Citation Impact
Citing Papers
Anti-Markovnikov alkene oxidation by metal-oxo–mediated enzyme catalysis
2017 StandoutScienceNobel
DNA-Encoded Chemical Libraries: A Selection System Based on Endowing Organic Compounds with Amplifiable Information
2018
Comprehensive computational design of ordered peptide macrocycles
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Palladium‐Catalyzed Cross‐Coupling Reactions in Total Synthesis
2005 Standout
CeCl3·7H2O/IBX-promoted oxidation of 3-alkylindoles to 3-hydroxyoxindoles
2007
Glycopolymer probes of signal transduction
2013
Tumor-targeting peptides from combinatorial libraries
2016
Brønsted Acid Catalyzed, Conjugate Addition of β‐Dicarbonyls to In Situ Generated ortho‐Quinone Methides—Enantioselective Synthesis of 4‐Aryl‐4H‐Chromenes
2014
Asymmetric Counteranion‐Directed Catalysis: Concept, Definition, and Applications
2012 StandoutNobel
Synthesis of Natural Product Inspired Compound Collections
2009
Proton-Coupled Electron Transfer in Organic Synthesis: Fundamentals, Applications, and Opportunities
2016
The evolving role of natural products in drug discovery
2005 Standout
Macrocyclization by Ring‐Closing Metathesis in the Total Synthesis of Natural Products: Reaction Conditions and Limitations
2006
Modern methods to produce natural-product libraries
2002
Potential therapeutics for obesity and atherosclerosis: Inhibitors of neutral lipid metabolism from microorganisms
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Hypervalent Iodine‐Catalyzed Oxidative Functionalizations Including Stereoselective Reactions
2014
A practical synthesis of a high-loading solid-supported IBX amide for the oxidation of alcohols
2005
Dynamic Covalent Chemistry
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Catalytic Three‐Component Ugi Reaction
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Recent advances in homogeneous nickel catalysis
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A Structurally Diverse Library of Polycyclic Lactams Resulting from Systematic Placement of Proximal Functional Groups
2006
The remarkable metal-catalysed olefin metathesis reaction
2007 StandoutNature
Exploring privileged structures: the combinatorial synthesis of cyclic peptides
2002
Catalytic Asymmetric Conjugate Addition/Oxidative Dearomatization Towards Multifunctional Spirocyclic Compounds
2011 StandoutNobel
Natural products as an inspiration in the diversity-oriented synthesis of bioactive compound libraries
2008
Brønsted Acid Catalyzed Asymmetric SN2‐Type O‐Alkylations
2013 StandoutNobel
Pyrrolidinyl‐Spirooxindole Natural Products as Inspirations for the Development of Potential Therapeutic Agents
2007 Standout
Convenient Syntheses of Fluorous Aryl Iodides and Hypervalent Iodine Compounds: ArI(L)n Reagents That Are Recoverable by Simple Liquid/Liquid Biphase Workups, and Applications in Oxidations of Hydroquinones
2002
2‐Iodoxybenzoic Acid—A Simple Oxidant with a Dazzling Array of Potential Applications
2011
A one-bead, one-stock solution approach to chemical genetics: part 1
2001
Genetically programmed chiral organoborane synthesis
2017 StandoutNatureNobel
New Reactions of IBX: Oxidation of Nitrogen‐ and Sulfur‐Containing Substrates To Afford Useful Synthetic Intermediates
2003
Novel Oxygenations with IBX
2009
Advancing chemistry and biology through diversity-oriented synthesis of natural product-like libraries
2005
Protein structure similarity clustering and natural product structure as guiding principles in drug discovery
2005
Chiral amine/chiral acid as an excellent organocatalytic system for the enantioselective tandem oxa-Michael-aldol reaction
2009
Biomimetic Synthesis of (+)‐Ledene, (+)‐Viridiflorol, (−)‐Palustrol, (+)‐Spathulenol, and Psiguadial A, C, and D via the Platform Terpene (+)‐Bicyclogermacrene
2014
Hindered Aryllithium Reagents as Partners in Palladium‐Catalyzed Cross‐Coupling: Synthesis of Tri‐ and Tetra‐ortho‐Substituted Biaryls under Ambient Conditions
2013 StandoutNobel
Phosphoramidites: Privileged Ligands in Asymmetric Catalysis
2010 StandoutNobel
Lead compounds discovered from libraries
2001
The discovery of antibacterial agents using diversity-oriented synthesis
2009
Diversity-oriented synthesis: exploring the intersections between chemistry and biology
2005
Solid-supported reagents in organic synthesis
1999
o‐Iodoxybenzoic Acid (IBX): pKa and Proton‐Affinity Analysis
2006
A Bioorthogonal Reaction of N‐Oxide and Boron Reagents
2015 StandoutNobel
Tetrafluoro‐IBA and‐IBX: Hypervalent Iodine Reagents
2007
Drug Targets in Mycobacterial Sulfur Metabolism
2007
Combinatorial synthesis of novel and potent inhibitors of NADH:ubiquinone oxidoreductase
2000
Design and Enantioselective Synthesis of Cashmeran Odorants by Using “Enol Catalysis”
2015 StandoutNobel
Metathesis Reactions in Total Synthesis
2005
Inhibitors of HIV‐1 Protease by Using In Situ Click Chemistry
2006 StandoutNobel
Enantio‐ and Diastereoselective Access to Distant Stereocenters Embedded within Tetrahydroxanthenes: Utilizing ortho‐Quinone Methides as Reactive Intermediates in Asymmetric Brønsted Acid Catalysis
2014
The Organocatalytic Asymmetric Prins Cyclization
2015 StandoutNobel
Antibacterial drug discovery in the resistance era
2016 StandoutNature
A Versatile and Highly Reactive Polyfluorinated Hypervalent Iodine(III) Compound
2010
IBX Amides: A New Family of Hypervalent Iodine Reagents
2003
Design of compound libraries based on natural product scaffolds and protein structure similarity clustering (PSSC)
2005
Sulfatase-activated fluorophores for rapid discrimination of mycobacterial species and strains
2013 StandoutNobel
IBX/I2-mediated oxidation of alkenes and alkynes in water: a facile synthesis of α-iodoketones
2008
Expedient access to fused quinoxalines via Dess–Martin periodinane-mediated cyclization of unsymmetrical phenylenediamide derivatives
2009
Natural Products as Leads to Potential Drugs: An Old Process or the New Hope for Drug Discovery?
2008
Iodine(III)-mediated aromatic amidation vs olefin amidohydroxylation. The amide N-substituent makes the difference
2004
Natural product-derived building blocks for combinatorial synthesis. Part 1. Fragmentation of natural products from myxobacteria
2002
New chiral hypervalent iodine(V) compounds as stoichiometric oxidants
2010
Chemical Genetics
2006
Catalytic Asymmetric Addition of Aldehydes to Oxocarbenium Ions: A Dual Catalytic System for the Synthesis of Chromenes
2012
Mild Oxidation of Alcohols with o‐Iodoxybenzoic Acid (IBX) in a Water/CH2Cl2 Mixture in the Presence of Phase‐Transfer Catalyst
2006
Chemistry of Polyvalent Iodine
2008 Standout
The chemistry of the carbon–transition metal double and triple bond: annual survey covering the year 1999
2001
Polyvalent iodine in organic chemistry: Recent developments, 2002–2005
2006
Drug Discovery and Natural Products: End of an Era or an Endless Frontier?
2009 StandoutScience
Stereocontrolled synthesis of spirocyclics
1999
Room-Temperature Ionic Liquids: Solvents for Synthesis and Catalysis. 2
2011 Standout
A synthon approach to spiro compounds
2005
Targeted Covalent Inhibitors for Drug Design
2016
Traceless Solid-Phase Organic Synthesis
2002
Synthesis of oxa-aza spirobicycles by intramolecular hydrogen atom transfer promoted by N-radicals in carbohydrate systems
2009
Playing with the Molecules of Life
2018
An Unexpected α‐Oxidation of Cyclic Ketones with 1,4‐Benzoquinone by Enol Catalysis
2018 StandoutNobel
Engineering enzymes for noncanonical amino acid synthesis
2018 StandoutNobel
Deracemization of α-Aryl Hydrocoumarins via Catalytic Asymmetric Protonation of Ketene Dithioacetals
2012 StandoutNobel
Recyclable 2nd generation ionic liquids as green solvents for the oxidation of alcohols with hypervalent iodine reagents
2004
2-Iodoxybenzenesulfonic Acid as an Extremely Active Catalyst for the Selective Oxidation of Alcohols to Aldehydes, Ketones, Carboxylic Acids, and Enones with Oxone
2008
o-Iodoxybenzoic Acid (IBX) as a Viable Reagent in the Manipulation of Nitrogen- and Sulfur-Containing Substrates: Scope, Generality, and Mechanism of IBX-Mediated Amine Oxidations and Dithiane Deprotections
2004
Ein kurzer, atomökonomischer Zugang zu Tetrahydroxanthenonen
2003
Control of the Regioselectivity of Sulfonamidyl Radical Cyclization by Vinylic Halogen Substitution
2007
Ion-dependent protein–surface interactions from intrinsic solvent response
2021 StandoutNobel
Self-Assembling 2D Arrays with de Novo Protein Building Blocks
2019 StandoutNobel
The chemistry of the carbon–transition metal double and triple bond: annual survey covering the year 1998
2000
Modified o-methyl-substituted IBX: room temperature oxidation of alcohols and sulfides in common organic solvents
2007
Biocompatible SuFEx Click Chemistry: Thionyl Tetrafluoride (SOF4)‐Derived Connective Hubs for Bioconjugation to DNA and Proteins
2019 StandoutNobel
Copper-Catalyzed Synthesis of Mixed Alkyl Aryl Phosphonates
2014 StandoutNobel
Stereoinduced cyclization of acyloxyalkenes using iodosylbenzene via a 1,3-dioxan-2-yl cation
2008
Palladium-Mediated Intramolecular Carbonylative Annulation of o-Alkynylphenols To Synthesize Benzo[b]furo[3,4-d]furan-1-ones
2001
Boron Reagents in Process Chemistry: Excellent Tools for Selective Reductions
2006
2018
The chemistry of the carbon-transition metal double and triple bond: annual survey covering the year 1997
1999
Tumor Selectivity of Hsp90 Inhibitors: The Explanation Remains Elusive
2006
The first one-pot oxidative Michael reaction of Baylis–Hillman adducts with indoles promoted by iodoxybenzoic acid
2007
IBX‐Mediated Conversion of Primary Alcohols and Aldehydes to N‐Hydroxysuccinimide Esters
2004
Organohypervalent Iodine: Development, Applications, and Future Directions
2005
Engineering Biomolecular Self‐Assembly at Solid–Liquid Interfaces
2020 StandoutNobel
Rational Tuning of Fluorobenzene Probes for Cysteine‐Selective Protein Modification
2018 StandoutNobel
Palladiumkatalysierte Kreuzkupplungen in der Totalsynthese
2005
New Selenium-Based Safety-Catch Linkers: Solid-Phase Semisynthesis of Vancomycin
2000
Suzuki−Miyaura Cross-Coupling of Aryl Carbamates and Sulfamates: Experimental and Computational Studies
2011
Boronic Acids and Esters in the Petasis-Borono Mannich Multicomponent Reaction
2010
Convenient preparation of unsymmetrical 2,5-disubstituted 1,3,4-oxadiazoles promoted by Dess–Martin reagent
2009
Diverse Functional Roles of Reactive Cysteines
2012
IBX/LiBr-promoted one-pot oxidative anti-Markownikov bromohydroxylation/bromoalkoxylation of Baylis–Hillman olefins
2008
Comprehensive Survey of Combinatorial Library Synthesis: 2005
2006
N,N-DiethylO-Carbamate: Directed Metalation Group and Orthogonal Suzuki−Miyaura Cross-Coupling Partner
2009
Chemically tunable mucin chimeras assembled on living cells
2015 StandoutNobel
Recent Developments in the Chemistry of Polyvalent Iodine Compounds
2002
The Combinatorial Synthesis of Bicyclic Privileged Structures or Privileged Substructures
2003 Standout
High Oxidation State Multiple Metal−Carbon Bonds
2001 StandoutNobel
Enantio‐ and Diastereoselective Access to Distant Stereocenters Embedded within Tetrahydroxanthenes: Utilizing ortho‐Quinone Methides as Reactive Intermediates in Asymmetric Brønsted Acid Catalysis
2014
Adventures in Carbohydrate Chemistry: New Synthetic Technologies, Chemical Synthesis, Molecular Design, and Chemical Biology
2001
Adventures in Carbohydrate Chemistry: New Synthetic Technologies, Chemical Synthesis, Molecular Design, and Chemical Biology A list of abbreviations can be found at the end of this article. Telemachos Charalambous was an inspiring teacher at the Pancyprian Gymnasium, Nicosia, Cyprus.
2001
Advances in Synthetic Applications of Hypervalent Iodine Compounds
2016 Standout
Expedient synthesis and solvent dependent oxidation behavior of a water-soluble IBX derivative
2008
A Heck–Matsuda Process for the Synthesis of β‐Arylethenesulfonyl Fluorides: Selectively Addressable Bis‐electrophiles for SuFEx Click Chemistry
2016 StandoutNobel
Impact of Natural Products on Developing New Anti-Cancer Agents
2009 Standout
Der Stand der Totalsynthese zu Beginn des 21. Jahrhunderts
2000
What is a “DNA-Compatible” Reaction?
2016
Asymmetric Catalysis of the Carbonyl-Amine Condensation: Kinetic Resolution of Primary Amines
2017 StandoutNobel
Organoiodine(V) Reagents in Organic Synthesis
2011
Chiral Organic Contact Ion Pairs in Metal-Free Catalytic Asymmetric Allylic Substitutions
2011
A facile route to a polymer-supported IBX reagent
2003
A one-bead, one-stock solution approach to chemical genetics: part 2
2001
Diastereoselective Aminooxygenation and Diamination of Alkenes with Amidines by Hypervalent Iodine(III) Reagents
2014
Catalytic Asymmetric Intramolecular [4+2] Cycloaddition of In Situ Generated ortho‐Quinone Methides
2017 StandoutNobel
Asymmetric Catalysis via Cyclic, Aliphatic Oxocarbenium Ions
2017 StandoutNobel
Hypervalent iodine-mediated oxygenative phenol dearomatization reactions
2010
Oxidative Dearomatization of Phenols and Anilines via λ3- and λ5-Iodane-Mediated Phenylation and Oxygenation
2005
De Novo Asymmetric Bio- and Chemocatalytic Synthesis of Saccharides − Stereoselective Formal O-Glycoside Bond Formation Using Palladium Catalysis
2003 StandoutNobel
Privileged Structures: Efficient Chemical “Navigators” toward Unexplored Biologically Relevant Chemical Spaces
2014
Protein Glycoengineering Enabled by the Versatile Synthesis of Aminooxy Glycans and the Genetically Encoded Aldehyde Tag
2011 StandoutNobel
Catalytic Asymmetric Synthesis of Cyclic Ethers Containing an α‐Tetrasubstituted Stereocenter
2013
2-Iodoxybenzoic acid (IBX): an efficient hypervalent iodine reagent
2010
Solar Synthesis: Prospects in Visible Light Photocatalysis
2014 StandoutScience
Brønsted‐Säure‐katalysierte konjugierte Addition von β‐Dicarbonylverbindungen an in situ erzeugte ortho‐Chinomethide – enantioselektive Synthese von 4‐Aryl‐4H‐chromenen
2014
Protein Assembly: Versatile Approaches to Construct Highly Ordered Nanostructures
2016
Cyclic [2]Pseudorotaxane Tetramers Consisting of Two Rigid Rods Threaded through Two Bis-Macrocycles: Copper(I)-Templated Synthesis and X-ray Structure Studies
2008 StandoutNobel
Z-Selective Copper-Catalyzed Asymmetric Allylic Alkylation with Grignard Reagents
2012 StandoutNobel
Solvent-free synthesis of 1-(p-toluenesulfonyloxy)-1,2-benziodoxol-3(1H)-one from Dess–Martin periodinane and its synthetic utility for α-tosyloxylation of ketones
2008
On the Phenyliodine(III)‐Bis(trifluoroacetate)‐Mediated Olefin Amidohydroxylation Reaction
2006
A new and practical PIFA-promoted olefin amidohydroxylation: six- versus five-membered ring formation
2003
N‐Carboxyanhydride Polymerization of Glycopolypeptides That Activate Antigen‐Presenting Cells through Dectin‐1 and Dectin‐2
2018 StandoutNobel
Phenyliodonium Zwitterion as an Efficient Electrophile in the Palladium-Catalyzed Suzuki-Type Reaction: A Novel Method for the Synthesis of 3-Aryl-4-hydroxycoumarins
2002
Synthetic Applications of Proton-Coupled Electron Transfer
2016
Generation of Anti-trypanosomal Agents through Concise Synthesis and Structural Diversification of Sesquiterpene Analogues
2011 StandoutNobel
Works of Sofía Barluenga being referenced
Expanding the Scope of PNA‐Encoded Synthesis (PES): Mtt‐Protected PNA Fully Orthogonal to Fmoc Chemistry and a Broad Array of Robust Diversity‐Generating Reactions
2012
Identification of Covalent Bromodomain Binders through DNA Display of Small Molecules
2015
Selection of a synthetic glycan oligomer from a library of DNA-templated fragments against DC-SIGN and inhibition of HIV gp120 binding to dendritic cells
2011
PNA-encoded chemical libraries
2015
Discovery of Novel Antibacterial Agents Active Against Methicillin-ResistantStaphylococcus aureus from Combinatorial Benzopyran Libraries
2001
Diversity‐Oriented Synthesis of Diverse Polycyclic Scaffolds Inspired by the Logic of Sesquiterpene Lactones Biosynthesis
2012
Bromotyrosine-Derived Natural and Synthetic Products as Inhibitors of Mycothiol-S-Conjugate Amidase
2002
Combinatorial Synthesis through Disulfide Exchange: Discovery of Potent Psammaplin A Type Antibacterial Agents Active against Methicillin-ResistantStaphylococcus aureus (MRSA)
2001
Diversity-oriented synthesis of novel polycyclic scaffolds using polymer-bound reagents
2008
Modular Asymmetric Synthesis of Pochonin C
2004
DNA-templated release of functional molecules with an azide-reduction-triggered immolative linker
2011
Natural Product-like Combinatorial Libraries Based on Privileged Structures. 1. General Principles and Solid-Phase Synthesis of Benzopyrans
2000
Total Synthesis of the Novel Immunosuppressant Sanglifehrin A
2000
DNA display of fragment pairs as a tool for the discovery of novel biologically active small molecules
2014
Polymer-supported selenium reagents for organic synthesis
1998
Unexpected Thermal Benzannulation of 1,3,5-Metallahexatrienes: Synthesis of o-Alkoxyphenol-Containing Polycycles
1999
Totalsynthese von Sanglifehrin A
1999
Iodine(V) Reagents in Organic Synthesis. Part 3. New Routes to Heterocyclic Compounds via o-Iodoxybenzoic Acid-Mediated Cyclizations: Generality, Scope, and Mechanism
2002
Diversity‐Oriented Synthesis of Diverse Polycyclic Scaffolds Inspired by the Logic of Sesquiterpene Lactones Biosynthesis
2012
Solid-phase synthesis of benzimidazole libraries biased for RNA targets
2003
Reactions of 2‐Amino‐1,3‐butadienes and Fischer Alkynyl Carbenes: Up to Nine C−C Bonds and Seven Stereogenic Centers Created in a Stereoselective Manner through a Cascade Process
1998
Modular Asymmetric Synthesis of Pochonin C
2004
Screening for covalent inhibitors using DNA-display of small molecule libraries functionalized with cysteine reactive moieties
2016
Enantioselective synthesis of six membered carbocycles through [4+2] cycloaddition reactions of chiral 2-amino-1,3-butadienes and tungsten vinyl Fischer type carbene complexes
1997
Tandem Cycloaddition-Cyclopentannulation Processes of 2-Aminobuta-1,3-dienes and Fischer Alkynylcarbene Complexes as a Tool for the Preparation of Complex Polycyclic Scaffolds
1998
Total Synthesis of Sanglifehrin A
1999
Natural Product-like Combinatorial Libraries Based on Privileged Structures. 3. The “Libraries from Libraries” Principle for Diversity Enhancement of Benzopyran Libraries
2000
Natural Product-like Combinatorial Libraries Based on Privileged Structures. 2. Construction of a 10 000-Membered Benzopyran Library by Directed Split-and-Pool Chemistry Using NanoKans and Optical Encoding
2000
Design, Synthesis, and Biological Evaluation of HSP90 Inhibitors Based on Conformational Analysis of Radicicol and Its Analogues
2005
Self-Assembled Antibody Multimers through Peptide Nucleic Acid Conjugation
2012
Stereospecific [4+2] Reaction between 2-Morpholino-1,3-butadienes and α,β-Unsaturated Exocyclic Chromium Carbene Complexes. Preparation of Enantiomerically Pure Spiro Compounds
1997
Cysteine Mapping in Conformationally Distinct Kinase Nucleotide Binding Sites: Application to the Design of Selective Covalent Inhibitors
2011