Citation Impact

Citing Papers

Incorporation of azides into recombinant proteins for chemoselective modification by the Staudinger ligation
2001 StandoutNobel
Part 1: Structure–Activity Relationship (SAR) investigations of fused pyrazoles as potent, selective and orally available inhibitors of p38α mitogen-activated protein kinase
2009
Synthesis of Naturally Occurring Polyynes
2006
Cellular and Gene Expression Responses Involved in the Rapid Growth Inhibition of Human Cancer Cells by RNA Interference-mediated Depletion of Telomerase RNA
2005 StandoutNobel
Shape-persistent macrocycle with a self-complementary recognition pattern based on diacetylene-linked alternating hexylbenzene and perfluorobenzene rings
2006 StandoutNobel
The αvintegrin antagonists as novel anticancer agents: an update
2002
Aminomutases: mechanistic diversity, biotechnological applications and future perspectives
2011 StandoutNobel
A targeted contrast agent for magnetic resonance imaging of thrombus: Implications of spatial resolution
2001
A self assembled molecular zipper based on a perfluorophenyl-phenyl diacetylene motif
2006 StandoutNobel
Future Therapeutic Directions in Reverse Cholesterol Transport
2010
Genetically programmed chiral organoborane synthesis
2017 StandoutNatureNobel
PI3Kγ inhibition: towards an 'aspirin of the 21st century'?
2006
Peptidomimetic design
1998
A Stepwise Huisgen Cycloaddition Process: Copper(I)-Catalyzed Regioselective “Ligation” of Azides and Terminal Alkynes
2002 StandoutNobel
Oncogenic Mutations Counteract Intrinsic Disorder in the EGFR Kinase and Promote Receptor Dimerization
2012 StandoutNobel
Click Chemistry: Diverse Chemical Function from a Few Good Reactions
2001 StandoutNobel
Update on strategies to increase HDL quantity and function
2009
Shape-persistent macrocycles comprising perfluorinated benzene subunits: synthesis, aggregation behaviour and unexpected μ-rod formation
2009 StandoutNobel
Mechanism‐Inspired Engineering of Phenylalanine Aminomutase for Enhanced β‐Regioselective Asymmetric Amination of Cinnamates
2011 StandoutNobel
Iron catalysed direct alkylation of amines with alcohols
2014 StandoutNobel
Stereoselective Synthesis of the Side Chains of Mycolactones A and B Featuring Stepwise Double Substitutions of 1,1‐Dibromo‐1‐alkenes
2006 StandoutNobel
A Catalytic Asymmetric 6 π Electrocyclization: Enantioselective Synthesis of 2‐Pyrazolines
2009 StandoutNobel
Copper(I)‐Catalyzed Cycloaddition of Organic Azides and 1‐Iodoalkynes
2009 StandoutNobel
The PtdIns(3,4)P2 phosphatase INPP4A is a suppressor of excitotoxic neuronal death
2010 StandoutNatureNobel
Progress and challenges in translating the biology of atherosclerosis
2011 StandoutNature
The PI3K Pathway in Human Disease
2017 Standout
Cholesterol Efflux Capacity, High-Density Lipoprotein Function, and Atherosclerosis
2011 Standout
Integrins
2002 Standout
Binding Site Detection and Druggability Index from First Principles
2009
Asymmetric 1,3-Dipolar Cycloaddition Reactions
1998 Standout
An efficient copper(II)-catalyzed synthesis of benzothiazoles through intramolecular coupling-cyclization of N-(2-chlorophenyl)benzothioamides
2010
Synthesis of Marine Polyacetylenes Callyberynes A−C by Transition-Metal-Catalyzed Cross-Coupling Reactions to sp Centers
2006
Iron Catalysis in Organic Synthesis
2015 Standout
Two-Dimensional Self-Assembly of Linear Molecular Rods at the Liquid/Solid Interface
2011 StandoutNobel
Copper-Mediated Coupling Reactions and Their Applications in Natural Products and Designed Biomolecules Synthesis
2008 Standout
3d Transition Metals for C–H Activation
2018 Standout
Highly Efficient and Selective Synthesis of Conjugated Triynes and Higher Oligoynes of Biological and Materials Chemical Interest via Palladium-Catalyzed Alkynyl−Alkenyl Coupling
2006 StandoutNobel
Bond Formations between Two Nucleophiles: Transition Metal Catalyzed Oxidative Cross-Coupling Reactions
2011 Standout
PALLADIUM- AND/OR COPPER-MEDIATED CROSS-COUPLING REACTIONS BETWEEN 1-ALKYNES AND VINYL, ARYL, 1-ALKYNYL, 1,2-PROPADIENYL, PROPARGYL AND ALLYLIC HALIDES OR RELATED COMPOUNDS. A REVIEW
1995
Chemistry of Polyvalent Iodine
2008 Standout
Copper-catalyzed decarboxylative cross-coupling of propiolic acids and terminal alkynes
2010
A convenient route to unsymmetrical conjugated diynes
1996
Acetylenkupplungen: eine leistungsfähige Methode für den Aufbau von Molekülen
2000
Strictly “Pair”-Selective and Economical Synthesis of Conjugated Diynes via Pd-Catalyzed Reaction of Terminal Alkynes with 1,1-Dichloroethylene, Elimination with LDA, and Subsequent Transformations
2003 StandoutNobel
Supramolecular Hydrogelators and Hydrogels: From Soft Matter to Molecular Biomaterials
2015 Standout
Single and double asymmetric induction in the cycloaddition of chiral nitrones to achiral and chiral vinylphosphine oxides
1991
Factor Xa Inhibitors: Next-Generation Antithrombotic Agents
2010
An expeditious entry to carbohydrate derived enynes and ene-diynes via Sonogashira coupling of halo-exo-glycals
2004
C−H Activation for the Construction of C−B Bonds
2009 Standout
Magnetic Iron Oxide Nanoparticles: Synthesis, Stabilization, Vectorization, Physicochemical Characterizations, and Biological Applications
2008 Standout
Advances in Transition Metal (Pd,Ni,Fe)-Catalyzed Cross-Coupling Reactions Using Alkyl-organometallics as Reaction Partners
2011 Standout
Discovery of Pyridazinopyridinones as Potent and Selective p38 Mitogen-Activated Protein Kinase Inhibitors
2010
Optically active isoxazolidines via asymmetric cycloaddition reactions of nitrones with alkenes: applications in organic synthesis
1997
The Sonogashira Reaction:  A Booming Methodology in Synthetic Organic Chemistry
2007 Standout
Fragment-guided design of subnanomolar β-lactamase inhibitors active in vivo
2012
Current methods for the synthesis of 2-substituted azoles
2004
Palladium-Catalyzed Alkynylation
2003
Two Dimensional Chiral Networks Emerging from the Aryl−F···H Hydrogen-Bond-Driven Self-Assembly of Partially Fluorinated Rigid Molecular Structures
2008 StandoutNobel
Selected Patented Cross-Coupling Reaction Technologies
2006 Standout
Catalytic Dehydrogenative Cross-Coupling: Forming Carbon−Carbon Bonds by Oxidizing Two Carbon−Hydrogen Bonds
2011 Standout
Aromatic Borylation/Amidation/Oxidation:  A Rapid Route to 5-Substituted 3-Amidophenols
2006
Enantiospecific and diastereoselective synthesis of anti α-hydrazino- and α-amino-β-hydroxyacids through “electrophilic amination” of β-hydroxyesters
1988
Potent, Orally Active GPIIb/IIIa Antagonists Containing a Nipecotic Acid Subunit. Structure−Activity Studies Leading to the Discovery of RWJ-53308
1999
Transition-Metal-Catalyzed C−S, C−Se, and C−Te Bond Formation via Cross-Coupling and Atom-Economic Addition Reactions
2011 Standout
Applications of aliphatic unsaturated non-proteinogenic α-H-α-amino acids
2000
A Field Guide to Foldamers
2001 Standout
Chemicals from Alkynes with Palladium Catalysts
2013
First total synthesis of the brominated polyacetylenes (+)-diplyne A and D: proof of absolute configuration
2004
Aerobic Copper-Catalyzed Organic Reactions
2013 Standout
Click Chemistry: Diverse Chemical Function from a Few Good Reactions
2001 StandoutNobel
Comprehensive Survey of Combinatorial Library Synthesis:  2005
2006
Recent Advances in Electrocatalytic Hydrogen Evolution Using Nanoparticles
2019 Standout
New Chiral Phosphorus Ligands for Enantioselective Hydrogenation
2003 Standout
Natural and Synthetic Small Boron-Containing Molecules as Potential Inhibitors of Bacterial and Fungal Quorum Sensing
2010
The Combinatorial Synthesis of Bicyclic Privileged Structures or Privileged Substructures
2003 Standout
Recent Advances in Efficient and Selective Synthesis of Di-, Tri-, and Tetrasubstituted Alkenes via Pd-Catalyzed Alkenylation−Carbonyl Olefination Synergy
2008 StandoutNobel
Advances in Synthetic Applications of Hypervalent Iodine Compounds
2016 Standout
Metal-catalyzed coupling reactions on an olefin template: the total synthesis of Bupleurynol
2003
Iron-catalyzed synthesis of heterocycles
2014
Applications of Palladium-Catalyzed C–N Cross-Coupling Reactions
2016 Standout
The Enantiospecific Synthesis of an Isoxazoline. A RGD Mimic Platelet GPIIb/IIIa Antagonist
1997
Diastereofacial selectivity in intermolecular nitrone cycloadditions to chiral allyl ethers. Application to Chiral Synthesis of Coniine
1992
Nickel-Catalyzed Oxidative Coupling Reactions of Two Different Terminal Alkynes Using O2 as the Oxidant at Room Temperature: Facile Syntheses of Unsymmetric 1,3-Diynes
2008
The diastereoselectivity of intermolecular nitrone cycloaddition to chiral allyl derivatives
1991
Stereoselective hydrogenation via dynamic kinetic resolution
1989 StandoutNobel
Iron phthalocyanine as an efficient and versatile catalyst for N-alkylation of heterocyclic amines with alcohols: one-pot synthesis of 2-substituted benzimidazoles, benzothiazoles and benzoxazoles
2013
Total synthesis of (+)-monomorine I via nitrone cycloaddition route
1991
A New, Iterative Strategy for the Synthesis of Unsymmetrical Polyynes:  Application to the Total Synthesis of 15,16-Dihydrominquartynoic Acid
2004
Rhodium-Catalyzed C−C Bond Formation via Heteroatom-Directed C−H Bond Activation
2009 Standout
Rearrangement of Nα-Protected l-Asparagines with Iodosobenzene Diacetate. A Practical Route to β-Amino-l-alanine Derivatives
1997
A Medicinal Chemist’s Guide to Molecular Interactions
2010 Standout
Bulky Trialkylsilyl Acetylenes in the Cadiot−Chodkiewicz Cross-Coupling Reaction
2002
Platelet Glycoprotein IIb-IIIa Antagonists as Prototypical Integrin Blockers:  Novel Parenteral and Potential Oral Antithrombotic Agents
2000
Synopsis of Some Recent Tactical Application of Bioisosteres in Drug Design
2011 Standout
Energetics of Displacing Water Molecules from Protein Binding Sites: Consequences for Ligand Optimization
2009

Works of John Wityak being referenced

Discovery and initial SAR of imidazoquinoxalines as inhibitors of the Src-family kinase p56Lck
2002
Discovery and initial SAR of 2-amino-5-carboxamidothiazoles as inhibitors of the Src-family kinase p56Lck
2003
Discovery of 2-amino-heteroaryl-benzothiazole-6-anilides as potent p56lck inhibitors
2003
Bisbenzamidine isoxazoline derivatives as factor Xa inhibitors
1997
Synthesis of 1,3-Diynes Using Palladium-Copper Catalysis
1991
N-Acylthiadiazolines, a New Class of Liver X Receptor Agonists with Selectivity for LXRβ
2007
Orally Active Isoxazoline GPIIb/IIIa Antagonists
1998
Discovery of Potent Isoxazoline Glycoprotein IIb/IIIa Receptor Antagonists
1997
5-Cyanopyrimidine Derivatives as a Novel Class of Potent, Selective, and Orally Active Inhibitors of p38α MAP Kinase
2005
A 1,3-dipolar cycloaddition route to the 3(R)- and 3(S)-hydroxy-2(S)-arginines
1987
Isoxazolines as Potent Antagonists of the Integrin αvβ3
1999
Synthesis of Thrombin Inhibitor DuP 714
1995
Section Review: Cardiovascular & Renal: Glycoprotein IIb/IIIa antagonists
1996
Biosynthesis of streptothricin F
1991
Rankless by CCL
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