Citation Impact
Citing Papers
Effect of secretin on release of heterogeneous forms of gastrin.
1975 StandoutNobel
Preclinical Development and First-in-Human Study of KA2507, a Selective and Potent Inhibitor of Histone Deacetylase 6, for Patients with Refractory Solid Tumors
2021
Diversity oriented clicking delivers β-substituted alkenyl sulfonyl fluorides as covalent human neutrophil elastase inhibitors
2022 StandoutNobel
Expansive discovery of chemically diverse structured macrocyclic oligoamides
2024 StandoutScienceNobel
Metabolic and hypoxic adaptation to anti‐angiogenic therapy: a target for induced essentiality
2015
Microenvironmental regulation of tumour angiogenesis
2017
The EGLN-HIF O 2 -Sensing System: Multiple Inputs and Feedbacks
2017 StandoutNobel
Pharmacology of AMPA/Kainate Receptor Ligands and Their Therapeutic Potential in Neurological and Psychiatric Disorders
2000
The ever-expanding role of HIF in tumour and stromal biology
2016
Methyl 2‐[bis(acetyl)ethenyl]aminopropenoate in the synthesis of heterocyclic systems
1997
Ampakines and the threefold path to cognitive enhancement
2006
Glutamate receptor ion channels
2005 Standout
Glutamate Receptor Ion Channels: Structure, Regulation, and Function
2010 Standout
Persistent kallikrein 5 activation induces atopic dermatitis-like skin architecture independent of PAR2 activity
2017 StandoutNobel
Failure to limit quantities of benzodiazepine hypnotic drugs for outpatients: Placing the elderly at risk
1990
Involvement of Cholecystokinin/Gastrin‐Related Peptides and their Receptors in Clinical Gastrointestinal Disorders
2002
Drugs and Falls in Older People: A Systematic Review and Meta‐analysis: I. Psychotropic Drugs
1999 Standout
mTORC2 Promotes Tumorigenesis via Lipid Synthesis
2017
Marine natural products
1990 Standout
Myeloid-derived suppressor cells in the era of increasing myeloid cell diversity
2021 Standout
The multifaceted roles of fatty acid synthesis in cancer
2016
Hypoxia-Inducible Factors: Master Regulators of Cancer Progression
2016 StandoutNobel
Hepatocellular carcinoma
2021 Standout
Characteristics of the Cholecystokinin-Induced Depolarization of Pacemaking Activity in Cultured Interstitial Cells of Cajal from Murine Small Intestine
2013 Standout
Cholecystokinin antagonists: Pharmacological and therapeutic potential
2003
Acetylcholinesterase: ‘classical’ and ‘non-classical’ functions and pharmacology
2005
Natural products to drugs: natural product-derived compounds in clinical trials
2008 Standout
Tissue Kallikrein Inhibitors Based on the Sunflower Trypsin Inhibitor Scaffold – A Potential Therapeutic Intervention for Skin Diseases
2016 StandoutNobel
Memory enhancement: the search for mechanism-based drugs
2002
The evolving tumor microenvironment: From cancer initiation to metastatic outgrowth
2023 Standout
Coumarinic derivatives as mechanism-based inhibitors of α-chymotrypsin and human leukocyte elastase
2000
Natural products to drugs: natural product derived compounds in clinical trials
2005
Transition‐Metal‐Catalyzed Direct Arylation of (Hetero)Arenes by CH Bond Cleavage
2009 Standout
Dialdehyde sesquiterpenes and other terpenoids as vanilloids
1998
Discovery and resupply of pharmacologically active plant-derived natural products: A review
2015 Standout
VEGF in Signaling and Disease: Beyond Discovery and Development
2019 Standout
Metabolic adaptation of cancer and immune cells mediated by hypoxia-inducible factors
2018 StandoutNobel
Rigid‐Strut‐Containing Crown Ethers and [2]Catenanes for Incorporation into Metal–Organic Frameworks
2009 StandoutNobel
Iron Catalysis in Organic Synthesis
2015 Standout
Synthesis of Organochalcogen Propargyl Aryl Ethers and Their Application in the Electrophilic Cyclization Reaction: An Efficient Preparation of 3-Halo-4-Chalcogen-2H-Benzopyrans
2009
Over One Hundred Peptide-Activated G Protein-Coupled Receptors Recognize Ligands with Turn Structure
2005
Solid-Phase Intramolecular N-Acyliminium Pictet−Spengler Reactions as Crossroads to Scaffold Diversity
2004 StandoutNobel
Synthesis, Characterization, Cytotoxic Activities, and DNA-Binding Studies of Ternary Copper(II) Complexes with New Coumarin Derivatives
2010
The metaRbolomics Toolbox in Bioconductor and beyond
2019
Coordinating Radiometals of Copper, Gallium, Indium, Yttrium, and Zirconium for PET and SPECT Imaging of Disease
2010 Standout
Iron(III) Chloride/Diorganyl Diselenides‐Promoted Regioselective Cyclization of Alkynyl Aryl Ketones: Synthesis of 3‐Organoselenyl Chromenones under Ambient Atmosphere
2011
Steric and Dynamic Parameters Influencing In Situ Cycloadditions to Form Triazole Inhibitors with Crystalline Acetylcholinesterase
2016 StandoutNobel
Synthesis of Heterocycles via Electrophilic Cyclization of Alkynes Containing Heteroatom
2011 Standout
A novel strapped porphyrin receptor for molecular recognition
2003
Palladium-Catalyzed Arylation of Fluoroalkylamines
2015
Iron-catalyzed atom transfer radical polymerization
2014
Fluorine and Fluorinated Motifs in the Design and Application of Bioisosteres for Drug Design
2018 Standout
Synthesis of novel 1,2,4-thiadiazinane 1,1-dioxidesviathree component SuFEx type reaction
2018
Efficient and highly regioselective direct C-2 arylation of azoles, including free (NH)-imidazole, -benzimidazole and -indole, with aryl halides
2006
Accessing Elaborated 2,1-Borazaronaphthalene Cores Using Photoredox/Nickel Dual-Catalytic Functionalization
2016
Oxidative Coupling between Two Hydrocarbons: An Update of Recent C–H Functionalizations
2015 Standout
Poly(ethylene oxide)-based electrolytes for lithium-ion batteries
2015 Standout
1-Oxo-1-fluoro-1,2,4-benzothiadiazines—A new type of cyclic sulfonimidoyl fluorides
2014
π-Stacking Interactions and CH···X (X = O, Aryl) Hydrogen Bonding as Directing Features of the Supramolecular Self-Association in 3-Carboxy and 3-Amido Coumarin Derivatives
2002
SuFEx Chemistry of Thionyl Tetrafluoride (SOF4) with Organolithium Nucleophiles: Synthesis of Sulfonimidoyl Fluorides, Sulfoximines, Sulfonimidamides, and Sulfonimidates
2018 StandoutNobel
Phosphine Organocatalysis
2018 Standout
Environmentally Friendly Iron-Catalyzed Cascade Synthesis of 1,2,4-Benzothiadiazine 1,1-Dioxide and Quinazolinone Derivatives
2009
Toward the First Class of Suicide Inhibitors of Kallikreins Involved in Skin Diseases
2014
Alkyl 2‐(2‐benzoyl‐2‐ethoxycarbonyl‐1‐ethenyl)amino‐3‐dimethylaminopropenoates in the synthesis of heterocyclic systems
1997
Vanilloid (Capsaicin) Receptors and Mechanisms
1999 Standout
The synthesis and transformations of substituted 2-hydroxy-3-dimethylaminopropenoates. The preparation of condensed 3-hydroxypyran-2-ones
1998
The effects of somatostatin and metiamide on tachyphylaxis of pentagastrin stimulated gastric acid and pepsin secretion in the conscious cat.
1977 StandoutNobel
Deciphering the Mechanism of Carbonic Anhydrase Inhibition with Coumarins and Thiocoumarins
2009
Human TKTL1 implies greater neurogenesis in frontal neocortex of modern humans than Neanderthals
2022 StandoutScienceNobel
Combination therapy in combating cancer
2017 Standout
The synthesis of methyl 2‐(benzyloxycarbonyl)amino‐3‐dimethylaminopropenoate. The synthesis of trisubstituted pyrroles, 3‐amino‐2H‐pyran‐2‐ones, fused 2H‐pyran‐2‐ones and 4H‐pyridin‐4‐ones
1999
6-Substituted 2-Oxo-2H-1-benzopyran-3-carboxylic Acid as a Core Structure for Specific Inhibitors of Human Leukocyte Elastase
1999
The Combinatorial Synthesis of Bicyclic Privileged Structures or Privileged Substructures
2003 Standout
TRIPHENYPHOSPHINE-MEDIATED EFFICIENT SYNTHESIS OF FUNCTIONALIZED 2-OXO-2H-CHROMENES
2004
2,5-Diketopiperazines: Synthesis, Reactions, Medicinal Chemistry, and Bioactive Natural Products
2012
Iron-catalyzed synthesis of heterocycles
2014
Applications of Palladium-Catalyzed C–N Cross-Coupling Reactions
2016 Standout
Photoredox Catalysis in Organic Chemistry
2016 Standout
Pharmaceuticals that contain polycyclic hydrocarbon scaffolds
2015
Advances in Copper Complexes as Anticancer Agents
2013 Standout
Natural Products as Sources of New Drugs from 1981 to 2014
2016 Standout
The Traditional Medicine and Modern Medicine from Natural Products
2016 Standout
Visible‐Light Photocatalysis: Does It Make a Difference in Organic Synthesis?
2018 Standout
β-Turned Dipeptoids as Potent and Selective CCK1 Receptor Antagonists
2000
Chemistry and Biology Of Multicomponent Reactions
2012 Standout
Regioselective Ortho Olefination of Aryl Sulfonamide via Rhodium-Catalyzed Direct C–H Bond Activation
2014
Rhodium-Catalyzed C−C Bond Formation via Heteroatom-Directed C−H Bond Activation
2009 Standout
Iron-catalyzed oxidative synthesis of N-heterocycles from primary alcohols
2014
Synthesis and biological activity of pyrrole, pyrroline and pyrrolidine derivatives with two aryl groups on adjacent positions
2006 Standout
Irreversible Inhibitors of Serine, Cysteine, and Threonine Proteases
2002 Standout
Synthesis of Heterocycles from Alkyl 3-(Dimethylamino)propenoates and Related Enaminones
2004 Standout
Crystal Engineering Using the Versatility of 2,5-Dichloro-3,6-dihydroxy-1,4-benzoquinone with Organic and Metal Complex Partners
2003 StandoutNobel
MetaboAnalyst 5.0: narrowing the gap between raw spectra and functional insights
2021 Standout
Multiple Binding Modes of Inhibitors to Carbonic Anhydrases: How to Design Specific Drugs Targeting 15 Different Isoforms?
2012 Standout
Peptide Receptors as Molecular Targets for Cancer Diagnosis and Therapy
2003
Works of Pascal De Tullio being referenced
Synthesis and pharmacological activity of N-(2,2-dimethyl-3,4-dihydro-2H-1-benzopyran-4-yl)-4H-1,2,4-benzothiadiazine-3-carboxamides 1,1-dioxides on rat uterus, rat aorta and rat pancreatic β-cells
2012
Therapeutic and chemical developments of cholecystokinin receptor ligands
2000
New Trends in the Design of Drugs Against Alzheimer's Disease
2004
Blocking Lipid Synthesis Overcomes Tumor Regrowth and Metastasis after Antiangiogenic Therapy Withdrawal
2014
Evaluation of Long-Term Triazolam Use in an Ambulatory Veterans Administration Medical Center Population
1989
PepsNMR for 1H NMR metabolomic data pre-processing
2018
Effect of Head-to-Head Addition in Vinyl Acetate Controlled Radical Polymerization: Why Is Co(acac)2-Mediated Polymerization so Much Better?
2013
Effect onKATPChannel Activation Properties and Tissue Selectivity of the Nature of the Substituent in the 7- and the 3-Position of 4H-1,2,4-Benzothiadiazine 1,1-Dioxides
2005
Recent Advances in the Chemistry of Cholecystokinin Receptor Ligands (Agonists and Antagonists)
1999
Design, Synthesis, and Pharmacology of Novel 7-Substituted 3,4-Dihydro-2H-1,2,4-benzothiadiazine 1,1-Dioxides as Positive Allosteric Modulators of AMPA Receptors
2007
1,4,2-Benzo/pyridodithiazine 1,1-Dioxides Structurally Related to the ATP-Sensitive Potassium Channel Openers 1,2,4-Benzo/pyridothiadiazine 1,1-Dioxides Exert a Myorelaxant Activity Linked to a Distinct Mechanism of Action
2013
Selective pharmacological inhibitors of HDAC6 reveal biochemical activity but functional tolerance in cancer models
2019
Recent Advances in Inducible Cyclooxygenase (COX-2) Inhibition.
2000
Synthetic studies on biologically active natural compounds. Part III. Stereospecific transformation of uvidin A into (−)-cinnamosmolide.
1991
Esters and Amides of 6-(Chloromethyl)-2-oxo-2H-1-benzopyran-3-carboxylic Acid as Inhibitors of α-Chymotrypsin: Significance of the “Aromatic” Nature of the Novel Ester-Type Coumarin for Strong Inhibitory Activity
1996
Toward Tissue-Selective Pancreatic B-Cells KATP Channel Openers Belonging to 3-Alkylamino-7-halo-4H-1,2,4-benzothiadiazine 1,1-Dioxides
2003
Hydroxylated Analogues of ATP-Sensitive Potassium Channel Openers Belonging to the Group of 6- and/or 7-Substituted 3-Isopropylamino-4H-1,2,4-benzothiadiazine 1,1-Dioxides: Toward an Improvement in Sulfonylurea Receptor 1 Selectivity and Metabolism Stability
2011
Development of Thiophenic Analogues of Benzothiadiazine Dioxides as New Powerful Potentiators of 2-Amino-3-(3-hydroxy-5-methylisoxazol-4-yl)propionic Acid (AMPA) Receptors
2013
New Fluorinated 1,2,4-Benzothiadiazine 1,1-Dioxides: Discovery of an Orally Active Cognitive Enhancer Acting through Potentiation of the 2-Amino-3-(3-hydroxy-5-methylisoxazol-4-yl)propionic Acid Receptors
2010
4H-1,2,4-Pyridothiadiazine 1,1-Dioxides and 2,3-Dihydro-4H-1,2,4-pyridothiadiazine 1,1-Dioxides Chemically Related to Diazoxide and Cyclothiazide as Powerful Positive Allosteric Modulators of (R/S)-2-Amino-3-(3-hydroxy-5-methylisoxazol-4-yl)propionic Acid Receptors: Design, Synthesis, Pharmacology, and Structure−Activity Relationships
1998
Design, Synthesis, and Pharmacological Evaluation ofR/S-3,4-Dihydro-2,2-dimethyl- 6-halo-4-(phenylaminocarbonylamino)-2H-1-benzopyrans: Toward Tissue-Selective Pancreatic β-CellKATPChannel Openers Structurally Related to (±)-Cromakalim
2006
New substituted aryl esters and aryl amides of 3,4-dihydro-2H-1,2,4-benzothiadiazine 1,1-dioxides as positive allosteric modulators of AMPA receptors
2011
3-Alkylamino-4H-1,2,4-benzothiadiazine 1,1-Dioxides as ATP-Sensitive Potassium Channel Openers: Effect of 6,7-Disubstitution on Potency and Tissue Selectivity
2005