Citation Impact
Citing Papers
Expanded therapeutic potential in activity space of next-generation 5-nitroimidazole antimicrobials with broad structural diversity
2013 StandoutNobel
SuFEx-enabled, agnostic discovery of covalent inhibitors of human neutrophil elastase
2019 StandoutNobel
Sulfur [ 18 F]Fluoride Exchange Click Chemistry Enabled Ultrafast Late-Stage Radiosynthesis
2021 StandoutNobel
Diversity oriented clicking delivers β-substituted alkenyl sulfonyl fluorides as covalent human neutrophil elastase inhibitors
2022 StandoutNobel
Bioorthogonal Chemistry: Fishing for Selectivity in a Sea of Functionality
2009 StandoutNobel
Multiwfn: A multifunctional wavefunction analyzer
2011 Standout
“On Water”: Unique Reactivity of Organic Compounds in Aqueous Suspension
2005 StandoutNobel
Noxious compounds activate TRPA1 ion channels through covalent modification of cysteines
2007 StandoutNatureNobel
Modular click chemistry libraries for functional screens using a diazotizing reagent
2019 StandoutNatureNobel
The capsaicin receptor: a heat-activated ion channel in the pain pathway
1997 StandoutNatureNobel
Mechanically bonded macromolecules
2009 StandoutNobel
Biocompatible Carbon Nanotubes Generated by Functionalization with Glycodendrimers
2008 StandoutNobel
A Stepwise Huisgen Cycloaddition Process: Copper(I)-Catalyzed Regioselective “Ligation” of Azides and Terminal Alkynes
2002 StandoutNobel
Oncogenic Mutations Counteract Intrinsic Disorder in the EGFR Kinase and Promote Receptor Dimerization
2012 StandoutNobel
Click Chemistry: Diverse Chemical Function from a Few Good Reactions
2001 StandoutNobel
Efficiency and Fidelity in a Click‐Chemistry Route to Triazole Dendrimers by the Copper(I )‐Catalyzed Ligation of Azides and Alkynes
2004 StandoutNobel
Synthesis and Microcontact Printing of Dual End‐Functionalized Mucin‐like Glycopolymers for Microarray Applications
2009 StandoutNobel
AutoDock4 and AutoDockTools4: Automated docking with selective receptor flexibility
2009 Standout
A Light‐Stimulated Molecular Switch Driven by Radical–Radical Interactions in Water
2011 StandoutNobel
Click Chemistry In Situ: Acetylcholinesterase as a Reaction Vessel for the Selective Assembly of a Femtomolar Inhibitor from an Array of Building Blocks
2002 StandoutNobel
SuFEx‐Based Synthesis of Polysulfates
2014 StandoutNobel
Organic Switches for Surfaces and Devices
2012 StandoutNobel
Impact of EGFR point mutations on the sensitivity to gefitinib: Insights from comparative structural analyses and molecular dynamics simulations
2006
Reactivity of Biarylazacyclooctynones in Copper-Free Click Chemistry
2012 StandoutNobel
Oxime-assisted Acetylcholinesterase Catalytic Scavengers of Organophosphates That Resist Aging
2011 StandoutNobel
Sulfur(VI) Fluoride Exchange (SuFEx): Another Good Reaction for Click Chemistry
2014 StandoutNobel
AutoDock Vina: Improving the speed and accuracy of docking with a new scoring function, efficient optimization, and multithreading
2009 Standout
SuFEx‐Based Polysulfonate Formation from Ethenesulfonyl Fluoride–Amine Adducts
2017 StandoutNobel
Copper(I)-Catalyzed Synthesis of Azoles. DFT Study Predicts Unprecedented Reactivity and Intermediates
2004 StandoutNobel
Enantioselective synthesis of the optical isomers of broad-spectrum orally active antifungal azoles, Sch 42538 and Sch 45012
1994
Adjustable Receptor Based on a [3]Rotaxane Whose Two Threaded Rings Are Rigidly Attached to Two Porphyrinic Plates: Synthesis and Complexation Studies
2009 StandoutNobel
SuFEx Click Chemistry Enabled Late-Stage Drug Functionalization
2018 StandoutNobel
Fluorine in Pharmaceutical Industry: Fluorine-Containing Drugs Introduced to the Market in the Last Decade (2001–2011)
2013 Standout
Self-Assembled Monolayers of Thiolates on Metals as a Form of Nanotechnology
2005 Standout
Pillar[5]arene as a Co-Factor in Templating Rotaxane Formation
2013 StandoutNobel
Multidimensional SuFEx Click Chemistry: Sequential Sulfur(VI) Fluoride Exchange Connections of Diverse Modules Launched From An SOF4 Hub
2017 StandoutNobel
Cooperative capture synthesis: yet another playground for copper-free click chemistry
2016 StandoutNobel
Development of a Bioorthogonal and Highly Efficient Conjugation Method for Quantum Dots Using Tetrazine−Norbornene Cycloaddition
2010 StandoutNobel
A Liquid‐Crystalline Bistable [2]Rotaxane
2007 StandoutNobel
Docking and scoring in virtual screening for drug discovery: methods and applications
2004 Standout
Cooperative Reactivity in an Extended-Viologen-Based Cyclophane
2016 StandoutNobel
Chemical space as a source for new drugs
2010
Biocompatible SuFEx Click Chemistry: Thionyl Tetrafluoride (SOF4)‐Derived Connective Hubs for Bioconjugation to DNA and Proteins
2019 StandoutNobel
Dual-Controlled Nanoparticles Exhibiting AND Logic
2009 StandoutNobel
Analysis of HIV Wild-Type and Mutant Structures via in Silico Docking against Diverse Ligand Libraries
2007
Click-Chemie: diverse chemische Funktionalität mit einer Handvoll guter Reaktionen
2001 StandoutNobel
Mono N-arylation of piperazine(III): metal-catalyzed N-arylation and its application to the novel preparations of the antifungal posaconazole and its advanced intermediate
2002
Click Chemistry: Diverse Chemical Function from a Few Good Reactions
2001 StandoutNobel
Mechanism and Scope of Base‐Controlled Catalyst‐Free N‐Arylation of Amines with Unactivated Fluorobenzenes
2016 StandoutNobel
A Heck–Matsuda Process for the Synthesis of β‐Arylethenesulfonyl Fluorides: Selectively Addressable Bis‐electrophiles for SuFEx Click Chemistry
2016 StandoutNobel
SK&F 96365, a novel inhibitor of receptor-mediated calcium entry
1990
Synthesis and Late-Stage Functionalization of Complex Molecules through C–H Fluorination and Nucleophilic Aromatic Substitution
2014
Acid−Base Actuation of [c2]Daisy Chains
2009 StandoutNobel
Arylfluorosulfates Inactivate Intracellular Lipid Binding Protein(s) through Chemoselective SuFEx Reaction with a Binding Site Tyr Residue
2016 StandoutNobel
The GAMESS-UK electronic structure package: algorithms, developments and applications
2005
Mechanical Bond-Induced Radical Stabilization
2012 StandoutNobel
Second-Generation Difluorinated Cyclooctynes for Copper-Free Click Chemistry
2008 StandoutNobel
Sulfur(VI) Fluoride Exchange (SuFEx)-Enabled High-Throughput Medicinal Chemistry
2020 StandoutNobel
A New Portal to SuFEx Click Chemistry: A Stable Fluorosulfuryl Imidazolium Salt Emerging as an “F−SO2+” Donor of Unprecedented Reactivity, Selectivity, and Scope
2017 StandoutNobel
Sequential mono-N-arylation of piperazine nitrogens. Part 1: A simplified method and its application to the preparation of a key N,N′-biaryl piperazine antifungal intermediate
1999
Works of Jan Heeres being referenced
Inhibition and substrate recognition – a computational approach applied to HIV protease
2003
Evolution of anti-HIV drug candidates. Part 3: diarylpyrimidine (DAPY) analogues
2001
Antimycotic azoles. 7. Synthesis and antifungal properties of a series of novel triazol-3-ones
1984
Conazoles
2010
Preparation and antimycotic properties of derivatives of 1-phenethylimidazole
1969
Antimycotic azoles. 6. Synthesis and antifungal properties of terconazole, a novel triazole ketal
1983
SYNOPSIS: SYNthesize and OPtimize System in Silico
2003
Antimycotic imidazoles. Part 4. Synthesis and antifungal activity of ketoconazole, a new potent orally active broad-spectrum antifungal agent
1979