Citation Impact
Citing Papers
A monomeric G protein-coupled receptor isolated in a high-density lipoprotein particle efficiently activates its G protein
2007 StandoutNobel
Ionotropic and metabotropic glutamate receptor structure and pharmacology
2005
Structure−Activity Relationship of N-(Phenylalkyl)cinnamides as Novel NR2B Subtype-Selective NMDA Receptor Antagonists
1999
Pharmacology of AMPA/Kainate Receptor Ligands and Their Therapeutic Potential in Neurological and Psychiatric Disorders
2000
Mitigating risk in academic preclinical drug discovery
2015
Catalytic enantiocontrol over a non-classical carbocation
2020 StandoutNobel
Palladium-catalyzed direct ortho-C–H ethoxycarboxylation of anilides at room temperature
2014
Potent and Selective Triazole-Based Inhibitors of the Hypoxia-Inducible Factor Prolyl-Hydroxylases with Activity in the Murine Brain
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Subtype-selective antagonism of NMDA receptors by nylidrin
1997
Glutamate receptor ion channels
2005 Standout
Glutamate Receptor Ion Channels: Structure, Regulation, and Function
2010 Standout
Pharmacological Characterization of Ro 63-1908 (1-[2-(4-Hydroxy-phenoxy)-ethyl]-4-(4-methyl-benzyl)-piperidin-4-ol), a Novel Subtype-Selective N-Methyl-d-Aspartate Antagonist
2002
Synergistic effects of caspase inhibitors and MK‐801 in brain injury after transient focal cerebral ischaemia in mice
1998
Inhibition of the NMDA response by pregnenolone sulphate reveals subtype selective modulation of NMDA receptors by sulphated steroids
2002
C–C, C–O and C–N bond formation via rhodium(iii)-catalyzed oxidative C–H activation
2012 Standout
Channel opening and gating mechanism in AMPA-subtype glutamate receptors
2017 StandoutNatureNobel
D-Alanine Added to Antipsychotics for the Treatment of Schizophrenia
2005
Design and evaluation of 1,7-naphthyridones as novel KDM5 inhibitors
2016
Photoaffinity labeling and its application in structural biology
2007
Piezo2 is required for Merkel-cell mechanotransduction
2014 StandoutNatureNobel
Recent advances in organocatalytic methods for the synthesis of disubstituted 2- and 3-indolinones
2012 Standout
Mechanochemistry: opportunities for new and cleaner synthesis
2011 Standout
The adolescent brain and age-related behavioral manifestations
2000 Standout
Role of GABAA Receptors in the Regulation of Sleep: Initial Sleep Responses to Peripherally Administered Modulators and Agonists
1999
Endogenous and synthetic neurosteroids in treatment of Niemann–Pick Type C disease
2007
Palladium‐Catalyzed Cross‐Coupling: A Historical Contextual Perspective to the 2010 Nobel Prize
2012 Standout
Enzymatic assembly of carbon–carbon bonds via iron-catalysed sp3 C–H functionalization
2018 StandoutNatureNobel
Non-competitive metabotropic glutamate 1 receptor antagonists block activity of slowly adapting type I mechanoreceptor units in the rat sinus hair follicle
2009
Estimation of Blood-Brain Barrier Crossing of Drugs Using Molecular Size and Shape, and H-Bonding Descriptors
1998
A comparative assessment of the efficacy and side-effect liability of neuroprotective compounds in experimental stroke
2001
Competitive AMPA receptor antagonists
2006
Modulation of GABAA receptor desensitization uncouples sleep onset and maintenance in Drosophila
2008 StandoutNobel
Subtype-Selective N-Methyl-d -Aspartate Receptor Antagonists: Synthesis and Biological Evaluation of 1-(Heteroarylalkynyl)-4-benzylpiperidines
2000
Direct addition of alkynes to imines and related CN electrophiles: A convenient access to propargylamines
2006
Photoactivation of a nanoporous crystal for on-demand guest trapping and conversion
2010 StandoutNobel
Thiourea‐Enhanced Flavin Photooxidation of Benzyl Alcohol
2007
Neuroactive Steroid Modulators of the Stress Response
1995
Catalytic asymmetric synthesis of chromenes and tetrahydroquinolines via sequential allylic alkylation and intramolecular Heck coupling
2012 StandoutNobel
Iron-catalyzed ene-type propargylation of diarylethylenes with propargyl alcohols
2011
Asymmetric Alkynylation of Imines by Cooperative Hydrogen Bonding and Metal Catalysis
2009
The Cross‐Dehydrogenative Coupling of CH Bonds: A Versatile Strategy for CC Bond Formations
2013 Standout
SwissADME: a free web tool to evaluate pharmacokinetics, drug-likeness and medicinal chemistry friendliness of small molecules
2017 Standout
Oxamides as novel NR2B selective NMDA receptor antagonists
2004
Structural Bases of Desensitization in AMPA Receptor-Auxiliary Subunit Complexes
2017 StandoutNobel
Chlorinated phenyl azides as photolabeling reagents. Synthesis of an ortho,ortho'-dichlorinated arylazido PCP receptor ligand
1993
Organic Azides: An Exploding Diversity of a Unique Class of Compounds
2005 Standout
Synthesis, 3D-QSAR, and docking studies of 1-phenyl-1H-1,2,3-triazoles as selective antagonists for β3 over α1β2γ2 GABA receptors
2007
Structural Model of the N-Methyl-D-aspartate Receptor Glycine Site Probed by Site-directed Chemical Coupling
2003
Activity-dependent regulation of dendritic synthesis and trafficking of AMPA receptors
2004 StandoutNobel
GABA mechanisms and sleep
2002
Autochthonous tumors driven by Rb1 loss have an ongoing requirement for the RBP2 histone demethylase
2018 StandoutNobel
Click Chemistry for Drug Development and Diverse Chemical–Biology Applications
2013 Standout
Iron Catalysis in Organic Synthesis
2015 Standout
Elucidation of AMPA receptor–stargazin complexes by cryo–electron microscopy
2016 StandoutScienceNobel
Physiological Implications of Hydrogen Sulfide: A Whiff Exploration That Blossomed
2012 Standout
Solvent-Free Heterocyclic Synthesis
2009
Tetrahydroquinoline and tetrahydroisoquinoline mixed ligand rhenium complexes with the SNS/S donor atom set
2007
Supramolecular Coordination: Self-Assembly of Finite Two- and Three-Dimensional Ensembles
2011 Standout
Chemical Strategies To Target Bacterial Virulence
2017
Organic Photoredox Catalysis
2016 Standout
New four-component reactions in water: a convergent approach to the metal-free synthesis of spiro[indoline/acenaphthylene-3,4′-pyrazolo[3,4-b]pyridine derivatives
2011
Catalyzed Propargylic Substitution
2009
State of the Art and Prospects in Metal–Organic Framework (MOF)-Based and MOF-Derived Nanocatalysis
2019 Standout
Mild metal-catalyzed C–H activation: examples and concepts
2016 Standout
Comparison of Phenylcarbene and Phenylnitrene
1995
N-Heterocyclic Carbenes in Late Transition Metal Catalysis
2009 Standout
Large-Size Linear and Star-Shaped Dihydropyrazine Fused Pyrazinacenes
2012
Advances in the Chemistry of Tetrahydroquinolines
2011 Standout
Kinetics, Spectroscopy, and Computational Chemistry of Arylnitrenes
2006
NR2B subtype-selective NMDA receptor antagonists: 2001 – 2004
2005
Remarkable tolerance of ethynyl steroids to air and water in microwave-assisted hydrophosphinylation: Reaction scope and limitations
2006
Genetic identification of HSD-1, a conserved steroidogenic enzyme that directs larval development inCaenorhabditis elegans
2008 StandoutNobel
Asymmetric Organocatalytic Tandem Cyclization/Transfer Hydrogenation: A Synthetic Strategy for Enantioenriched Nitrogen Heterocycles
2013
Chemical reagents in photoaffinity labeling
1995
Silyl modification of biologically active compounds. 11. Synthesis, physico‐chemical and biological evaluation of N‐(trialkoxysilylalkyl)tetrahydro(iso,silaiso) quinoline derivatives
2005
Reversible Photocontrol of Biological Systems by the Incorporation of Molecular Photoswitches
2013 StandoutNobel
Microwave-Assisted Synthesis in Water as Solvent
2007 Standout
The Glutamate Receptor Ion Channels
1999 Standout
About Sleep's Role in Memory
2013 Standout
The Essential Roles of Chemistry in High-Throughput Screening Triage
2014
Ischemic Cell Death in Brain Neurons
1999 Standout
The Combinatorial Synthesis of Bicyclic Privileged Structures or Privileged Substructures
2003 Standout
Total Synthesis of Ningalin B Utilizing a Heterocyclic Azadiene Diels−Alder Reaction and Discovery of a New Class of Potent Multidrug Resistant (MDR) Reversal Agents
2000
Reactive Oxygen Species (ROS)-Based Nanomedicine
2019 Standout
Synthetic Applications of Pd(II)-Catalyzed C−H Carboxylation and Mechanistic Insights: Expedient Routes to Anthranilic Acids, Oxazolinones, and Quinazolinones
2009
Direct Synthesis of 4-Arylpiperidines via Palladium/Copper(I)-Cocatalyzed Negishi Coupling of a 4-Piperidylzinc Iodide with Aromatic Halides and Triflates
2004
Post-synthetically modified MOF for the A3-coupling reaction of aldehyde, amine, and alkyne
2018
A Photoactivatable Push−Pull Fluorophore for Single-Molecule Imaging in Live Cells
2008 StandoutNobel
Organocatalytic Reduction of Carbon−Carbon Double Bonds in Racemization-Sensitive Compounds
2011 StandoutNobel
Complete Field Guide to Asymmetric BINOL-Phosphate Derived Brønsted Acid and Metal Catalysis: History and Classification by Mode of Activation; Brønsted Acidity, Hydrogen Bonding, Ion Pairing, and Metal Phosphates
2014 Standout
The glutamate receptor ion channels.
1999
Gold-Catalyzed Carbon−Heteroatom Bond-Forming Reactions
2011 Standout
Photoaffinity Labeling Introduction
1997
Chemistry: Chemical con artists foil drug discovery
2014 StandoutNature
Heterocyclic Nanographenes and Other Polycyclic Heteroaromatic Compounds: Synthetic Routes, Properties, and Applications
2016 Standout
Azido Push−Pull Fluorogens Photoactivate to Produce Bright Fluorescent Labels
2009 StandoutNobel
Lamellarins and Related Pyrrole-Derived Alkaloids from Marine Organisms
2007 Standout
Chiral amine–imine ligands based on trans-2,5-disubstituted pyrrolidines and their application in the palladium-catalyzed allylic alkylation
2009
C−F Bond Activation in Organic Synthesis
2009
Recent Trends in Photoaffinity Labeling
1995
In Vivo Protein Transduction: Delivery of a Biologically Active Protein into the Mouse
1999 StandoutScience
Works of Jon E. Hawkinson being referenced
Correlation of neuroactive steroid modulation of [35S]t-butylbicyclophosphorothionate and [3H]flunitrazepam binding and gamma-aminobutyric acidA receptor function.
1994
Characterization of the Anticonvulsant Properties of Ganaxolone (CCD 1042; 3α-Hydroxy-3β-methyl-5α-pregnan-20-one), a Selective, High-Affinity, Steroid Modulator of the γ-Aminobutyric AcidA Receptor
1997
3 alpha-Hydroxy-3 beta-trifluoromethyl-5 alpha-pregnan-20-one (Co 2-1970): a partial agonist at the neuroactive steroid site of the gamma-aminobutyric acidA receptor.
1996
CCD-3693: An Orally Bioavailable Analog of the Endogenous Neuroactive Steroid, Pregnanolone, Demonstrates Potent Sedative Hypnotic Actions in the Rat
1997
Synthesis and SAR of 5-, 6-, 7- and 8-Aza Analogues of 3-Aryl-4-hydroxyquinolin-2(1H)-one as NMDA/Glycine Site Antagonists
2001
The metabotropic glutamate receptor antagonist l-2-amino-3-phosphonopropionic acid inhibits phosphoserine phosphatase
1996
Photoaffinity Ligands for the [3H]tbob Binding Site of the GabaAReceptor
1991
Subtype-Selective N-Methyl-d -aspartate Receptor Antagonists: Synthesis and Biological Evaluation of 1-(Arylalkynyl)-4-benzylpiperidines
1999
From HTS to Phase I: The Institute for Therapeutics Discovery and Development at the University of Minnesota
2014
Formation of d ‐Serine from l ‐Phosphoserine in Brain Synaptosomes
1996
Synthesis and SAR of novel di- and trisubstituted 1,4-dihydroquinoxaline-2,3-diones related to licostinel (Acea 1021) as NMDA/glycine site antagonists
2003
The N-methyl-d-aspartate (NMDA) receptor glycine site antagonist ACEA 1021 does not produce pathological changes in rat brain
1997
Photoactivatable 2-[(4'-azido)tetrafluorophenyl]-5-tert-butyl-1,3-dithiane bissulfone and related compounds as candidate irreversible probes for the GABA-gated chloride channels
1994
Probing the S2′ Subsite of the Anthrax Toxin Lethal Factor Using Novel N-Alkylated Hydroxamates
2015
Diazocyclohexadienones as photoaffinity ligands: Syntheses of trioxabicyclooctane probes for the convulsant binding site of the GABAA receptor
1989
N-methyl-D-aspartate antagonists for stroke and head trauma
1997
Preparation and Optimization of a Series of 3-Carboxamido-5-phenacylaminopyrazole Bradykinin B1 Receptor Antagonists
2007
Synthesis of N-Substituted 4-(4-Hydroxyphenyl)piperidines, 4-(4-Hydroxybenzyl)piperidines, and (±)-3-(4-Hydroxyphenyl)pyrrolidines: Selective Antagonists at the 1a /2B NMDA Receptor Subtype
2000
Structure−Activity Relationships of Alkyl- and Alkoxy-Substituted 1,4-Dihydroquinoxaline-2,3-diones: Potent and Systemically Active Antagonists for the Glycine Site of the NMDA Receptor
1997
5-(N-Oxyaza)-7-substituted-1,4-dihydroquinoxaline-2,3-diones: Novel, Systemically Active and Broad Spectrum Antagonists for NMDA/glycine, AMPA, and Kainate Receptors
1997
4-Hydroxy-1-[2-(4-hydroxyphenoxy)ethyl]-4-(4-methylbenzyl)piperidine: A Novel, Potent, and Selective NR1/2B NMDA Receptor Antagonist
1999
3α-Hydroxy-3β-(phenylethynyl)-5β-pregnan-20-ones: Synthesis and Pharmacological Activity of Neuroactive Steroids with High Affinity for GABAA Receptors
1997
Characterization of the anticonvulsant properties of ganaxolone (CCD 1042; 3alpha-hydroxy-3beta-methyl-5alpha-pregnan-20-one), a selective, high-affinity, steroid modulator of the gamma-aminobutyric acid(A) receptor.
1997
Synthesis and Structure−Activity Relationships of 1,2,3,4-Tetrahydroquinoline-2,3,4-trione 3-Oximes: Novel and Highly Potent Antagonists for NMDA Receptor Glycine Site
1996
Analogs of 3-Hydroxy-1H-1-benzazepine-2,5-dione: Structure−Activity Relationship atN-Methyl-d -aspartate Receptor Glycine Sites
1996