Citation Impact
Citing Papers
Synthesis, Anti‐B reast Cancer Activity, and Molecular Modeling of Some Benzothiazole and Benzoxazole Derivatives
2013
Synthesis of novel inhibitors of β-glucuronidase based on benzothiazole skeleton and study of their binding affinity by molecular docking
2011
Part 1: Structure–Activity Relationship (SAR) investigations of fused pyrazoles as potent, selective and orally available inhibitors of p38α mitogen-activated protein kinase
2009
The influence of drug-like concepts on decision-making in medicinal chemistry
2007 Standout
Synthesis of potent and selective inhibitors of Candida albicans N-myristoyltransferase based on the benzothiazole structure
2005
Benzothiazoles: Search for anticancer agents
2012
Mammalian phosphoinositide kinases and phosphatases
2009 StandoutNobel
New anticancer active and selective phenylene-bisbenzothiazoles: Synthesis, antiproliferative evaluation and DNA binding
2013
New Substructure Filters for Removal of Pan Assay Interference Compounds (PAINS) from Screening Libraries and for Their Exclusion in Bioassays
2010 Standout
Partial Restoration of Mutant Enzyme Homeostasis in Three Distinct Lysosomal Storage Disease Cell Lines by Altering Calcium Homeostasis
2008
Inhibiting eukaryotic transcription. Which compound to choose? How to evaluate its activity?
2011 Standout
Synthesis of pyrazolo[1,5-a]pyrimidine linked aminobenzothiazole conjugates as potential anticancer agents
2013
Benzothiazoles: How Relevant in Cancer Drug Design Strategy?
2014
PI3Kγ inhibition: towards an 'aspirin of the 21st century'?
2006
Pharmaceutical and medicinal significance of sulfur (SVI)-Containing motifs for drug discovery: A critical review
2018 Standout
Design and synthesis of novel 4-benzothiazole amino quinazolines Dasatinib derivatives as potential anti-tumor agents
2013
SwissParam: A fast force field generation tool for small organic molecules
2011 Standout
Iron catalysed direct alkylation of amines with alcohols
2014 StandoutNobel
4-Thiazolidinone – A biologically active scaffold
2007 Standout
The PtdIns(3,4)P2 phosphatase INPP4A is a suppressor of excitotoxic neuronal death
2010 StandoutNatureNobel
The PI3K Pathway in Human Disease
2017 Standout
Transition‐Metal‐Catalyzed Direct Arylation of (Hetero)Arenes by CH Bond Cleavage
2009 Standout
Solid‐Phase Synthesis of Tetrahydro‐β‐carbolines and Tetrahydroisoquinolines by Stereoselective Intramolecular N‐Carbamyliminium Pictet–Spengler Reactions
2006 StandoutNobel
Features of Selective Kinase Inhibitors
2005
International Union of Pharmacology. XLVII. Nomenclature and Structure-Function Relationships of Voltage-Gated Sodium Channels
2005 Standout
Asymmetric Multicomponent Reactions (AMCRs): The New Frontier
2005 Standout
Synthesis and antimosquito properties of 2,6-substituted benzo[d]thiazole and 2,4-substituted benzo[d]thiazole analogues against Anopheles arabiensis
2013
Synthesis and anticancer evaluation of bis(benzimidazoles), bis(benzoxazoles), and benzothiazoles
2006
A comprehensive review in current developments of benzothiazole-based molecules in medicinal chemistry
2014 Standout
Solid-Phase Synthesis of Pyrroloisoquinolines via the Intramolecular N-Acyliminium Pictet−Spengler Reaction
2005 StandoutNobel
Can a Ketone Be More Reactive than an Aldehyde? Catalytic Asymmetric Synthesis of Substituted Tetrahydrofurans
2018 StandoutNobel
An efficient copper(II)-catalyzed synthesis of benzothiazoles through intramolecular coupling-cyclization of N-(2-chlorophenyl)benzothioamides
2010
Iron Catalysis in Organic Synthesis
2015 Standout
Discovery of Kinase Inhibitors by High-Throughput Docking and Scoring Based on a Transferable Linear Interaction Energy Model
2008
Property-Based Design: Optimization of Drug Absorption and Pharmacokinetics
2001
Iron-catalyzed hydroxylation of β-ketoesters with hydrogen peroxide as oxidant
2008
Fluorine and Fluorinated Motifs in the Design and Application of Bioisosteres for Drug Design
2018 Standout
Scaffold Diversity through Intramolecular Cascade Reactions of Solid-Supported Cyclic N-Acyliminium Intermediates
2007 StandoutNobel
A Survey of the Role of Noncovalent Sulfur Interactions in Drug Design
2015
A Thio-Staudinger Reaction: Thermolysis of a Vinyl Azide in the Presence of t -Butyl Mercaptan
2003
Iodobenzene Diacetate–Promoted N–N and N–O Bond Formation for Pyrazolo- and Isoxazolopyrimidine Syntheses
2009
Zirconium(IV) oxide chloride and anhydrous copper(II) sulfate mediated synthesis of 2-substituted benzothiazoles
2006
C−H Activation for the Construction of C−B Bonds
2009 Standout
1,4-Thiazepines, 1,4-Benzothiazepin-5-ones, and 1,4-Benzothioxepin Orthoamides via Multicomponent Reactions of Isocyanides
2003
Discovery of Imidazo[1,5-a]pyrido[3,2-e]pyrazines as a New Class of Phosphodiesterase 10A Inhibitiors
2010
Practical Methodologies for the Synthesis of Indoles
2006 Standout
Mechanistic Studies on the Cu-Catalyzed Three-Component Reactions of Sulfonyl Azides, 1-Alkynes and Amines, Alcohols, or Water: Dichotomy via a Common Pathway
2008 StandoutNobel
Recent Developments in Isocyanide Based Multicomponent Reactions in Applied Chemistry
2005 Standout
The Origin of Chalcogen-Bonding Interactions
2017 Standout
Stereoselective Enzymatic Synthesis of Heteroatom-Substituted Cyclopropanes
2018 StandoutNobel
Efficient Long-Range Stereochemical Communication and Cooperative Effects in Self-Assembled Fe4L6 Cages
2012 StandoutNobel
Metabolism-guided drug design
2012
Discovery of Novel and Cardioselective Diltiazem-like Calcium Channel Blockers via Virtual Screening
2008
Aromatic Borylation/Amidation/Oxidation: A Rapid Route to 5-Substituted 3-Amidophenols
2006
Transition-Metal-Catalyzed C−S, C−Se, and C−Te Bond Formation via Cross-Coupling and Atom-Economic Addition Reactions
2011 Standout
Novel Diamidino-Substituted Derivatives of Phenyl Benzothiazolyl and Dibenzothiazolyl Furans and Thiophenes: Synthesis, Antiproliferative and DNA Binding Properties
2010
Synthesis of benzothiazole derivatives and their biological evaluation as anticancer agents
2011
Adapting Proteostasis for Disease Intervention
2008 StandoutScience
Detection of Calcium Transients inDrosophilaMushroom Body Neurons with Camgaroo Reporters
2003 StandoutNobel
Comprehensive Survey of Combinatorial Library Synthesis: 2005
2006
Enantioselective Copper-Catalyzed Alkynylation of Benzopyranyl Oxocarbenium Ions
2015
The Physiology of Phosphoinositides
2007 StandoutNobel
The “Cyclopropyl Fragment” is a Versatile Player that Frequently Appears in Preclinical/Clinical Drug Molecules
2016
Controlling the Transmission of Stereochemical Information through Space in Terphenyl-Edged Fe4L6 Cages
2011
The Combinatorial Synthesis of Bicyclic Privileged Structures or Privileged Substructures
2003 Standout
Enzyme Immobilization: The Quest for Optimum Performance
2007 Standout
Advances in Synthetic Applications of Hypervalent Iodine Compounds
2016 Standout
Gold(I)-Catalyzed Benz[c]azepin-4-ol Synthesis by Intermolecular [5 + 2] Cycloaddition
2013
Microwave assisted organic synthesis—a review
2001 Standout
Iron-catalyzed synthesis of heterocycles
2014
Applications of Palladium-Catalyzed C–N Cross-Coupling Reactions
2016 Standout
Aromatic Trifluoromethylation with Metal Complexes
2011 Standout
A Dual Lewis Base Activation Strategy for Enantioselective Carbene-Catalyzed Annulations
2013
MOLECULAR DETERMINANTS OF DRUG BINDING AND ACTION ON L-TYPE CALCIUM CHANNELS
1997
Asymmetric Catalysis via Cyclic, Aliphatic Oxocarbenium Ions
2017 StandoutNobel
MetaSite: Understanding Metabolism in Human Cytochromes from the Perspective of the Chemist
2005
Iron phthalocyanine as an efficient and versatile catalyst for N-alkylation of heterocyclic amines with alcohols: one-pot synthesis of 2-substituted benzimidazoles, benzothiazoles and benzoxazoles
2013
Kann ein Keton reaktiver als ein Aldehyd sein? Katalytische asymmetrische Synthese von substituierten Tetrahydrofuranen
2018 StandoutNobel
Fluoro organics: Facile syntheses of novel 2- or 4-trifluoromethyl-1H-arylo-1,5-diazepines, oxazepines, thiazepines, 2 -(1,1,1-trifluoroacetonyl)imidazoles, oxazoles and thiazoles
1997
Solar Synthesis: Prospects in Visible Light Photocatalysis
2014 StandoutScience
Novel Cyano- and Amidinobenzothiazole Derivatives: Synthesis, Antitumor Evaluation, and X-ray and Quantitative Structure−Activity Relationship (QSAR) Analysis
2009
Synthesis and antimicrobial evaluation of some new fluorinated spiro[[1,5] -benzothiazepin-2,3′[3′H]-indol]-2′(1′H)-ones
1998
Metal–Organic Frameworks for Heterogeneous Basic Catalysis
2017 Standout
Benzylamines via Iron-Catalyzed Direct Amination of Benzyl Alcohols
2015 StandoutNobel
Microbial/enzymatic synthesis of chiral intermediates for pharmaceuticals
2002
Gold(I)-Catalyzed Activation of Alkynes for the Construction of Molecular Complexity
2015 Standout
Fluorination in Medicinal Chemistry: Methods, Strategies, and Recent Developments
2008 Standout
Works of Robert V. Moquin being referenced
Benzazepinone calcium channel blockers. 4. Structure-activity overview and intracellular binding site
1992
Identification of 2-amino-5-(thioaryl)thiazoles as inhibitors of nerve growth factor receptor TrkA
2007
Discovery and initial SAR of 2-amino-5-carboxamidothiazoles as inhibitors of the Src-family kinase p56Lck
2003
Synthesis, initial SAR and biological evaluation of 1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridin-4-amine derived inhibitors of IκB kinase
2009
Benzazepinone calcium channel blockers. 2. Structure activity and drug metabolism studies leading to potent antihypertensive agents. Comparison with benzothiazepinones
1992
Discovery of 2-amino-heteroaryl-benzothiazole-6-anilides as potent p56lck inhibitors
2003
Pyrazolo-pyrimidines: A novel heterocyclic scaffold for potent and selective p38α inhibitors
2008
Molecular design, synthesis, and structure–Activity relationships leading to the potent and selective p56lck inhibitor BMS-243117
2003
Synthesis and SAR of novel imidazoquinoxaline-Based Lck inhibitors: improvement of cell potency
2002
Synthesis of benzazepinone and 3-methylbenzothiazepinone analogs of diltiazem
1990
Synthesis of imidazo[1,5-a]quinoxalin-4(5H)-one template via a novel intramolecular cyclization process
2001
Synthesis and photochemistry of heterocyclic norbornenyl ketones
1987