Citation Impact
Citing Papers
Palladium-catalyzed N-arylation of 2-aminobenzothiazole-4-carboxylates/carboxamides: facile synthesis of PARP14 inhibitors
2014
Synthesis, Anti‐B reast Cancer Activity, and Molecular Modeling of Some Benzothiazole and Benzoxazole Derivatives
2013
Synthesis of novel inhibitors of β-glucuronidase based on benzothiazole skeleton and study of their binding affinity by molecular docking
2011
Part 1: Structure–Activity Relationship (SAR) investigations of fused pyrazoles as potent, selective and orally available inhibitors of p38α mitogen-activated protein kinase
2009
Synthesis of potent and selective inhibitors of Candida albicans N-myristoyltransferase based on the benzothiazole structure
2005
Benzothiazoles: Search for anticancer agents
2012
Mammalian phosphoinositide kinases and phosphatases
2009 StandoutNobel
New anticancer active and selective phenylene-bisbenzothiazoles: Synthesis, antiproliferative evaluation and DNA binding
2013
Synthesis and cytotoxic evaluation of thiourea and N-bis-benzothiazole derivatives: A novel class of cytotoxic agents
2011
Inhibiting eukaryotic transcription. Which compound to choose? How to evaluate its activity?
2011 Standout
Synthesis of pyrazolo[1,5-a]pyrimidine linked aminobenzothiazole conjugates as potential anticancer agents
2013
Benzothiazoles: How Relevant in Cancer Drug Design Strategy?
2014
PI3Kγ inhibition: towards an 'aspirin of the 21st century'?
2006
Pharmacological targeting of the HIF hydroxylases – A new field in medicine development
2016 StandoutNobel
Lead compounds discovered from libraries: Part 2
2003
Oxidative Geminal Functionalization of Organoboron Compounds
2012
Pharmaceutical and medicinal significance of sulfur (SVI)-Containing motifs for drug discovery: A critical review
2018 Standout
Oncogenic Mutations Counteract Intrinsic Disorder in the EGFR Kinase and Promote Receptor Dimerization
2012 StandoutNobel
Design and synthesis of novel 4-benzothiazole amino quinazolines Dasatinib derivatives as potential anti-tumor agents
2013
SwissParam: A fast force field generation tool for small organic molecules
2011 Standout
Iron catalysed direct alkylation of amines with alcohols
2014 StandoutNobel
4-Thiazolidinone – A biologically active scaffold
2007 Standout
The PtdIns(3,4)P2 phosphatase INPP4A is a suppressor of excitotoxic neuronal death
2010 StandoutNatureNobel
Comprehensive analysis of kinase inhibitor selectivity
2011 Standout
The PI3K Pathway in Human Disease
2017 Standout
Features of Selective Kinase Inhibitors
2005
Discovery and resupply of pharmacologically active plant-derived natural products: A review
2015 Standout
Electrochemical Intramolecular CH Amination: Synthesis of Benzoxazoles and Benzothiazoles
2015
Synthesis and antimosquito properties of 2,6-substituted benzo[d]thiazole and 2,4-substituted benzo[d]thiazole analogues against Anopheles arabiensis
2013
Synthesis and anticancer evaluation of bis(benzimidazoles), bis(benzoxazoles), and benzothiazoles
2006
A comprehensive review in current developments of benzothiazole-based molecules in medicinal chemistry
2014 Standout
Binding Site Detection and Druggability Index from First Principles
2009
An efficient copper(II)-catalyzed synthesis of benzothiazoles through intramolecular coupling-cyclization of N-(2-chlorophenyl)benzothioamides
2010
Electrochemical intramolecular dehydrogenative C–S bond formation for the synthesis of benzothiazoles
2017
Iron Catalysis in Organic Synthesis
2015 Standout
Discovery of Kinase Inhibitors by High-Throughput Docking and Scoring Based on a Transferable Linear Interaction Energy Model
2008
Fluorine and Fluorinated Motifs in the Design and Application of Bioisosteres for Drug Design
2018 Standout
Scaffold Diversity through Intramolecular Cascade Reactions of Solid-Supported Cyclic N-Acyliminium Intermediates
2007 StandoutNobel
A Survey of the Role of Noncovalent Sulfur Interactions in Drug Design
2015
Outstanding challenges in protein–ligand docking and structure‐based virtual screening
2011
Iodobenzene Diacetate–Promoted N–N and N–O Bond Formation for Pyrazolo- and Isoxazolopyrimidine Syntheses
2009
Zirconium(IV) oxide chloride and anhydrous copper(II) sulfate mediated synthesis of 2-substituted benzothiazoles
2006
Palladium-Catalyzed Synthesis of 2-Substituted Benzothiazoles via a C−H Functionalization/Intramolecular C−S Bond Formation Process
2008
The Medicinal Chemist’s Toolbox: An Analysis of Reactions Used in the Pursuit of Drug Candidates
2011 Standout
C−H Activation for the Construction of C−B Bonds
2009 Standout
Discovery of Pyridazinopyridinones as Potent and Selective p38 Mitogen-Activated Protein Kinase Inhibitors
2010
Molecular Docking and Structure-Based Drug Design Strategies
2015 Standout
Stereoelectronic Effects Dictate Molecular Conformation and Biological Function of Heterocyclic Amides
2014
The Origin of Chalcogen-Bonding Interactions
2017 Standout
Stereoselective Enzymatic Synthesis of Heteroatom-Substituted Cyclopropanes
2018 StandoutNobel
Organic and Polymeric Semiconductors Enhanced by Noncovalent Conformational Locks
2017
Current methods for the synthesis of 2-substituted azoles
2004
Single-Junction Organic Solar Cell with over 15% Efficiency Using Fused-Ring Acceptor with Electron-Deficient Core
2019 Standout
Fluorophore Labeling of the Glycine-Rich Loop as a Method of Identifying Inhibitors That Bind to Active and Inactive Kinase Conformations
2010
Aromatic Borylation/Amidation/Oxidation: A Rapid Route to 5-Substituted 3-Amidophenols
2006
Transition-Metal-Catalyzed C−S, C−Se, and C−Te Bond Formation via Cross-Coupling and Atom-Economic Addition Reactions
2011 Standout
Novel Diamidino-Substituted Derivatives of Phenyl Benzothiazolyl and Dibenzothiazolyl Furans and Thiophenes: Synthesis, Antiproliferative and DNA Binding Properties
2010
Synthesis of benzothiazole derivatives and their biological evaluation as anticancer agents
2011
Synthetic Organic Electrochemical Methods Since 2000: On the Verge of a Renaissance
2017 Standout
Comprehensive Survey of Combinatorial Library Synthesis: 2005
2006
Controlling Conformations of Conjugated Polymers and Small Molecules: The Role of Nonbonding Interactions
2013
The Physiology of Phosphoinositides
2007 StandoutNobel
Molecular Docking: Challenges, Advances and its Use in Drug Discovery Perspective
2018 Standout
The “Cyclopropyl Fragment” is a Versatile Player that Frequently Appears in Preclinical/Clinical Drug Molecules
2016
In situclick chemistry: a powerful means for lead discovery
2006 StandoutNobel
The Combinatorial Synthesis of Bicyclic Privileged Structures or Privileged Substructures
2003 Standout
Advances in Synthetic Applications of Hypervalent Iodine Compounds
2016 Standout
Iron-catalyzed synthesis of heterocycles
2014
Applications of Palladium-Catalyzed C–N Cross-Coupling Reactions
2016 Standout
Visible Light Photoredox Catalysis with Transition Metal Complexes: Applications in Organic Synthesis
2013 Standout
Iron phthalocyanine as an efficient and versatile catalyst for N-alkylation of heterocyclic amines with alcohols: one-pot synthesis of 2-substituted benzimidazoles, benzothiazoles and benzoxazoles
2013
Rhodium-Catalyzed C−C Bond Formation via Heteroatom-Directed C−H Bond Activation
2009 Standout
Chalcogen Bonding: An Overview
2018 Standout
Synthesis and biological activity of pyrrole, pyrroline and pyrrolidine derivatives with two aryl groups on adjacent positions
2006 Standout
Principles and Applications of Halogen Bonding in Medicinal Chemistry and Chemical Biology
2012 Standout
A Medicinal Chemist’s Guide to Molecular Interactions
2010 Standout
Novel Cyano- and Amidinobenzothiazole Derivatives: Synthesis, Antitumor Evaluation, and X-ray and Quantitative Structure−Activity Relationship (QSAR) Analysis
2009
Palladium-Catalyzed Ligand-Directed C−H Functionalization Reactions
2010 Standout
Synthesis and antimicrobial activity of novel 2-thiazolylimino-5-arylidene-4-thiazolidinones
2006
The influence of intramolecular sulfur–lone pair interactions on small-molecule drug design and receptor binding
2016
Synopsis of Some Recent Tactical Application of Bioisosteres in Drug Design
2011 Standout
Benzylamines via Iron-Catalyzed Direct Amination of Benzyl Alcohols
2015 StandoutNobel
Energetics of Displacing Water Molecules from Protein Binding Sites: Consequences for Ligand Optimization
2009
Works of Sidney Pitt being referenced
Utilization of a nitrogen–sulfur nonbonding interaction in the design of new 2-aminothiazol-5-yl-pyrimidines as p38α MAP kinase inhibitors
2010
Discovery and initial SAR of imidazoquinoxalines as inhibitors of the Src-family kinase p56Lck
2002
Discovery and initial SAR of 2-amino-5-carboxamidothiazoles as inhibitors of the Src-family kinase p56Lck
2003
Synthesis and SAR of p38α MAP kinase inhibitors based on heterobicyclic scaffolds
2007
Discovery of novel 2-(aminoheteroaryl)-thiazole-5-carboxamides as potent and orally active Src-family kinase p56Lck inhibitors
2004
The identification of novel p38α isoform selective kinase inhibitors having an unprecedented p38α binding mode
2013
Benzothiazole based inhibitors of p38α MAP kinase
2008
Discovery of 2-amino-heteroaryl-benzothiazole-6-anilides as potent p56lck inhibitors
2003
Pyrazolo-pyrimidines: A novel heterocyclic scaffold for potent and selective p38α inhibitors
2008
Molecular design, synthesis, and structure–Activity relationships leading to the potent and selective p56lck inhibitor BMS-243117
2003
5-Cyanopyrimidine Derivatives as a Novel Class of Potent, Selective, and Orally Active Inhibitors of p38α MAP Kinase
2005