Citation Impact
Citing Papers
TRP channel activation by reversible covalent modification
2006 StandoutNobel
Piezo1 and Piezo2 Are Essential Components of Distinct Mechanically Activated Cation Channels
2010 StandoutScienceNobel
A Modular PIP 2 Binding Site as a Determinant of Capsaicin Receptor Sensitivity
2003 StandoutScienceNobel
Radial stretch reveals distinct populations of mechanosensitive mammalian somatosensory neurons
2008 StandoutNobel
Structure of the human TRPM4 ion channel in a lipid nanodisc
2017 StandoutScienceNobel
Cytoplasmic ankyrin repeats of transient receptor potential A1 (TRPA1) dictate sensitivity to thermal and chemical stimuli
2011 StandoutNobel
4-Hydroxynonenal, an endogenous aldehyde, causes pain and neurogenic inflammation through activation of the irritant receptor TRPA1
2007 StandoutNobel
The endocannabinoid nervous system
2001
A-425619 [1-Isoquinolin-5-yl-3-(4-trifluoromethyl-benzyl)-urea], a Novel Transient Receptor Potential Type V1 Receptor Antagonist, Relieves Pathophysiological Pain Associated with Inflammation and Tissue Injury in Rats
2005
Arresting a Transient Receptor Potential (TRP) Channel
2010 StandoutNobel
ANKTM1, a TRP-like Channel Expressed in Nociceptive Neurons, Is Activated by Cold Temperatures
2003 StandoutNobel
New perspectives on enigmatic vanilloid receptors
2000
International Union of Pharmacology. XXVII. Classification of Cannabinoid Receptors
2002 Standout
Structure of the TRPA1 ion channel suggests regulatory mechanisms
2015 StandoutNatureNobel
Characterisation using FLIPR of human vanilloid VR1 receptor pharmacology
2001
High-Affinity Partial Agonists of the Vanilloid Receptor
2003
Noxious compounds activate TRPA1 ion channels through covalent modification of cysteines
2007 StandoutNatureNobel
Molecular mechanisms of nociception
2001 StandoutNatureNobel
Hypothalamic regulation of sleep and circadian rhythms
2005 StandoutNature
Vanilloid receptors on capsaicin‐sensitive sensory nerves mediate relaxation to methanandamide in the rat isolated mesenteric arterial bed and small mesenteric arteries
2000
A possible role of lipoxygenase in the activation of vanilloid receptors by anandamide in the guinea‐pig bronchus
2001
Structure‐activity relationship for the endogenous cannabinoid, anandamide, and certain of its analogues at vanilloid receptors in transfected cells and vas deferens
2001
Highly Selective CB1 Cannabinoid Receptor Ligands and Novel CB1/VR1 Vanilloid Receptor “Hybrid” Ligands
2001
Voltage is a partial activator of rat thermosensitive TRP channels
2007
2-Aminoethoxydiphenyl Borate Is a Common Activator of TRPV1, TRPV2, and TRPV3
2004
Opposite thermosensor in fruitfly and mouse
2003 StandoutNatureNobel
Proton Activation Does Not Alter Antagonist Interaction with the Capsaicin-Binding Pocket of TRPV1
2005
Investigation of the role of TRPV1 receptors in acute and chronic nociceptive processes using gene-deficient mice
2005
Irritant-evoked activation and calcium modulation of the TRPA1 receptor
2020 StandoutNatureNobel
Heat-evoked Activation of TRPV4 Channels in a HEK293 Cell Expression System and in Native Mouse Aorta Endothelial Cells
2002
Functionality of the TRPV subfamily of TRP ion channels: add mechano-TRP and osmo-TRP to the lexicon!
2005
Anandamide acts as a vasodilator of dural blood vessels in vivo by activating TRPV1 receptors
2004
A Bivalent Tarantula Toxin Activates the Capsaicin Receptor, TRPV1, by Targeting the Outer Pore Domain
2010 StandoutNobel
Optical Control of TRPV1 Channels
2013
The vanilloid receptor TRPV1: 10 years from channel cloning to antagonist proof-of-concept
2007 Standout
Biochemistry and pharmacology of endovanilloids
2007
Ganglion-specific splicing of TRPV1 underlies infrared sensation in vampire bats
2011 StandoutNatureNobel
An Alternative Splicing Product of the Murine trpv1 Gene Dominant Negatively Modulates the Activity of TRPV1 Channels
2004
Anandamide activates peripheral nociceptors in normal and arthritic rat knee joints
2001
Characterization of the mouse cold‐menthol receptor TRPM8 and vanilloid receptor type‐1 VR1 using a fluorometric imaging plate reader (FLIPR) assay
2004
The VR1 Antagonist Capsazepine Reverses Mechanical Hyperalgesia in Models of Inflammatory and Neuropathic Pain
2003
TRP channels as cellular sensors
2003 StandoutNature
A-425619 [1-Isoquinolin-5-yl-3-(4-trifluoromethyl-benzyl)-urea], a Novel and Selective Transient Receptor Potential Type V1 Receptor Antagonist, Blocks Channel Activation by Vanilloids, Heat, and Acid
2005
A Cell-Penetrating Scorpion Toxin Enables Mode-Specific Modulation of TRPA1 and Pain
2019 StandoutNobel
TRPV1 structures in distinct conformations reveal activation mechanisms
2013 StandoutNatureNobel
Induction of vanilloid receptor channel activity by protein kinase C
2000 Nature
Molecular basis of infrared detection by snakes
2010 StandoutNatureNobel
Cannabinoid receptors and pain
2001
Bradykinin and nerve growth factor release the capsaicin receptor from PtdIns(4,5)P2-mediated inhibition
2001 StandoutNatureNobel
Temperature-dependent activation of recombinant rat vanilloid VR1 receptors expressed in HEK293 cells by capsaicin and anandamide
2001
Protein kinase C activation potentiates gating of the vanilloid receptor VR1 by capsaicin, protons, heat and anandamide
2001
The TRPV1 receptor and nociception
2006
Structure of the TRPV1 ion channel determined by electron cryo-microscopy
2013 StandoutNatureNobel
Identification of a cold receptor reveals a general role for TRP channels in thermosensation
2002 StandoutNatureNobel
N-(4-Tertiarybutylphenyl)-4-(3-cholorphyridin-2-yl)tetrahydropyrazine -1(2 H)-carbox-amide (BCTC), a Novel, Orally Effective Vanilloid Receptor 1 Antagonist with Analgesic Properties: II. In Vivo Characterization in Rat Models of Inflammatory and Neuropathic Pain
2003
A TRP Channel that Senses Cold Stimuli and Menthol
2002 StandoutNobel
Structural snapshots of TRPV1 reveal mechanism of polymodal functionality
2021 StandoutNobel
Cellular and Molecular Mechanisms of Pain
2009 StandoutNobel
Voltage‐ and time‐dependent properties of the recombinant rat vanilloid receptor (rVR1)
2000
Potentiation of TRPV3 channel function by unsaturated fatty acids
2006
Origin and physiological roles of inflammation
2008 StandoutNature
Noxious Cold Ion Channel TRPA1 Is Activated by Pungent Compounds and Bradykinin
2004 StandoutNobel
Cannabinoid inhibition of the capsaicin‐induced calcium response in rat dorsal root ganglion neurones
2001
Molecular Basis for Species-Specific Sensitivity to “Hot” Chili Peppers
2002 StandoutNobel
The menthol receptor TRPM8 is the principal detector of environmental cold
2007 StandoutNatureNobel
Endovanilloids
2004
AMG 9810 [(E)-3-(4-t-Butylphenyl)-N-(2,3-dihydrobenzo[b][1,4] dioxin-6-yl)acrylamide], a Novel Vanilloid Receptor 1 (TRPV1) Antagonist with Antihyperalgesic Properties
2005
Cannabinoid receptors and their ligands
2002
Overlap between the ligand recognition properties of the anandamide transporter and the VR1 vanilloid receptor: inhibitors of anandamide uptake with negligible capsaicin‐like activity
2000
Anandamide-Evoked Activation of Vanilloid Receptor 1 Contributes to the Development of Bladder Hyperreflexia and Nociceptive Transmission to Spinal Dorsal Horn Neurons in Cystitis
2004
Modulation of the release of endogenous γ-aminobutyric acid by cannabinoids in the guinea pig ileum
2002
Mustard oils and cannabinoids excite sensory nerve fibres through the TRP channel ANKTM1
2004 StandoutNatureNobel
Spider toxins activate the capsaicin receptor to produce inflammatory pain
2006 StandoutNatureNobel
Systematic analysis of genes required for synapse structure and function
2005 StandoutNatureNobel
TRPA1 Mediates the Inflammatory Actions of Environmental Irritants and Proalgesic Agents
2006 StandoutNobel
TRPV3 is a temperature-sensitive vanilloid receptor-like protein
2002 Nature
Cannabinoid receptor ligands: clinical and neuropharmacological considerations, relevant to future drug discovery and development
2000
Discovery of SB-705498: A potent, selective and orally bioavailable TRPV1 antagonist suitable for clinical development
2006
Ethanol elicits and potentiates nociceptor responses via the vanilloid receptor-1
2002
Vanilloid (Capsaicin) Receptors in Health and Disease
2002
Conservation of Functional and Pharmacological Properties in the Distantly Related Temperature Sensors TRPV1 and TRPM8
2005
The Super-Cooling Agent Icilin Reveals a Mechanism of Coincidence Detection by a Temperature-Sensitive TRP Channel
2004 StandoutNobel
Activation of TRPV4 Channels (hVRL-2/mTRP12) by Phorbol Derivatives
2002
The molecular neurobiology of depression
2008 StandoutNature
Pharmacology of Vanilloid Transient Receptor Potential Cation Channels
2009
A role of melanin-concentrating hormone producing neurons in the central regulation of paradoxical sleep
2003
Body weight is regulated by the brain: a link between feeding and emotion
2005
Differential effects of anandamide on acetylcholine release in the guinea‐pig ileum mediated via vanilloid and non‐CB1 cannabinoid receptors
2001
Nociceptors: the sensors of the pain pathway
2010 StandoutNobel
Molecular targets for cannabidiol and its synthetic analogues: effect on vanilloid VR1 receptors and on the cellular uptake and enzymatic hydrolysis of anandamide
2001
Anandamide Excites Central Terminals of Dorsal Root Ganglion Neurons via Vanilloid Receptor-1 Activation
2001
Molecular mechanism of TRPV2 channel modulation by cannabidiol
2019
Δ9-Tetrahydrocannabinol and Cannabinol Activate Capsaicin-Sensitive Sensory Nerves via a CB1 and CB2 Cannabinoid Receptor-Independent Mechanism
2002
Pungent products from garlic activate the sensory ion channel TRPA1
2005 StandoutNobel
Impaired Thermosensation in Mice Lacking TRPV3, a Heat and Camphor Sensor in the Skin
2005 StandoutScienceNobel
An endogenous capsaicin-like substance with high potency at recombinant and native vanilloid VR1 receptors
2002
Turning up the Heat on Pain: TRPV1 Receptors in Pain and Inflammation
2005
Cannabinoid-Induced Presynaptic Inhibition of Glutamatergic EPSCs in Substantia Gelatinosa Neurons of the Rat Spinal Cord
2001
Two amino acid residues determine 2-APB sensitivity of the ion channels TRPV3 and TRPV4
2009 StandoutNobel
Identification and Biological Evaluation of 4-(3-Trifluoromethylpyridin-2-yl)piperazine-1-carboxylic Acid (5-Trifluoromethylpyridin-2-yl)amide, a High Affinity TRPV1 (VR1) Vanilloid Receptor Antagonist
2004
Optische Kontrolle von TRPV1‐Kanälen
2013
TRPA1 mediates formalin-induced pain
2007 StandoutNobel
AN INTRODUCTION TO TRP CHANNELS
2005 Standout
The Vanilloid Receptor: A Molecular Gateway to the Pain Pathway
2001 StandoutNobel
Emerging Targets in Photopharmacology
2016 StandoutNobel
Presynaptic Facilitation of Glutamatergic Synapses to Dopaminergic Neurons of the Rat Substantia Nigra by Endogenous Stimulation of Vanilloid Receptors
2003
Photopharmacology: Beyond Proof of Principle
2014 StandoutNobel
Vanilloid and TRP channels: a family of lipid-gated cation channels
2002
Structural insights into TRPM8 inhibition and desensitization
2019 StandoutScienceNobel
Lys49 myotoxin from the Brazilian lancehead pit viper elicits pain through regulated ATP release
2017 StandoutNobel
Works of S. Nasir being referenced
Identification and characterisation of SB-366791, a potent and selective vanilloid receptor (VR1/TRPV1) antagonist
2003
The distribution of the mRNA and protein products of the melanin‐concentrating hormone (MCH) receptor gene, slc‐1, in the central nervous system of the rat
2000
The endogenous lipid anandamide is a full agonist at the human vanilloid receptor (hVR1)
2000