Citation Impact
Citing Papers
Diversity oriented clicking delivers β-substituted alkenyl sulfonyl fluorides as covalent human neutrophil elastase inhibitors
2022 StandoutNobel
Pharmacology of AMPA/Kainate Receptor Ligands and Their Therapeutic Potential in Neurological and Psychiatric Disorders
2000
In situ click chemistry generation of cyclooxygenase-2 inhibitors
2017 Standout
Oral Torsemide in Patients With Chronic Congestive Heart Failure: Effects on Body Weight, Edema, and Electrolyte Excretion
1994
Methyl 2‐[bis(acetyl)ethenyl]aminopropenoate in the synthesis of heterocyclic systems
1997
Carbonic anhydrase inhibitors: Valdecoxib binds to a different active site region of the human isoform II as compared to the structurally related cyclooxygenase II ‘selective’ inhibitor celecoxib
2005
DARPP-32 knockout mice exhibit impaired reversal learning in a discriminated operant task
2000 StandoutNobel
Persistent kallikrein 5 activation induces atopic dermatitis-like skin architecture independent of PAR2 activity
2017 StandoutNobel
Contribution of platelets to tumour metastasis
2011 Standout
2009 Focused Update Incorporated Into the ACC/AHA 2005 Guidelines for the Diagnosis and Management of Heart Failure in Adults
2009 Standout
The adolescent brain and age-related behavioral manifestations
2000 Standout
Synthesis and biological evaluation of substituted 2-sulfonyl-phenyl-3-phenyl-indoles: a new series of selective COX-2 inhibitors
2003
Anti-Inflammatory Drugs in the 21st Century
2007
Nitric Oxide and Peroxynitrite in Health and Disease
2007 Standout
Overexpression of cyclooxygenase-2 correlates with advanced stages of colorectal cancer
2002
Screening of the Pan-African Natural Product Library Identifies Ixoratannin A-2 and Boldine as Novel HIV-1 Inhibitors
2015 StandoutNobel
Swelling of glial cells in lactacidosis and by glutamate: significance of Cl—-transport
1993
Inflammation and Colon Cancer
2010 Standout
1,2,4-Triazole derivatives as transient inactivators of kallikreins involved in skin diseases
2013
Tissue Kallikrein Inhibitors Based on the Sunflower Trypsin Inhibitor Scaffold – A Potential Therapeutic Intervention for Skin Diseases
2016 StandoutNobel
Psychosis as a State of Aberrant Salience: A Framework Linking Biology, Phenomenology, and Pharmacology in Schizophrenia
2002 Standout
Role of Oxidative Modifications in Atherosclerosis
2004 Standout
Carbonic anhydrase inhibitors. Inhibition of the prokariotic beta and gamma-class enzymes from Archaea with sulfonamides
2004
Carbonic anhydrases: novel therapeutic applications for inhibitors and activators
2008 Standout
Protein Kinase A-mediated Phosphorylation of Serine 357 of the Mouse Prostacyclin Receptor Regulates Its Coupling to Gs-, to Gi-, and to Gq-coupled Effector Signaling
2001
Direct transition metal-catalyzed functionalization of heteroaromatic compounds
2007 Standout
Sulpiride antagonizes the biphasic locomotor effects of quinpirole in weanling rats
1995
Selective COX-2 inhibitors. Part 1: Synthesis and biological evaluation of phenylazobenzenesulfonamides
2006
Microenvironmental regulation of metastasis
2008 Standout
Dopaminergic Supersensitivity in G Protein-Coupled Receptor Kinase 6-Deficient Mice
2003 StandoutNobel
Seven-transmembrane receptors
2002 StandoutNobel
Transition‐Metal‐Catalyzed Direct Arylation of (Hetero)Arenes by CH Bond Cleavage
2009 Standout
Dopamine in Motivational Control: Rewarding, Aversive, and Alerting
2010 Standout
DAD1- and DAD2-like agonist effects on motor activity of C57 mice: Differences compared to rats
1997
Platelet–cancer interactions: mechanisms and pharmacology of tumour cell‐induced platelet aggregation
2004
The involvement of nucleus accumbens dopamine in appetitive and aversive motivation
1994
Protein Kinase A-mediated Phosphorylation of the β2-Adrenergic Receptor Regulates Its Coupling to Gs and Gi
2002 StandoutNobel
Rigid‐Strut‐Containing Crown Ethers and [2]Catenanes for Incorporation into Metal–Organic Frameworks
2009 StandoutNobel
Antiplatelet therapy: in search of the 'magic bullet'
2003
Asymmetric 1,3-Dipolar Cycloaddition Reactions
1998 Standout
Click Chemistry for Drug Development and Diverse Chemical–Biology Applications
2013 Standout
ACC/AHA 2005 Guideline Update for the Diagnosis and Management of Chronic Heart Failure in the Adult
2005 Standout
Over One Hundred Peptide-Activated G Protein-Coupled Receptors Recognize Ligands with Turn Structure
2005
Solid-Phase Intramolecular N-Acyliminium Pictet−Spengler Reactions as Crossroads to Scaffold Diversity
2004 StandoutNobel
Preparation of inclusion complex of piroxicam with cyclodextrin by using supercritical carbon dioxide
2008
Synthesis, Characterization, Cytotoxic Activities, and DNA-Binding Studies of Ternary Copper(II) Complexes with New Coumarin Derivatives
2010
Carboranyl Substituted Siloxanes and Octasilsesquioxanes: Synthesis, Characterization, and Reactivity
2008
A novel strapped porphyrin receptor for molecular recognition
2003
Synthesis of novel 1,2,4-thiadiazinane 1,1-dioxidesviathree component SuFEx type reaction
2018
Efficient and highly regioselective direct C-2 arylation of azoles, including free (NH)-imidazole, -benzimidazole and -indole, with aryl halides
2006
Conjugate systems in the construction of heterocycles and quaternary stereocenters
2007
The Asymmetric Intramolecular Heck Reaction in Natural Product Total Synthesis
2003 Standout
Synthesis of Novel Tricyclic Pyrimido[4,5-b][1,4]benzothiazepines via Bischler−Napieralski-Type Reactions
2005
Regiocontrolled Synthesis of 1,2‐Diaryl‐1H‐imidazoles by Palladium‐ and Copper‐Mediated Direct Coupling of 1‐Aryl‐1H‐imidazoles with Aryl Halides under Ligandless Conditions
2005
Phosphine Organocatalysis
2018 Standout
Occurrence, Biogenesis, and Synthesis of Biologically Active Carbazole Alkaloids
2012 Standout
Chromone: A Valid Scaffold in Medicinal Chemistry
2014 Standout
Review: A History of Cyclodextrins
2014 Standout
Toward the First Class of Suicide Inhibitors of Kallikreins Involved in Skin Diseases
2014
Alkyl 2‐(2‐benzoyl‐2‐ethoxycarbonyl‐1‐ethenyl)amino‐3‐dimethylaminopropenoates in the synthesis of heterocyclic systems
1997
Metal-Catalyzed Decarboxylative C–H Functionalization
2017 Standout
Copper-Catalyzed Synthesis of Mixed Alkyl Aryl Phosphonates
2014 StandoutNobel
The synthesis and transformations of substituted 2-hydroxy-3-dimethylaminopropenoates. The preparation of condensed 3-hydroxypyran-2-ones
1998
Aryl−Aryl Bond Formation by Transition-Metal-Catalyzed Direct Arylation
2007 Standout
Deciphering the Mechanism of Carbonic Anhydrase Inhibition with Coumarins and Thiocoumarins
2009
Transition-Metal-Catalyzed C−S, C−Se, and C−Te Bond Formation via Cross-Coupling and Atom-Economic Addition Reactions
2011 Standout
Asymmetric thermal reactions with oppolzer's camphor sultam
1993
Rational Tuning of Fluorobenzene Probes for Cysteine‐Selective Protein Modification
2018 StandoutNobel
Oxidative Stress: An Essential Factor in the Pathogenesis of Gastrointestinal Mucosal Diseases
2014 Standout
Synthetic Organic Electrochemical Methods Since 2000: On the Verge of a Renaissance
2017 Standout
A New Strategy toward Fused-Pyridine Heterocyclic Scaffolds: Bischler−Napieralski-type Cyclization, Followed by Sulfoxide Extrusion Reaction
2007
Recent Developments in the Chemistry of Cubic Polyhedral Oligosilsesquioxanes
2010 Standout
Overexpression of cyclooxygenase-2 correlates with advanced stages of colorectal cancer
2002
The synthesis of methyl 2‐(benzyloxycarbonyl)amino‐3‐dimethylaminopropenoate. The synthesis of trisubstituted pyrroles, 3‐amino‐2H‐pyran‐2‐ones, fused 2H‐pyran‐2‐ones and 4H‐pyridin‐4‐ones
1999
The Combinatorial Synthesis of Bicyclic Privileged Structures or Privileged Substructures
2003 Standout
Enzymes of the Cyclooxygenase Pathways of Prostanoid Biosynthesis
2011
TRIPHENYPHOSPHINE-MEDIATED EFFICIENT SYNTHESIS OF FUNCTIONALIZED 2-OXO-2H-CHROMENES
2004
Catalytic Asymmetric Synthesis of Quaternary Carbons Bearing Two Aryl Substituents. Enantioselective Synthesis of 3-Alkyl-3-Aryl Oxindoles by Catalytic Asymmetric Intramolecular Heck Reactions
2003
Advances in Copper Complexes as Anticancer Agents
2013 Standout
Endothelial cell activation by endotoxin involves superoxide/NO‐mediated nitration of prostacyclin synthase and thromboxane receptor stimulation
2003
Metal–Organic Frameworks in Biomedicine
2011 Standout
Definition of a Pharmacophore for Partial Agonists of Serotonin 5-HT3 Receptors
1999
β-Turned Dipeptoids as Potent and Selective CCK1 Receptor Antagonists
2000
Functional Significance of Cell Volume Regulatory Mechanisms
1998 Standout
Role of Monocytes in Atherogenesis
2003
Chemistry and Biology Of Multicomponent Reactions
2012 Standout
Cationic iridacarboranes [3-(arene)-3,1,2-IrC2B9H11]+ and [3-(MeCN)3-3,1,2-IrC2B9H11]+: Synthesis, reactivity, and bonding. Catalysis of oxidative coupling of benzoic acid with alkynes
2015
Electrochemical synthesis of polyhydroxylated aromatic derivatives substituted with mono- and dipyrimidinyl thioethers in aqueous medium
2008
Rhodium-Catalyzed C−C Bond Formation via Heteroatom-Directed C−H Bond Activation
2009 Standout
Synthesis and biological activity of pyrrole, pyrroline and pyrrolidine derivatives with two aryl groups on adjacent positions
2006 Standout
Irreversible Inhibitors of Serine, Cysteine, and Threonine Proteases
2002 Standout
Synthesis of Heterocycles from Alkyl 3-(Dimethylamino)propenoates and Related Enaminones
2004 Standout
Multiple Binding Modes of Inhibitors to Carbonic Anhydrases: How to Design Specific Drugs Targeting 15 Different Isoforms?
2012 Standout
An Efficient Low-Temperature Route to Polycyclic Isoquinoline Salt Synthesis via C−H Activation with [Cp*MCl2]2 (M = Rh, Ir)
2008 Standout
Works of J. Delarge being referenced
Studies of Thiaheterocyclic Derivatives .1. Synthesis and Pharmacological Screening
1984
Dibenzoazepine analogues: the electrophysiological properties of JL3, a potential atypical antidepressant
1996
Terbogrel, a dual-acting agent for thromboxane receptor antagonism and thromboxane synthase inhibition
2000
Effects of JL 3, a putative antidepressant, on rat noradrenergic and serotonergic systems
1999
Study of the Influence of Both Cyclodextrins and L-Lysine on the Aqueous Solubility of Nimesulide; Isolation and Characterization of Nimesulide–L-Lysine–Cyclodextrin Complexes
1997
New Trends in Thromboxane and Prostacyclin Modulators
2000
Evaluation of classical NSAIDs and COX-2 selective inhibitors on purified ovine enzymes and human whole blood
2001
Pharmacological evaluation of the novel thromboxane modulator BM-567 (II/II). Effects of BM-567 on osteogenic sarcoma-cell-induced platelet aggregation
2003
Anxiolytic potential of sulpiride, clozapine and derivatives in the open-field test
1990
Recent Advances in Inducible Cyclooxygenase (COX-2) Inhibition.
2000
Effects of specific dopaminergic agonists and antagonists in the open-field test
1991
Synthesis and Anticonvulsant Activity of 2(3 H )-Benzoxazolone and 2(3 H )-Benzothiazolone Derivatives
1998
Electrooxidation Potential as a Tool in the Early Screening for New Safer Clozapine-like Analogues
2001
Advances in the field of COX-2 inhibition
2002
Recent Advances in the Chemistry of Cholecystokinin Receptor Ligands (Agonists and Antagonists)
1999
Ligand effects in the hydrogenation of methacycline to doxycycline and epi-doxycycline catalysed by rhodium complexes molecular structure of the key catalyst [closo-3,3-(η2,3-C7H7CH2)-3,1,2-RhC2B9H11]
1997
Structure de l'hydrogénosulfate de la {[(chloro-3 phénylamino)-4 pyridyl-3] sulfonyl}-1 éthyl-3 méthyl-1 urée
1980
Recent Advances in Inducible Cyclooxygenase (COX-2) Inhibition.
2000
Thromboxane A2 inhibition: therapeutic potential in bronchial asthma.
2002
New dibenzazepine derivatives with disinhibitory and/or antidepressant potential
1995
6-Substituted 2-Oxo-2H-1-benzopyran-3-carboxylic Acid as a Core Structure for Specific Inhibitors of Human Leukocyte Elastase
1999
Esters and Amides of 6-(Chloromethyl)-2-oxo-2H-1-benzopyran-3-carboxylic Acid as Inhibitors of α-Chymotrypsin: Significance of the “Aromatic” Nature of the Novel Ester-Type Coumarin for Strong Inhibitory Activity
1996
Structures du 11-formyl-5-(4-méthylpipérazin-1-yl)-11H-pyrido[2,3-b][1,5]benzodiazépine et du 6-(4-méthylpipérazin-1-yl)-11-méthyl-11H-pyrido[2,3-b][1,4]benzodiazépine
1991
Structure du maléate de méthyl-1 (pyrido[2,3-f][1,5]benzoxazépinyl-5) 1H+ pipérazinium
1987
Diuretic activity of torasemide and furosemide in chronic heart failure: A comparative double blind cross-over study
1986
4H-1,2,4-Pyridothiadiazine 1,1-Dioxides and 2,3-Dihydro-4H-1,2,4-pyridothiadiazine 1,1-Dioxides Chemically Related to Diazoxide and Cyclothiazide as Powerful Positive Allosteric Modulators of (R/S)-2-Amino-3-(3-hydroxy-5-methylisoxazol-4-yl)propionic Acid Receptors: Design, Synthesis, Pharmacology, and Structure−Activity Relationships
1998
Torasemide inhibits NaCl reabsorption in the thick ascending limb of the loop of Henle
1986
Structure de la clothiapine
1987
Evaluation of the Inhibitory Activity on Serine and Aspartic Proteases of 4-Amino-4H-1,2,4-triazole and 5-Aminothiazole Derivatives Structurally Related to β-Lactam Antibiotics
1993