of Fluorine and Fluorine‐Containing Functional Groups
2013 Standout
Differential Recognition of the Type I and II H Antigen Acceptors by the Human ABO(H) Blood Group A and B Glycosyltransferases
2005
A novel interaction fingerprint derived from per atom score contributions: exhaustive evaluation of interaction fingerprint performance in docking based virtual screening
2018
The new era of 1,2,4-oxadiazoles
2009
SuFExable polymers with helical structures derived from thionyl tetrafluoride
2021 StandoutNobel
Synthesis of Oleanolic Acid Dimers as Inhibitors of Glycogen Phosphorylase
2010
Facile synthesis of N-glycosyl amides using a N-glycosyl-2,4-dinitrobenzenesulfonamide and thioacids
2009
Illumination of growth, division and secretion by metabolic labeling of the bacterial cell surface
2015 StandoutNobel
Click Chemistry: 1,2,3‐Triazoles as Pharmacophores
2011 Standout
Microwave-enhanced liquid-phase synthesis of thiohydantoins and thioxotetrahydropyrimidinones
2003
Cu-free click cycloaddition reactions in chemical biology
2010 StandoutNobel
The Polar Hydrophobicity of Fluorinated Compounds
2004
Challenges in the determination of the binding modes of non-standard ligands in X-ray crystal complexes
2010
Synthesis of glucoconjugates of oleanolic acid as inhibitors of glycogen phosphorylase
2009
Thiacycloalkynes for Copper‐Free Click Chemistry
2012 StandoutNobel
Crystallographic and computational studies on 4‐phenyl‐N‐(β‐D ‐glucopyranosyl)‐1H‐1,2,3‐triazole‐1‐acetamide, an inhibitor of glycogen phosphorylase: Comparison with α‐D ‐glucose, N‐acetyl‐β‐D ‐glucopyranosylamine and N‐benzoyl‐N′‐β‐D ‐glucopyranosyl urea binding
2007
A Bioorthogonal Reaction of N‐Oxide and Boron Reagents
2015 StandoutNobel
Mechanisms by which a Very-Low-Calorie Diet Reverses Hyperglycemia in a Rat Model of Type 2 Diabetes
2017
Bringing chemistry to life
2011 StandoutNobel
A Gibbs free energy correlation for automated docking of carbohydrates
2007
Controlled Microwave Heating in Modern Organic Synthesis
2004 Standout
A Fluorogenic Aryl Fluorosulfate for Intraorganellar Transthyretin Imaging in Living Cells and in Caenorhabditis elegans
2015 StandoutNobel
Tetrazine Ligation: Fast Bioconjugation Based on Inverse-Electron-Demand Diels−Alder Reactivity
2008
Targeting Innate Immunity in Cancer Therapy
2021
Click Chemistry for Drug Development and Diverse Chemical–Biology Applications
2013 Standout
Monofluorination of Organic Compounds: 10 Years of Innovation
2015 Standout
SuFEx Click Chemistry Enabled Late-Stage Drug Functionalization
2018 StandoutNobel
Fluorine in Pharmaceutical Industry: Fluorine-Containing Drugs Introduced to the Market in the Last Decade (2001–2011)
2013 Standout
Data-Mining for Sulfur and Fluorine: An Evaluation of Pharmaceuticals To Reveal Opportunities for Drug Design and Discovery
2013 Standout
Mechanisms of Insulin Action and Insulin Resistance
2018 Standout
Multidimensional SuFEx Click Chemistry: Sequential Sulfur(VI) Fluoride Exchange Connections of Diverse Modules Launched From An SOF4 Hub
2017 StandoutNobel
Diversity‐Oriented Syntheses by Combining CuAAC and Stereoselective INCIC Reactions with Peptides
2017 StandoutNobel
Cooperative capture synthesis: yet another playground for copper-free click chemistry
2016 StandoutNobel
An Automated Force Field Topology Builder (ATB) and Repository: Version 1.0
2011 Standout
The Hitchhiker’s Guide to Flow Chemistry
2017 Standout
Development of a Bioorthogonal and Highly Efficient Conjugation Method for Quantum Dots Using Tetrazine−Norbornene Cycloaddition
2010 StandoutNobel
The Medicinal Chemist’s Toolbox: An Analysis of Reactions Used in the Pursuit of Drug Candidates
2011 Standout
Expeditious Synthesis of a Common Intermediate of l -1-Deoxyallonojirimycin and l -1-Deoxymannojirimycin
2009
Amide-1,2,3-triazole bioisosterism: the glycogen phosphorylase case
2009
The Many Roles for Fluorine in Medicinal Chemistry
2008 Standout
Oxadiazoles in Medicinal Chemistry
2011 Standout
Next Generation of Fluorine-Containing Pharmaceuticals, Compounds Currently in Phase II–III Clinical Trials of Major Pharmaceutical Companies: New Structural Trends and Therapeutic Areas
2016 Standout
First synthesis of parazoanthine-A and its O-Me derivative
2012
Fluorine in Pharmaceuticals: Looking Beyond Intuition
2007 StandoutScience
A fluorogenic screening platform enables directed evolution of an alkyne biosynthetic tool
2016 StandoutNobel
Molecular Docking: Shifting Paradigms in Drug Discovery
2019 Standout
Analysis of Past and Present Synthetic Methodologies on Medicinal Chemistry: Where Have All the New Reactions Gone?
2015 Standout
Traceless synthesis of hydantoin by focused microwave irradiation
2003
Fluorine in medicinal chemistry: Recent therapeutic applications of fluorinated small molecules
2006 Standout
Structural and Biochemical Studies of a Fluoroacetyl-CoA-Specific Thioesterase Reveal a Molecular Basis for Fluorine Selectivity
2010 StandoutNobel
Diastereoselective Allylation of Carbonyl Compounds and Imines: Application to the Synthesis of Natural Products
2013 Standout
Synthetic Organic Electrochemical Methods Since 2000: On the Verge of a Renaissance
2017 Standout
A Bioorthogonal Quadricyclane Ligation
2011 StandoutNobel
Design of an Amide N-Glycoside Derivative of β-Glucogallin: A Stable, Potent, and Specific Inhibitor of Aldose Reductase
2013
Diversity Oriented Clicking (DOC): Divergent Synthesis of SuFExable Pharmacophores from 2‐Substituted‐Alkynyl‐1‐Sulfonyl Fluoride (SASF) Hubs
2020 StandoutNobel
Fluorosulfuryl Isocyanate Enabled SuFEx Ligation of Alcohols and Amines
2021 StandoutNobel
First Total Synthesis of 1-O-β-d -Glucopyranosyl-5-deoxyadenophorine and Its Aglycon Congener: Determination of the Absolute Configuration
2004
Synthesis of 3-oxadiazolyl/triazolyl morpholines: Novel scaffolds for drug discovery
2016
Cu-Catalyzed Click Reaction in Carbohydrate Chemistry
2016
Synthetic Approaches and Pharmacological Activity of 1,3,4-Oxadiazoles: A Review of the Literature from 2000–2012
2012
Enantioselective Total Synthesis of (−)-Clavosolide B
2007
Glycosyltransferases: Structures, Functions, and Mechanisms
2007 Standout
Applications of Fluorine in Medicinal Chemistry
2015 Standout
Microwave-assisted traceless synthesis of thiohydantoin
2003
Works of Tibor Docsa being referenced
Synthesis of variously coupled conjugates of d-glucose, 1,3,4-oxadiazole, and 1,2,3-triazole for inhibition of glycogen phosphorylase
2011
Glycogen Phosphorylase Inhibitor N-(3,5-Dimethyl-Benzoyl)-N’-(β-D-Glucopyranosyl)Urea Improves Glucose Tolerance under Normoglycemic and Diabetic Conditions and Rearranges Hepatic Metabolism
2013
Binding of N‐acetyl‐N ′‐β‐d ‐glucopyranosyl urea and N‐benzoyl‐N ′‐β‐d ‐glucopyranosyl urea to glycogen phosphorylase b
2002
Glucose Analog Inhibitors of Glycogen Phosphorylases as Potential Antidiabetic Agents: Recent Developments
2003
Synthesis of 4-amidomethyl-1-glucosyl-1,2,3-triazoles and evaluation as glycogen phosphorylase inhibitors
2014
Efficient inhibition of muscle and liver glycogen phosphorylases by a new glucopyranosylidene-spiro-thiohydantoin
1999
Synthesis of N-(β-d-glucopyranosyl) monoamides of dicarboxylic acids as potential inhibitors of glycogen phosphorylase
2006
Kinetic and crystallographic studies on 2‐(β‐D‐glucopyranosyl)‐5‐methyl‐1, 3, 4‐oxadiazole, ‐benzothiazole, and ‐benzimidazole, inhibitors of muscle glycogen phosphorylase b. Evidence for a new binding site
2005
Kinetic and Crystallographic Studies of Glucopyranosylidene Spirothiohydantoin Binding to Glycogen Phosphorylase b
2002
Synthesis and glycogen phosphorylase inhibitor activity of 2,3-dihydrobenzo[1,4]dioxin derivatives
2007
Synthesis of 1-(d-glucopyranosyl)-1,2,3-triazoles and their evaluation as glycogen phosphorylase inhibitors
2009
Crystallographic studies on two bioisosteric analogues, N-acetyl-β-d-glucopyranosylamine and N-trifluoroacetyl-β-d-glucopyranosylamine, potent inhibitors of muscle glycogen phosphorylase
2005
Synthesis of N-(β-D-glucopyranosyl)- and N-(2-acetamido-2-deoxy-β-D-glucopyranosyl) amides as inhibitors of glycogen phosphorylase
2004
Synthesis of and a Comparative Study on the Inhibition of Muscle and Liver Glycogen Phosphorylases by Epimeric Pairs of d -Gluco- and d -Xylopyranosylidene-spiro-(thio)hydantoins and N-(d -Glucopyranosyl) Amides
2001
Crystallographic Studies on α- and β-D-glucopyranosyl Formamide Analogues, Inhibitors of Glycogen Phosphorylase
2003
In Search of Glycogen Phosphorylase Inhibitors: 5‐Substituted 3‐C‐Glucopyranosyl‐1,2,4‐oxadiazoles from β‐D ‐Glucopyranosyl Cyanides upon Cyclization of O‐Acylamidoxime Intermediates
2006
Tethered derivatives of d-glucose and pentacyclic triterpenes for homo/heterobivalent inhibition of glycogen phosphorylase
2010