Citation Impact
Citing Papers
Topological control of cytokine receptor signaling induces differential effects in hematopoiesis
2019 StandoutScienceNobel
Palladium‐Catalyzed Cross‐Coupling Reactions in Total Synthesis
2005 Standout
Microwave chemistry for inorganic nanomaterials synthesis
2010 Standout
Biased ligands at G-protein-coupled receptors: promise and progress
2014
Structure of the µ-opioid receptor–Gi protein complex
2018 NatureNobel
Trends in GPCR drug discovery: new agents, targets and indications
2017 Standout
Insights into subtype selectivity of opioid agonists by ligand-based and structure-based methods
2010
Psychedelics
2016 Standout
Structure-based discovery of opioid analgesics with reduced side effects
2016 NatureNobel
How Ligands Illuminate GPCR Molecular Pharmacology
2017
Molecular Dynamics Simulation for All
2018 Standout
Pyrrolidinyl‐Spirooxindole Natural Products as Inspirations for the Development of Potential Therapeutic Agents
2007 Standout
Controlled microwave heating in modern organic synthesis: highlights from the 2004–2008 literature
2009
Recent developments in biased agonism
2013 Nobel
Covalent organic frameworks (COFs): from design to applications
2012 Standout
The impact of microwave synthesis on drug discovery
2005
Recent updates on GPCR biased agonism
2016
The use of spirocyclic scaffolds in drug discovery
2014 Standout
Functional selectivity of GPCR signaling in animals
2013
Peptide therapeutics: current status and future directions
2014 Standout
A randomized, phase 2 study investigating TRV130, a biased ligand of the μ-opioid receptor, for the intravenous treatment of acute pain
2015
Recent Advances in Ligand-Based Drug Design: Relevance and Utility of the Conformationally Sampled Pharmacophore Approach
2010
Allosteric and Biased G Protein-Coupled Receptor Signaling Regulation: Potentials for New Therapeutics
2014
Multicomponent reactions for the synthesis of pyrroles
2010 Standout
Iron Catalysis in Organic Synthesis
2015 Standout
Further exploring r metrics for validation of QSPR models
2011 Standout
RECENT ADVANCES IN THE SYNTHESIS OF PYRROLES
2001
Biased ligand quantification in drug discovery: from theory to high throughput screening to identify new biased μ opioid receptor agonists
2016
Construction of a Virtual Opioid Bioprofile: A Data-Driven QSAR Modeling Study to Identify New Analgesic Opioids
2021
The Medicinal Chemist’s Toolbox: An Analysis of Reactions Used in the Pursuit of Drug Candidates
2011 Standout
Recent advances in the synthesis of pyrroles by multicomponent reactions
2014 Standout
Molecular Docking and Structure-Based Drug Design Strategies
2015 Standout
Optimization of the Additive CHARMM All-Atom Protein Force Field Targeting Improved Sampling of the Backbone ϕ, ψ and Side-Chain χ1 and χ2 Dihedral Angles
2012 Standout
Synthesis, Anticonvulsant Activity, and Structure−Activity Relationships of Sodium Channel Blocking 3-Aminopyrroles
1998
Structure-inspired design of β-arrestin-biased ligands for aminergic GPCRs
2017
Computational design of environmental sensors for the potent opioid fentanyl
2017 StandoutNobel
PubChem 2023 update
2022 Standout
Microwave-Assisted Synthesis in Water as Solvent
2007 Standout
Green chemistry by nano-catalysis
2010 Standout
A Review on the Use of Sodium Triacetoxyborohydride in the Reductive Amination of Ketones and Aldehydes
2006
Comprehensive Survey of Combinatorial Library Synthesis: 2004
2005
Thioamides as Useful Synthons in the Synthesis of Heterocycles
2002 Standout
Quantitative Conformationally Sampled Pharmacophore for δ Opioid Ligands: Reevaluation of Hydrophobic Moieties Essential for Biological Activity
2007
Three-Component Coupling Synthesis of Diversely Substituted N-Aryl Pyrroles Catalyzed by Iron(III) Chloride
2013
Gold-Catalyzed Carbon−Heteroatom Bond-Forming Reactions
2011 Standout
Synthesis and biological activity of pyrrole, pyrroline and pyrrolidine derivatives with two aryl groups on adjacent positions
2006 Standout
Pyrrole: a resourceful small molecule in key medicinal hetero-aromatics
2015 Standout
A Review on the Use of Sodium Triacetoxyborohydride in the Reductive Amination of Ketones and Aldehydes
2007
Gold(I)-Catalyzed Cyclization of β-Allenylhydrazones: An Efficient Synthesis of MultisubstitutedN-Aminopyrroles
2010
Works of Philip Pitis being referenced
Parallel methods for the preparation and SAR exploration of N-ethyl-4-[(8-alkyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-aryl-methyl]-benzamides, powerful mu and delta opioid agonists
2004
N , N -Dialkyl-4-[(8-azabicyclo[3.2.1]-oct-3-ylidene)phenylmethyl]benzamides, potent, selective δ opioid agonists
2004
The Novel, Orally Active, Delta Opioid RWJ-394674 Is Biotransformed to the Potent Mu Opioid RWJ-413216
2006
A G Protein-Biased Ligand at the μ-Opioid Receptor Is Potently Analgesic with Reduced Gastrointestinal and Respiratory Dysfunction Compared with Morphine
2013
Aroyl(aminoacyl)pyrroles, a New Class of Anticonvulsant Agents
1997
Structure–Activity Relationships and Discovery of a G Protein Biased μ Opioid Receptor Ligand, [(3-Methoxythiophen-2-yl)methyl]({2-[(9R)-9-(pyridin-2-yl)-6-oxaspiro-[4.5]decan-9-yl]ethyl})amine (TRV130), for the Treatment of Acute Severe Pain
2013