Citation Impact
Citing Papers
Diversity oriented clicking delivers β-substituted alkenyl sulfonyl fluorides as covalent human neutrophil elastase inhibitors
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Bifluoride Ion Mediated SuFEx Trifluoromethylation of Sulfonyl Fluorides and Iminosulfur Oxydifluorides
2019 StandoutNobel
Palladium-catalyzed N-arylation of 2-aminobenzothiazole-4-carboxylates/carboxamides: facile synthesis of PARP14 inhibitors
2014
First enantioselective addition of dialkylzinc to ketones promoted by titanium(IV) derivatives
1998
Disulfonimide‐Catalyzed Asymmetric Reduction of N‐Alkyl Imines
2015 StandoutNobel
Construction of a Tetracyclic Butterfly‐Like Scaffold: Palladium‐Catalyzed Heck/Arylation Cascade
2010
Dynamic Covalent Chemistry
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Oxindole synthesis by direct C–H, Ar–H coupling
2009
Carbon–heteroatom bond formation catalysed by organometallic complexes
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2010
Introduction of Fluorine and Fluorine‐Containing Functional Groups
2013 Standout
Structure-based design and optimization of 2-aminothiazole-4-carboxamide as a new class of CHK1 inhibitors
2013
Catalyst‐Controlled Chemoselective Arylation of 2‐Aminobenzimidazoles
2012
Formation of pentacyclic structures by a domino sequence on cyclic enamides
2009
A Highly Versatile Catalyst System for the Cross‐Coupling of Aryl Chlorides and Amines
2009
Transition metal-catalyzed N-arylations of amidines and guanidines
2012
A Powerful Brønsted Acid Catalyst for the Organocatalytic Asymmetric Transfer Hydrogenation of Imines
2005 StandoutNobel
Sulfonyl fluorides as targets and substrates in the development of new synthetic methods
2022
Palladium-catalyzed coupling of functionalized primary and secondary amines with aryl and heteroaryl halides: two ligands suffice in most cases
2010
Highly Reactive, General, and Long‐Lived Catalysts for Coupling Heteroaryl and Aryl Chlorides with Primary Nitrogen Nucleophiles
2005
BippyPhos: A Single Ligand With Unprecedented Scope in the Buchwald–Hartwig Amination of (Hetero)aryl Chlorides
2013
Monodentate Phosphines Provide Highly Active Catalysts for Pd‐Catalyzed CN Bond‐Forming Reactions of Heteroaromatic Halides/Amines and (H)N‐Heterocycles
2006
Design and Enantioselective Synthesis of Cashmeran Odorants by Using “Enol Catalysis”
2015 StandoutNobel
Recent Developments in Asymmetric Phase‐Transfer Reactions
2013
Stereochemical Communication within a Chiral Ion Pair Catalyst
2015 StandoutNobel
Chemoselective Amination of Propargylic C(sp3)H Bonds by Cobalt(II)‐Based Metalloradical Catalysis
2014
Fast, greener and scalable direct coupling of organolithium compounds with no additional solvents
2016 StandoutNobel
The First Polymer-Supported and Recyclable Chiral Catalyst for Enantioselective Olefin Metathesis
2002 StandoutNobel
Can a Ketone Be More Reactive than an Aldehyde? Catalytic Asymmetric Synthesis of Substituted Tetrahydrofurans
2018 StandoutNobel
Electroreductive acylation of aromatic imines with acylimidazoles
2007
SuFEx Click Chemistry Enabled Late-Stage Drug Functionalization
2018 StandoutNobel
Catalytic Asymmetric Reductive Condensation of N–H Imines: Synthesis of C2‐Symmetric Secondary Amines
2016 StandoutNobel
Atom Economy—A Challenge for Organic Synthesis: Homogeneous Catalysis Leads the Way
1995 Standout
Palladium-Catalyzed Hiyama Cross-Couplings of Aryl Arenesulfonates with Arylsilanes
2008
Synthesis of (Vinylallene)rhodium(III) Complex of Planar Structure: Perfect π → σ Conversion of 1,3-Diene System
1996
Iridium/Monodentate Phosphoramidite Catalyzed Asymmetric Hydrogenation ofN-Aryl Imines
2009 StandoutNobel
Palladium‐Catalyzed CN and CO Coupling–A Practical Guide from an Industrial Vantage Point†
2004
Fluorine in Pharmaceutical Industry: Fluorine-Containing Drugs Introduced to the Market in the Last Decade (2001–2011)
2013 Standout
Expedited Palladium-Catalyzed Amination of Aryl Nonaflates through the Use of Microwave-Irradiation and Soluble Organic Amine Bases
2005
Room-Temperature Ionic Liquids: Solvents for Synthesis and Catalysis. 2
2011 Standout
First enantioselective addition of diethylzinc and dimethylzinc to prostereogenic ketones catalysed by camphorsulfonamide-titanium alkoxide derivatives
1998
Palladium-Catalyzed N-Arylation of 2-Aminothiazoles
2012
Carbenoid Complexes of Electron‐Deficient Transition Metals—Syntheses of and with Short‐Lived Building Blocks
1997
Copper-Catalyzed Coupling of Tertiary Aliphatic Amines with Terminal Alkynes to Propargylamines via C−H Activation
2008
Engineered Biosynthesis of β‐Alkyl Tryptophan Analogues
2018 StandoutNobel
Synthesis of Pyridine and Dihydropyridine Derivatives by Regio- and Stereoselective Addition toN-Activated Pyridines
2012 Standout
Recent developments in solvent-free multicomponent reactions: a perfect synergy for eco-compatible organic synthesis
2012
Engineering enzymes for noncanonical amino acid synthesis
2018 StandoutNobel
Cyclometalated Phosphine-Based Pincer Complexes: Mechanistic Insight in Catalysis, Coordination, and Bond Activation
2003 Standout
Diastereoselective addition of methyllithium and dimethylcuprate-boron trifluoride to imines derived from (S)-1-phenylethylamine
1996
Catalytic Enantioselective Conversion of Epoxides to Thiiranes
2016 StandoutNobel
Chelation-assisted carbon–carbon bond activation by Rh(I) catalysts
2002
Evolution of Titanium(IV) Alkoxides and Raney Nickel for Asymmetric Reductive Amination of Prochiral Aliphatic Ketones
2005
Electron‐Reservoir Complexes [FeICp(arene)] as Selective Initiators for a Novel Electron Transfer Chain Catalyzed Reaction: General Synthesis of Fulvalene‐Bridged Homo‐ and Heterodinuclear Zwitterions
1994
Direct Dehydrative N-Pyridinylation of Amides
2008
Applicability Aspects of Transition Metal‐Catalyzed Aromatic Amination Protocols in Medicinal Chemistry
2007
A Multifunctional Reagent Designed for the Site-Selective Amination of Pyridines
2020
Titanium and Zirconium Complexes That Contain the Tridentate Diamido Ligands [(i-PrN-o-C6H4)2O]2-([i-PrNON]2-) and [(C6H11N-o-C6H4)2O]2-([CyNON]2-)
1999 StandoutNobel
Carboxylate-Assisted Transition-Metal-Catalyzed C−H Bond Functionalizations: Mechanism and Scope
2011 Standout
Rhodium(I)-Catalyzed Successive Double Cleavage of Carbon−Carbon Bonds of Strained Spiro Cyclobutanones
1997
[(CyPF-tBu)PdCl2]: An Air-Stable, One-Component, Highly Efficient Catalyst for Amination of Heteroaryl and Aryl Halides
2008
Transition Metal-Catalyzed [6+2] Cycloadditions of 2-Vinylcyclobutanones and Alkenes: A New Reaction for the Synthesis of Eight-Membered Rings
2000
Merging Nucleophilic and Hydrogen Bonding Catalysis: An Anion Binding Approach to the Kinetic Resolution of Propargylic Amines
2010
Palladium-Catalyzed C–N Cross Coupling of Sulfinamides and Aryl Halides
2012
The chemistry of group 10 metalacycles
1999
Efficient Catalytic Enantioselective Synthesis of Unsaturated Amines: Preparation of Small- and Medium-Ring Cyclic Amines through Mo-Catalyzed Asymmetric Ring-Closing Metathesis in the Absence of Solvent
2002 StandoutNobel
Copper-Catalyzed Synthesis of Mixed Alkyl Aryl Phosphonates
2014 StandoutNobel
The medicinal chemist's toolbox for late stage functionalization of drug-like molecules
2015
Synthesis, Structure, Magnetism, and Single Molecular Conductance of Linear Trinickel String Complexes with Sulfur‐Containing Ligands
2012
A convergent approach to the synthesis of aprepitant: a potent human NK-1 receptor antagonist
2007
Domino Palladium-Catalyzed Heck-Intermolecular Direct Arylation Reactions
2009
Transition Metal-Mediated Cycloaddition Reactions
1996 Standout
Asymmetric synthesis of amines by nucleophilic 1,2-addition of organometallic reagents to the CN-double bond
1997
Catalytic Dehydrogenative Cross-Coupling: Forming Carbon−Carbon Bonds by Oxidizing Two Carbon−Hydrogen Bonds
2011 Standout
Aryl−Aryl Bond Formation by Transition-Metal-Catalyzed Direct Arylation
2007 Standout
Electroreductive Acylation of Aromatic Ketones with Acylimidazoles
2005
A Bifunctional Reagent Designed for the Mild, Nucleophilic Functionalization of Pyridines
2017
Magnesiation of Pyridine N-Oxides via Iodine or Bromine−Magnesium Exchange: A Useful Tool for Functionalizing Pyridine N-Oxides
2008
Internal Activation of Peptidyl Prolyl Thioesters in Native Chemical Ligation
2016
Azine Activation via Silylium Catalysis
2021 StandoutNobel
Metal-Mediated Synthesis of Medium-Sized Rings
2000
Overcoming Resistance to β-Lactam Antibiotics
2013
Organocatalytic C–H Bond Arylation of Aldehydes to Bis-heteroaryl Ketones
2013
Computationally designed peptide macrocycle inhibitors of New Delhi metallo-β-lactamase 1
2021 StandoutNobel
Additions of Organometallic Reagents to CN Bonds: Reactivity and Selectivity
1998 Standout
Catalytic Non‐Enzymatic Kinetic Resolution
2011
Carbon−Carbon Bond Activation by Rhodium(I) in Solution. Comparison of sp2−sp3 vs sp3−sp3 C−C, C−H vs C−C, and Ar−CH3 vs Ar−CH2CH3 Activation
1998
Synthetic Organic Electrochemical Methods Since 2000: On the Verge of a Renaissance
2017 Standout
Regioselective Synthesis of Nitrones by Decarboxylative Oxidation of N-Alkyl-α-amino Acids and Application to the Synthesis of 1-Azabicyclic Alkaloids
1999
Regioselective synthesis of benzimidazole thiophene inhibitors of polo-like kinase 1
2008
Development of practical syntheses of potent non-nucleoside reverse transcriptase inhibitors
2009
C–H Functionalization of Azines
2017
Chiral Phosphoric Acid‐Catalyzed Asymmetric Aza‐Friedel–Crafts Reaction of Indoles with Cyclic N‐Acylketimines: Enantioselective Synthesis of Trifluoromethyldihydroquinazolines
2013
High Oxidation State Multiple Metal−Carbon Bonds
2001 StandoutNobel
Carenium−CalkylBond Making and Breaking: Key Process in the Platinum-Mediated Caryl−CalkylBond Formation. Analogies to Organic Electrophilic Aromatic Substitution
2001
Neue Entwicklungen bei asymmetrischen Phasentransferreaktionen
2013
Escape from Flatland: Increasing Saturation as an Approach to Improving Clinical Success
2009 Standout
Design, Synthesis, and Evaluation of 2-Methyl- and 2-Amino-N-aryl-4,5-dihydrothiazolo[4,5-h]quinazolin-8-amines as Ring-Constrained 2-Anilino-4-(thiazol-5-yl)pyrimidine Cyclin-Dependent Kinase Inhibitors
2010
Unusual Amino Acids in Medicinal Chemistry
2016
Applications of Palladium-Catalyzed C–N Cross-Coupling Reactions
2016 Standout
Chiral Allenes via Alkynylogous Mukaiyama Aldol Reaction
2016 StandoutNobel
IDPi Catalysis
2019 StandoutNobel
Asymmetric Catalysis of the Carbonyl-Amine Condensation: Kinetic Resolution of Primary Amines
2017 StandoutNobel
Synthesis and Late-Stage Functionalization of Complex Molecules through C–H Fluorination and Nucleophilic Aromatic Substitution
2014
Asymmetric Catalysis via Cyclic, Aliphatic Oxocarbenium Ions
2017 StandoutNobel
Transition Metal Catalyzed Cycloisomerizations of 1,n-Allenynes and -Allenenes
2011 Standout
Mechanistic Investigation of Catalytic Carbon−Carbon Bond Activation and Formation by Platinum and Palladium Phosphine Complexes
1998
Einführung von Fluor und fluorhaltigen funktionellen Gruppen
2013
New Electrosynthesis of Arylboronic Esters from Aromatic Halides and Pinacolborane
2003
Highly Reactive, General and Long-Lived Catalysts for Palladium-Catalyzed Amination of Heteroaryl and Aryl Chlorides, Bromides, and Iodides: Scope and Structure–Activity Relationships
2008
Palladium mediated intramolecular multiple C–X/C–H cross coupling and C–H activation: synthesis of carbazole alkaloids calothrixin B and murrayaquinone A
2014
Enantioselective addition of alkynes to imines in ionic liquids
2004
Copper-Catalyzed Enantioselective Additions to Oxocarbenium Ions: Alkynylation of Isochroman Acetals
2011
Synthesis of the benzo-β-carboline isoneocryptolepine: the missing indoloquinoline isomer in the alkaloid series cryptolepine, neocryptolepine and isocryptolepine
2004
Stapled β-Hairpins Featuring 4-Mercaptoproline
2021 StandoutNobel
Rhodium-Catalyzed C−C Bond Formation via Heteroatom-Directed C−H Bond Activation
2009 Standout
Asymmetric Enamine Catalysis
2007 StandoutNobel
A Rhodium-Catalyzed C−H Activation/Cycloisomerization Tandem
2007
Merging Nucleophilic and Hydrogen Bonding Catalysis: An Anion Binding Approach to the Kinetic Resolution of Amines
2009
The Heck Reaction as a Sharpening Stone of Palladium Catalysis
2000 Standout
Development of nonproprietary phosphine ligands for the Pd-catalyzed amination reaction
2006
Selective Hydrogenation for Fine Chemicals: Recent Trends and New Developments
2003
Atomökonomische Synthesen – eine Herausforderung in der Organischen Chemie: die Homogenkatalyse als wegweisende Methode
1995
Chemical Redox Agents for Organometallic Chemistry
1996 Standout
Catalytic Asymmetric Conjugate Addition of Indolizines to α,β‐Unsaturated Ketones
2017 StandoutNobel
Generation of Anti-trypanosomal Agents through Concise Synthesis and Structural Diversification of Sesquiterpene Analogues
2011 StandoutNobel
Works of Mark A. Huffman being referenced
Palladium‐Catalyzed Tandem Heck Reaction/CH Functionalization—Preparation of Spiro‐Indane‐Oxindoles
2008
Pd-Catalyzed N-Arylation of Heteroarylamines
2002
A General and Efficient 2-Amination of Pyridines and Quinolines
2007
Dimethyltitanocene: From Millimole to Kilomole
2004
Syntheses of morpholine-2,3-diones and 2-hydroxymorpholin-3-ones: intermediates in the synthesis of aprepitant
2004
Reaktion zwischen Pentacarbonyl(fulvalen)‐molybdänruthenium und Alkinen: Dynamik, Strukturen und Umlagerungen der Produkte sowie erste reversible Umwandlung eines side‐on‐koordinierten in einen semiüberbrückenden Alkenylidenliganden
1991
Synthesis of a selective estrogen receptor β-modulator via asymmetric phase-transfer catalysis
2007
Highly Diastereoselective Catalytic Meerwein−Ponndorf−Verley Reductions
2005
Pd‐Catalyzed N‐Arylation of Heteroarylamines.
2003
Lithium Alkoxides of Cinchona Alkaloids as Chiral Controllers for Enantioselective Acetylide Addition to Cyclic N-Acyl Ketimines
1995
A very concise synthesis of a potent N-(1,3-thiazol-2-yl)pyridin-2-amine KDR kinase inhibitor
2005
Alternatives to Vinyl Triflates for Cross-Coupling with Arylboronic Acids
1999
Direct and Convenient Conversion of Alcohols to Fluorides
2004
Nickel(0)-catalyzed synthesis of substituted phenols from cyclobutenones and alkynes
1991
Designed syntheses of heterobimetallic fulvalene complexes
1986
Route Development and Multikilogram GMP Delivery of a Somatostatin Receptor Antagonist
2012
Unique Reactivity of Heterodinuclear Pentacarbonyl(fulvalene)molybdenumruthenium with Alkynes: Fluxionality, Rearrangements, Structures, and First Reversible Conversion of a “Side‐on”‐ to a Semi‐Bridging Alkenylidene Ligand
1991
Palladium‐Catalyzed Tandem Heck Reaction/CH Functionalization—Preparation of Spiro‐Indane‐Oxindoles
2008
Reaction of cyclobutenones with low-valent metal reagents to form .eta.4- and .eta.2-vinylketene complexes. Reaction of .eta.4-vinylketene complexes with alkynes to form phenols
1992
Synthesis of a Potent hNK-1 Receptor Antagonist via an SN2 Reaction of an Enantiomerically Pure α-Alkoxy Sulfonate
2004
Improved stereoselectivity in the heterogeneous catalytic synthesis of enalapril obtained through multidimensional screening
1999
A Concise Synthesis of a β-Lactamase Inhibitor
2011
Rhodium(I)-catalyzed intramolecular carbocyclic ring fusion: a new approach to medium-sized-ring ketones
1993