Citation Impact
Citing Papers
SuFEx-enabled, agnostic discovery of covalent inhibitors of human neutrophil elastase
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Expansive discovery of chemically diverse structured macrocyclic oligoamides
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A Structure‐Guided Switch in the Regioselectivity of a Tryptophan Halogenase
2016
Copper-Catalyzed Enantioselective Michael Additions: Recent Progress with New Phosphorus Ligands
1998
Recent advances in the catalytic asymmetric synthesis of β-amino acids
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Late-stage C–H functionalization of complex alkaloids and drug molecules via intermolecular rhodium-carbenoid insertion
2015
Azobenzene as photoresponsive conformational switch in cyclic peptides*
2005
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2006
The Agrobacterium VirB/VirD4 T4SS: Mechanism and Architecture Defined Through In Vivo Mutagenesis and Chimeric Systems
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The road to fully programmable protein catalysis
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A new chemical probe for the detection of the cancer-linked galectin-3
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The World of β‐ and γ‐Peptides Comprised of Homologated Proteinogenic Amino Acids and Other Components
2004
Phosphoramidites: Privileged Ligands in Asymmetric Catalysis
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A New Chemical Probe for Proteomics of Carbohydrate‐Binding Proteins
2004
Direct enantio- and diastereoselective Mannich reactions of malonate and β-keto esters with N-Boc and N-Cbz aldimines catalysed by a bifunctional cinchonine derivative
2006
Dynamic Kinetic Resolution in the Asymmetric Synthesis of β‐Amino Acids by Organocatalytic Reduction of Enamines with Trichlorosilane
2008
Biosynthetic Manipulation of Tryptophan in Bacteria: Pathways and Mechanisms
2015
Highly Efficient Synthesis of Heterocyclic and Alicyclic β2‐Amino Acid Derivatives by Catalytic Asymmetric Hydrogenation
2013
Cryo-EM structure of a type IV secretion system
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Organic Azides: An Exploding Diversity of a Unique Class of Compounds
2005 Standout
In the Golden Age of Organocatalysis
2004 Standout
β2‐amino acids—syntheses, occurrence in natural products, and components of β‐peptides1,2
2004
Enantioselective synthesis of β2-amino acids using rhodium-catalyzed hydrogenation
2006 StandoutNobel
SuFEx Click Chemistry Enabled Late-Stage Drug Functionalization
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The Direct Catalytic Asymmetric Three-Component Mannich Reaction
2000 StandoutNobel
NaNO2–Ceric ammonium nitrate mediated conversion of acrylic esters and Baylis–Hillman derived acrylic esters into corresponding β-nitro acrylic esters
2003
Rhodium-Catalyzed Enantioselective Hydrogenation of β-Phthalimide Acrylates to Synthesis of β2-Amino Acids
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Ir-Catalyzed Allylic Amination/Ring-Closing Metathesis: A New Route to Enantioselective Synthesis of Cyclic β-Amino Alcohol Derivatives
2007
Copper-catalysed asymmetric conjugate addition of organometallic reagents to enones using S,O-ligands with a xylofuranose backbone
2000
Broad-Spectrum Kinase Profiling in Live Cells with Lysine-Targeted Sulfonyl Fluoride Probes
2017
Activation of H2O2 by Chiral Confined Brønsted Acids: A Highly Enantioselective Catalytic Sulfoxidation
2012 StandoutNobel
Copper(I) Thiolate Catalysts in Asymmetric Conjugate Addition Reactions
2004
Enantioselective Michael Reaction of Malonates to Nitroolefins Catalyzed by Bifunctional Organocatalysts
2003 Standout
Highly Diastereoselective Asymmetric Mannich Reactions of 1,3-Dicarbonyls with Acyl Imines
2006
A Convenient Enantioselective Synthesis of (S)-α-Trifluoromethylisoserine
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Late-Stage Diversification of Biologically Active Molecules via Chemoenzymatic C–H Functionalization
2016
A General Approach to the Synthesis of β2‐Amino Acid Derivatives via Highly Efficient Catalytic Asymmetric Hydrogenation of α‐Aminomethylacrylates
2010
Structure of the VirB4 ATPase, alone and bound to the core complex of a type IV secretion system
2012
Peptidic Amidomonophosphane Ligand for Copper‐Catalyzed Asymmetric Conjugate Addition of Diorganozincs to Cycloalkenones
2007
Direct Catalytic Enantioselective Mannich Reactions: Synthesis of Protected anti-α,β-Diamino Acids
2007
Bioorthogonal Chemistry: Applications in Activity-Based Protein Profiling
2011
Type IV secretion systems: Advances in structure, function, and activation
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One-pot multi-substrate enantioselective conjugate addition of diethylzinc to nitroalkenes
2002 StandoutNobel
Convenient Catalytic, Enantioselective Conjugate Reduction of Nitroalkenes Using CuF2
2004
Asymmetric conjugate addition of diethyl zinc to enones with chiral phosphine ligands
1997
Catalytic Enantioselective Conjugate Addition of Carbamates
2004
Acceleration of the conjugate addition of diethyl zinc to enones by either Cu(OTf)2 or trivalent phosphorus ligands
1997
Structural Biology of Bacterial Type IV Secretion Systems
2015
Chiroptical Molecular Switches
2000 StandoutNobel
Enantioselective Synthesis of β2-Amino Acids via Rh-Catalyzed Asymmetric Hydrogenation with BoPhoz-Type Ligands: Important Influence of an N−H Proton in the Ligand on the Enantioselectivity
2008
1,4-Addition of Diorganozincs to α,β-Unsaturated Ketones Catalyzed by a Copper(I)-Sulfonamide Combined System
2000 StandoutNobel
Catalytic Asymmetric Allylic and Homoallylic Diamination of Terminal Olefins via Formal C−H Activation
2008
Catalytic Enantioselective Synthesis of Prostaglandin E1 Methyl Ester Using a Tandem 1,4-Addition-Aldol Reaction to a Cyclopenten-3,5-dione Monoacetal
2001 StandoutNobel
Development and Applications of Disulfonimides in Enantioselective Organocatalysis
2015 StandoutNobel
Stereoselective Enzymatic Synthesis of Heteroatom-Substituted Cyclopropanes
2018 StandoutNobel
Synthesis and Application of Chiral Phosphorus Ligands Derived from TADDOL for the Asymmetric Conjugate Addition of Diethyl Zinc to Enones
2000
Catalyst Self-Adaptation in Conjugate Addition to Nitroalkenes and Nitroacrylates: Instant Chirality Control in Diphenylmethane-Based Phosphoramidite Ligands
2008
β-Peptides: From Structure to Function
2001 Standout
Asymmetric Mannich Reactions of β-Keto Esters with Acyl Imines Catalyzed by Cinchona Alkaloids
2005
Highly Enantioselective Copper-Catalyzed Conjugate Addition of Diethylzinc to Nitroalkenes
2004
ChemInform Abstract: Conjugate Addition of Organometallic Reagents
2000
Synthesis and Applications of β-Aminocarboxylic Acids Containing a Cyclopropane Ring
2003
Folding of a donor–acceptor polyrotaxane by using noncovalent bonding interactions
2008 StandoutNobel
Stereoselective synthesis of β2-amino acids by Michael addition of diorgano zinc reagents to nitro acrylates
2003
Asymmetric Conjugate Addition Reactions of Meldrum's Acid Derived Acceptors Employing Chiral Phosphoramidite Ligands
2003
Copper-catalysed asymmetric conjugate addition of organometallic reagents to linear enones using thiourethane ligands
1999
Unlocking Reactivity of TrpB: A General Biocatalytic Platform for Synthesis of Tryptophan Analogues
2017 StandoutNobel
Hydrazino Peptides as Foldamers: An Extension of the β-Peptide Concept
2000
Copper-Catalysed Asymmetric Conjugate Addition of Organometallic Reagents to Linear Enones
2000
Recent Advances in the Catalytic Asymmetric Synthesis of β2‐ and β2,2‐Amino Acids
2019
De novo design of covalently constrained mesosize protein scaffolds with unique tertiary structures
2017 StandoutNobel
Recent Advances in Stereoselective Synthesis and Application of β-Amino Acids
2009
Enantioselective Copper-Catalyzed Conjugate Addition of Dialkyl Zinc to Nitro-Olefins
2000
Highly Enantioselective Conjugate Addition of Dialkylzinc Reagents to Acyclic Nitroalkenes: A Catalytic Route to β2-Amino Acids, Aldehydes, and Alcohols
2003 StandoutNobel
Reversible Photocontrol of Biological Systems by the Incorporation of Molecular Photoswitches
2013 StandoutNobel
A Field Guide to Foldamers
2001 Standout
Engineering Orthogonal Polypeptide GalNAc-Transferase and UDP-Sugar Pairs
2019 StandoutNobel
Stereoselective Michael addition of trimethyl aluminium to nitro acrylates: a route to 2-methyl-3-amino propionic acid
2003
Enantioselective Conjugate Additions
2000
Dramatic Improvement of the Enantiomeric Excess in the Asymmetric Conjugate Addition Reaction Using New Experimental Conditions
2002
Click Chemistry with O-Dimethylpropargylcarbamate for Preparation of pH-Sensitive Functional Groups. A Case Study
2007
Reversible Optical Transcription of Supramolecular Chirality into Molecular Chirality
2004 StandoutScienceNobel
Regioselective Synthesis of Nitrones by Decarboxylative Oxidation of N-Alkyl-α-amino Acids and Application to the Synthesis of 1-Azabicyclic Alkaloids
1999
On the Mechanism of the Copper-Catalyzed Enantioselective 1,4-Addition of Grignard Reagents to α,β-Unsaturated Carbonyl Compounds
2006 StandoutNobel
Identification of simple arylfluorosulfates as potent agents against resistant bacteria
2021 StandoutNobel
Catalytic Asymmetric Conjugate Addition and Allylic Alkylation with Grignard Reagents
2008 StandoutNobel
Cu−Catalyzed Enantioselective Conjugate Addition of Alkylzincs to Cyclic Nitroalkenes: Catalytic Asymmetric Synthesis of Cyclic α-Substituted Ketones
2002
Catalytic Asymmetric Synthesis of Unprotected β2-Amino Acids
2021 StandoutNobel
Extending the application of biocatalysis to meet the challenges of drug development
2018
Chiral Sulfur Ligands for Asymmetric Catalysis
2007
Cu-catalysed asymmetric 1,4-addition of Me3Al to nitroalkenes. Synthesis of (+)-ibuprofen
2005
Preparation of Achiral and of Enantiopure Geminally Disubstituted β-Amino Acids for β-Peptide Synthesis
2000
Copper(I) phosphoramidite catalyzed asymmetric conjugate addition of dialkylzinc reagents of α,β-unsaturated nitroacetates; an enantioselective route to β-aryl-nitroalkanes
1999 StandoutNobel
Diastereoselective Synthesis of Thieno[3′,2′:4,5]cyclopenta[1,2‐d][1,3]oxazolines − New Ligands for the Copper‐Catalyzed Asymmetric Conjugate Addition of Diethylzinc to Enones
2004
Asymmetric Bioreductions of β-Nitro Acrylates as a Route to Chiral β2-Amino Acids
2006
Disulfonimide-Catalyzed Asymmetric Synthesis of β3-Amino Esters Directly from N-Boc-Amino Sulfones
2013 StandoutNobel
Organocatalytic Asymmetric Transferhydrogenation of β-Nitroacrylates: Accessing β2-Amino Acids
2008 StandoutNobel
Catalytic enantioselective conjugate addition of Grignard reagents to cyclic α,β-unsaturated carbonyl compounds
1999
Identification and Co-complex Structure of a New S. pyogenes SpeB Small Molecule Inhibitor
2015
Recent advances in enantioselective copper-catalyzed 1,4-addition
2009 StandoutNobel
An external chiral amidophosphine ligand for asymmetric conjugate addition of organocopper
1998
Organocatalytic Asymmetric Transfer Hydrogenation of Nitroolefins
2007 StandoutNobel
Searching for Periodic Structures in β-Peptides
2001
A study of conjugate addition to a γ,δ-dioxolanyl-α,β-unsaturated ester
2001
Copper-catalyzed asymmetric conjugate addition of Grignard reagents to cyclic enones
2004 StandoutNobel
An Unusual Flavin-Dependent Halogenase from the Metagenome of the Marine Sponge Theonella swinhoei WA
2017
Catalytic, Enantioselective Alkylation of α-Imino Esters Using Late Transition Metal Phosphine Complexes as Catalysts
1998
Conversion of Propargylic Alcohols to β‐Oxo Esters Catalyzed by Novel Ruthenium‐Phosphoramidite Complexes
2008
A new chiral 2-sulfonylamino-2′-phosphino-1,1′-binaphthyl ligand for highly enantioselective copper-catalyzed conjugate addition of diethylzinc to benzylideneacetones
2004
Arylfluorosulfates Inactivate Intracellular Lipid Binding Protein(s) through Chemoselective SuFEx Reaction with a Binding Site Tyr Residue
2016 StandoutNobel
Abc Amino Acids: Design, Synthesis, and Properties of New Photoelastic Amino Acids
2006
Alternate Heme Ligation Steers Activity and Selectivity in Engineered Cytochrome P450-Catalyzed Carbene-Transfer Reactions
2018 StandoutNobel
Enantioselective Copper-Catalyzed Conjugate Addition and Allylic Substitution Reactions
2008
The Proline-Catalyzed Direct Asymmetric Three-Component Mannich Reaction: Scope, Optimization, and Application to the Highly Enantioselective Synthesis of 1,2-Amino Alcohols
2002 StandoutNobel
Cu-Catalyzed Azide−Alkyne Cycloaddition
2008 StandoutNobel
Enantioselective Synthesis of Nitroalkanes Bearing All-Carbon Quaternary Stereogenic Centers through Cu-Catalyzed Asymmetric Conjugate Additions
2005
Asymmetric conjugate addition of diethyl zinc to enones with tartrate chiral phosphite ligands
1997
Dynamic Control of Chiral Space in a Catalytic Asymmetric Reaction Using a Molecular Motor
2011 StandoutScienceNobel
Recent advances in the stereoselective synthesis of β-amino acids
2002
Amine-Salt-Controlled, Catalytic Asymmetric Conjugate Addition of Various Amines and Asymmetric Protonation
2004
Asymmetric Enamine Catalysis
2007 StandoutNobel
Aldehyde Selective Wacker Oxidations of Phthalimide Protected Allylic Amines: A New Catalytic Route to β3-Amino Acids
2009 StandoutNobel
Photopharmacology: Beyond Proof of Principle
2014 StandoutNobel
Enzymatic Halogenation and Dehalogenation Reactions: Pervasive and Mechanistically Diverse
2017
Sulfur(VI) Fluoride Exchange (SuFEx)-Enabled High-Throughput Medicinal Chemistry
2020 StandoutNobel
Copper-catalysed asymmetric 1,4-addition of organometallic reagents to 2-cyclohexenone using novel phosphine-phosphite ligands
2000
Ligand-Induced Acceleration of the Intramolecular [3 + 2] Cycloaddition between Alkynes and Alkylidenecyclopropanes
2005
Cyclic Tetrapeptides from Nature and Design: A Review of Synthetic Methodologies, Structure, and Function
2019
“Inverse Drug Discovery” Strategy To Identify Proteins That Are Targeted by Latent Electrophiles As Exemplified by Aryl Fluorosulfates
2017 StandoutNobel
Highly enantioselective copper-catalyzed conjugate addition of diethylzinc to cyclic enones with spirocyclic phosphoramidite ligands
2005
Biologically Active Molecules with a “Light Switch”
2006
Chemical Glycoproteomics
2016 StandoutNobel
An alkaloid-mediated desymmetrization of meso-anhydrides via a nucleophilic ring opening with benzyl alcohol and its application in the synthesis of highly enantiomerically enriched β-amino acids
2003
Works of Norbert Sewald being referenced
An improved method for the solution cyclization of peptides under pseudo-high dilution conditions
2004
Synthetic Routes towards Enantiomerically Pure β‐Amino Acids
2003
Enzymatic Halogenation of Tryptophan on a Gram Scale
2014
Helicobacter exploits integrin for type IV secretion and kinase activation
2007 Nature
A Helical RGD Motif Promoting Cell Adhesion: Crystal Structures of the Helicobacter pylori Type IV Secretion System Pilus Protein CagL
2013
Affinity‐Based Tagging of Protein Families with Reversible Inhibitors: A Concept for Functional Proteomics
2003
Synthesis of photoswitchable amino acids based on azobenzene chromophores: building blocks with potential for photoresponsive biomaterials
2004
Stereoselective synthesis of?-amino acids via conjugate addition of nitrogen nucleophiles to?,?-unsaturated esters ? Recent advances
1996
Analogues of Neuropeptide Y Containing β‐Aminocyclopropane Carboxylic Acids are the Shortest Linear Peptides That Are Selective for the Y1 Receptor
2003
Chemical tools for activity-based proteomics
2006
The First Total Synthesis of Efrapeptin C
2002
Basic conformers in ?-peptides
1999
Mit Integrinen zu neuen Therapien
2002
Synthesis of cyclic RGD-peptides containing β-amino acids
1997
Are β-Amino Acids γ-Turn Mimetics? Exploring A New Design Principle for Bioactive Cyclopeptides
2000
Synthesis of α-trifluoromethyl substituted α-amino acid derivatives from methyl 3,3,3-trifluoro-2-diazopropionate
1996
Characterization of a Chemical Affinity Probe Targeting Akt Kinases
2013
First Synthesis of a β2-Homoamino Acid by Enantioselective Catalysis
2002
New efficient syntheses of α-diflyoromethyl- and α-trifluoromethyl-ornithine
1997
One-Pot Azidochlorination of Glycals
2011
Synthese 2‐Heteroaryl‐substituierter 3,3,3‐Trifluoralanin‐ und 3,3,3‐Trifluormilchsäure‐Derivate
1992
Conjugate Addition of Mixed Diorganozinc Compounds and Functionalized Organozinc Cuprates to Nitroolefins
2002
Synthesis of γ-oxo α-amino acids from L-aspartic acid
1996
Affinitätsbasierte Markierung von Proteinfamilien mit reversiblen Inhibitoren – ein Konzept für die funktionelle Proteomik
2003
Die erste Totalsynthese von Efrapeptin C
2002
Inhibitor‐based affinity probes for the investigation of JAK signaling pathways
2015
A High‐Throughput Fluorescence Assay to Determine the Activity of Tryptophan Halogenases
2016
Asymmetric synthesis of β‐amino acids and α‐deuterated β‐amino acids via conjugate addition of homochiral amidocuprates
1995
Enzymatische Halogenierung von Tryptophan im Gramm‐Maßstab
2014
Neuropeptid‐Y‐Analoga mit β‐Aminocyclopropancarbonsäure‐Einheiten sind die kürzesten linearen und selektiven Peptide am Y1‐Rezeptor
2003
Enantioselective copper(I) catalyzed 1,4-addition of diethylzinc to nitroolefins
1998
Enantioselective copper(I) catalyzed 1,4-addition of diethylzinc to cyclohexenone: asymmetric induction as an unexpected source of structural information
1997
Modular Combination of Enzymatic Halogenation of Tryptophan with Suzuki–Miyaura Cross‐Coupling Reactions
2016
Neue Wege zu enantiomerenreinen β‐Aminosäuren
2003
Proteolytically stable peptides by incorporation of α-Tfm amino acids
1997
Tandem Protocol for the Stereoselective Synthesis of Different Polyfunctional β-Amino Acids and 3-Amino-Substituted Carbohydrates
1998
Stereoselective synthesis of β-homothreonine and 3-amino substituted carbohydrates
1998
Regioselective Enzymatic Halogenation of Substituted Tryptophan Derivatives using the FAD‐Dependent Halogenase RebH
2014