Citation Impact

Citing Papers

In Vivo Imaging of Quantum Dots Encapsulated in Phospholipid Micelles
2002 StandoutScience
The Human Polyomavirus, JCV, Uses Serotonin Receptors to Infect Cells
2004 Science
Signaling from β1- and β2-adrenergic receptors is defined by differential interactions with PDE4
2008 StandoutNobel
BIMU1 Increases Associative Memory in Rats by Activating 5-HT 4 Receptors
1997
The effects of GR127935, a putative 5-HT1D receptor antagonist, on brain 5-HT metabolism, extracellular 5-HTT concentration and behaviour in the guinea pig
1995
Differential desensitization of μ‐ and δ‐ opioid receptors in selected neural pathways following chronic morphine treatment
1996
The Retinal Pigment Epithelium in Visual Function
2005 Standout
The 5-Hydroxytryptamine(1A) Receptor Is Stably Palmitoylated, and Acylation Is Critical for Communication of Receptor with Gi Protein
2004
The distribution of 5-HT1A and 5-HT2A receptor mRNA in human brain
1995
The pharmacology of headache
2000
5-HT2C receptors mediate penile erections in rats: actions of novel and selective agonists and antagonists
1997
Open probability of homomeric murine 5‐HT3A serotonin receptors depends on subunit occupancy
2001
In vivo effects of the 5‐HT6 antagonist SB‐271046 on striatal and frontal cortex extracellular concentrations of noradrenaline, dopamine, 5‐HT, glutamate and aspartate
2000
Molecular, pharmacological and functional diversity of 5-HT receptors
2002 Standout
Allosteric modulation of 5-HT3 receptors: focus on alcohols and anaesthetic agents
1996
The interaction of trichloroethanol with murine recombinant 5‐HT3 receptors
1995
Ability of 5‐HT4 receptor ligands to modulate rat striatal dopamine release in vitro and in vivo
1996
A receptor autoradiographic and in situ hybridization analysis of the distribution of the 5‐ht7 receptor in rat brain
1996
Descending control of pain
2002 Standout
Vascularized and functional human liver from an iPSC-derived organ bud transplant
2013 StandoutNature
Cyclic nucleotide phosphodiesterase (PDE) superfamily: A new target for the development of specific therapeutic agents
2005 Standout
Localization of 5-HT6 receptors at the plasma membrane of neuronal cilia in the rat brain
2000
Distinct Profiles of α7 nAChR Positive Allosteric Modulation Revealed by Structurally Diverse Chemotypes
2007
Cyclic Nucleotide Phosphodiesterases: Molecular Regulation to Clinical Use
2006 Standout
Actions of general anaesthetics on 5‐HT3 receptors in N1E‐115 neuroblastoma cells
1996
Characterization of the First Potent and Selective PDE9 Inhibitor Using a cGMP Reporter Cell Line
2005
Selective labelling of 5-HT7 receptor recognition sites in rat brain using [3H]5-carboxamidotryptamine
1998
A role for 5-ht6 receptors in retention of spatial learning in the Morris water maze
2001
Identification of 5‐hydroxytryptamine receptors positively coupled to adenylyl cyclase in rat cultured astrocytes
1997
Characterization of [3H]GR 113808 binding to 5-HT4 receptors in brain tissues from patients with neurodegenerative disorders
1995
Dual effect of serotonin on formalin-induced nociception in the rat spinal cord
1996
ChEMBL: a large-scale bioactivity database for drug discovery
2011 Standout
Differential Distribution of [ 3 H]Sumatriptan Binding Sites (5-HT 1B , 5-HT 1D and 5-HT 1F Receptors) in Human Brain: Focus on Brainstem and Spinal Cord
1997
5-HT 4 Receptors Improve Social Olfactory Memory in the Rat
1997
Localization of agonist and competitive antagonist binding sites on nicotinic acetylcholine receptors
2000
Identification of an Allosteric Binding Site for Zn2+on the β2 Adrenergic Receptor
2002 StandoutNobel
The Pharmacological and Functional Characteristics of the Serotonin 5-HT3A Receptor Are Specifically Modified by a 5-HT3B Receptor Subunit
1999
The 5-HT5A serotonin receptor is expressed predominantly by astrocytes in which it inhibits cAMP accumulation: A mechanism for neuronal suppression of reactive astrocytes
1996
Mechanisms of Actions of Inhaled Anesthetics
2003 Standout
Evidence that hypophagia induced by d-fenfluramine and d-norfenfluramine in the rat is mediated by 5-HT2C receptors
2001
Antisense Oligonucleotide‐Induced Reduction in 5‐Hydroxytryptamine7 Receptors in the Rat Hypothalamus Without Alteration in Exploratory Behaviour or Neuroendocrine Function
1998
Vertebrate Smoothened functions at the primary cilium
2005 StandoutNature
Neurotransmitter Release at the Thalamocortical Synapse Instructs Barrel Formation But Not Axon Patterning in the Somatosensory Cortex
2012 StandoutNobel
Indigenous Bacteria from the Gut Microbiota Regulate Host Serotonin Biosynthesis
2015 Standout
Cultured astrocytes express messenger RNA for multiple serotonin receptor subtypes, without functional coupling of 5-HT1 receptor subtypes to adenylyl cyclase
1998
The Non-Antiemetic Uses of Serotonin 5-HT3 Receptor Antagonists
1997
Distribution of the 5-hydroxytryptamine2C receptor protein in adult rat brain and spinal cord determined using a receptor-directed antibody: Effect of 5,7-dihydroxytryptamine
1997
The behavioral pharmacology of hallucinogens
2007
In vivo cancer targeting and imaging with semiconductor quantum dots
2004 Standout
Screening of the Pan-African Natural Product Library Identifies Ixoratannin A-2 and Boldine as Novel HIV-1 Inhibitors
2015 StandoutNobel
Characterization of a postjunctional 5-HT receptor mediating relaxation of guinea-pig isolated ileum
1995
Quantum dot bioconjugates for imaging, labelling and sensing
2005 Standout
Calcitonin Gene–Related Peptide Receptor Antagonist BIBN 4096 BS for the Acute Treatment of Migraine
2004 Standout
Serotonin receptors and their role in the pathophysiology and therapy of irritable bowel syndrome
2014
5-HT Receptor Classification and Nomenclature: Towards a Harmonization with the Human Genome
1997
Expression of serotonin receptor mRNAs in blood vessels
1995
Purification of 5‐hydroxytryptamine3 receptors from porcine brain
1997
Serotonin2C receptors tonically suppress the activity of mesocortical dopaminergic and adrenergic, but not serotonergic, pathways: A combined dialysis and electrophysiological analysis in the rat
2000
Distribution of serotonin 2A, 2C and 3 receptor mRNA in spinal cord and medulla oblongata
2001
Agonist and antagonist actions of antipsychotic agents at 5-HT1A receptors: a []GTPγS binding study
1998
Migraine — Current Understanding and Treatment
2002 Standout
Neurobiology of Depression
2002 Standout
Ligand-Gated Ion Channels
2001
Selective blockade of serotonin2C/2B receptors enhances dopamine release in the rat nucleus accumbens
1998
Localization of 5-ht5A receptor-like immunoreactivity in the rat brain
2000
Effects of the 5-HT1D receptor antagonist GR127935 on extracellular levels of 5-HT in the guinea-pig frontal cortex as measured by microdialysis
1995
Characterization and distribution of putative 5‐ht7receptors in guinea‐pig brain
1995
5-HT6 receptor antagonists: lead optimisation and biological evaluation of N-aryl and N-heteroaryl 4-amino-benzene sulfonamides
2001
Serotonergic modulation of hyperpolarization‐activated current in acutely isolated rat dorsal root ganglion neurons
1999
Neural Science: A Century of Progress and the Mysteries that Remain
2000 StandoutNobel
Functional mapping and annotation of genetic associations with FUMA
2017 Standout
A review of central 5-HT receptors and their function
1999 Standout
The induction of pain: an integrative review
1999
The structural basis of function in Cys-loop receptors
2010
Characterization of [125I]‐SB‐258585 binding to human recombinant and native 5‐HT6 receptors in rat, pig and human brain tissue
2000
[3H]Sumatriptan binding sites in human brain: regional-dependent labelling of 5-HT1D and 5-HT1F receptors
1996
Differential pharmacology between the guinea‐pig and the gorilla 5‐HT1D receptor as probed with isochromans (5‐HT1D‐selective ligands)
1999
Polymorphic Cytochrome P450 2D6: Humanized Mouse Model and Endogenous Substrates
2004
Characterization of SB‐271046: A potent, selective and orally active 5‐HT6 receptor antagonist
2000
Modified 5-HT3A receptor function by co-expression of alternatively spliced human 5-HT3A receptor isoforms
2000
Valvular Heart Disease in Patients Taking Pergolide
2002
5-HT3 receptors and neurotransmitter release in the CNS: a nerve ending story?
2000
Crystal structure of an ACh-binding protein reveals the ligand-binding domain of nicotinic receptors
2001 StandoutNature
Mapping of 5-HT-moduline binding sites in guinea-pig brain by film and digital autoradiography
1998
P2X1 and P2X3 receptors form stable trimers: a novel structural motif of ligand-gated ion channels
1998
Ultrastructural localization of 5-hydroxytryptamine1A receptors in the rat brain
1996
Discriminative stimulus properties of the novel serotonin (5-HT)2C receptor agonist, RO60-0175: a pharmacological analysis
1999
Desperately seeking subunits: are native 5-HT3 receptors really homomeric complexes?
1998
Autoradiographic mapping of serotonin 5-HT1A, 5-HT1D, 5-HT2A and 5-HT3 receptors in the aged human spinal cord
1996
Molecular Neurobiology and Genetics: Investigation of Neural Function and Dysfunction
1998
High hopes: can molecular electronics realise its potential?
2012 StandoutNobel
Phosphodiesterase: overview of protein structures, potential therapeutic applications and recent progress in drug development
2005
Nociceptors: the sensors of the pain pathway
2010 StandoutNobel
Pindolol‐insensitive [3H]‐5‐hydroxytryptamine binding in the rat hypothalamus; identity with 5‐hydroxytryptamine7 receptors
1999
Serotonin elevates the c-wave of the electroretinogram of the rabbit eye by increasing the transepithelial potential
1997
8-OH-DPAT-induced Spontaneous Tail-flicks in the Rat are Facilitated by the Selective Serotonin (5-HT) 2C Agonist, RO 60-0175: Blockade of its Actions by the Novel 5-HT 2C Receptor Antagonist SB 206,553
1997
Uropathic Observations in Mice Expressing a Constitutively Active Point Mutation in the 5-HT3AReceptor Subunit
2004 StandoutNobel
Pharmacological characterization of the apparent splice variants of the murine 5-HT3 R-A subunit expressed in Xenopus laevis oocytes
1994
Allosteric Modulators of the α7 Nicotinic Acetylcholine Receptor
2008
The transmitter-gated channels: a range of receptor types and structures
1996
β-Arrestin–Mediated Localization of Smoothened to the Primary Cilium
2008 StandoutScienceNobel
Novel Aza-analogous Ergoline Derived Scaffolds as Potent Serotonin 5-HT6 and Dopamine D2 Receptor Ligands.
2014
Molecular Physiology of P2X Receptors
2002 Standout
2-Substituted Tryptamines:  Agents with Selectivity for 5-HT6Serotonin Receptors
2000
Cellular and subcellular immunolocalization of the type 3 serotonin receptor in the rat central nervous system
1996
The 5-HT3Subtype of Serotonin Receptor Contributes to Nociceptive Processing via a Novel Subset of Myelinated and Unmyelinated Nociceptors
2002 StandoutNobel
Marine Indole Alkaloids: Potential New Drug Leads for the Control of Depression and Anxiety
2010 Standout
MOD-1 is a serotonin-gated chloride channel that modulates locomotory behaviour in C. elegans
2000 StandoutNatureNobel
Quantum Dots for Live Cells, in Vivo Imaging, and Diagnostics
2005 StandoutScience
Inactivation of a Serotonin-Gated Ion Channel by a Polypeptide Toxin from Marine Snails
1998 StandoutScienceNobel
μ-Opioid receptor desensitization by β-arrestin-2 determines morphine tolerance but not dependence
2000 StandoutNatureNobel
Generation of Candidate Ligands for Nicotinic Acetylcholine Receptors via in situ Click Chemistry with a Soluble Acetylcholine Binding Protein Template
2012 StandoutNobel
Regulation of Calcitonin Gene-Related Peptide Secretion by a Serotonergic Antimigraine Drug
1999
Spinal and Supraspinal Factors in Human Muscle Fatigue
2001 Standout
Evidence for presynaptic location of inhibitory 5-HT1D\-like autoreceptors in the guinea-pig brain cortex
1996
Advances in the Chemistry of Tetrahydroquinolines
2011 Standout
Characterization of the Serotonin Receptor Mediating Contraction in the Mouse Thoracic Aorta and Signal Pathway Coupling
2001
ACC/AHA 2006 Guidelines for the Management of Patients With Valvular Heart Disease
2006 Standout
Reciprocal autoreceptor and heteroreceptor control of serotonergic, dopaminergic and noradrenergic transmission in the frontal cortex: relevance to the actions of antidepressant agents
2000
Neural Science
2000 StandoutNobel
The Multiplicity of Serotonin Receptors: Uselessly Diverse Molecules or an Embarrassment of Riches?
2000
Two Parallel Signaling Pathways Couple 5HT1AReceptors to N- and L-Type Calcium Channels in C-Like Rat Dorsal Root Ganglion Cells
1997
Immuno-localization of serotonin 5-HT6 receptor-like material in the rat central nervous system
1997
Influence of Life Stress on Depression: Moderation by a Polymorphism in the 5-HTT Gene
2003 StandoutScience
Excessive Activation of Serotonin (5-HT) 1B Receptors Disrupts the Formation of Sensory Maps in Monoamine Oxidase A and 5-HT Transporter Knock-Out Mice
2001
Analysis of Biomolecular Interactions Using a Miniaturized Surface Plasmon Resonance Sensor
2002 StandoutNobel
5HT4Receptors Couple Positively to Tetrodotoxin-Insensitive Sodium Channels in a Subpopulation of Capsaicin-Sensitive Rat Sensory Neurons
1997
Therapeutic Potential of Serotonin 5-HT3 Antagonists in Neuropsychiatric Disorders
1995
Study of Ligand−Receptor Interactions by Fluorescence Correlation Spectroscopy with Different Fluorophores:  Evidence That the Homopentameric 5-Hydroxytryptamine Type 3AsReceptor Binds Only One Ligand
1999
Compartmentation of Cyclic Nucleotide Signaling in the Heart
2006
The Combinatorial Synthesis of Bicyclic Privileged Structures or Privileged Substructures
2003 Standout
Serotonin Receptors
2008
The Vanilloid Receptor: A Molecular Gateway to the Pain Pathway
2001 StandoutNobel
Targeting Cell Surface Receptors with Ligand-Conjugated Nanocrystals
2002
5-HT2B receptor-mediated serotonin morphogenetic functions in mouse cranial neural crest and myocardiac cells
1997
Autoradiographic characterization of [ 3 H]-5-HT-moduline binding sites in rodent brain and their relationship to 5-HT 1B  receptors
1997
Cellular and subcellular distribution of the serotonin 5-HT2A receptor in the central nervous system of adult rat
1999
A cell protection screen reveals potent inhibitors of multiple stages of the hepatitis C virus life cycle
2010 StandoutNobel
Applications of Palladium-Catalyzed C–N Cross-Coupling Reactions
2016 Standout
Medicinal Chemistry Driven Approaches Toward Novel and Selective Serotonin 5-HT6Receptor Ligands
2004
DESENSITIZATION OF G PROTEIN–COUPLED RECEPTORS AND NEURONAL FUNCTIONS
2004 StandoutNobel
5-ht6 Receptors as Emerging Targets for Drug Discovery
2000
5HT Increases Excitability of Nociceptor-Like Rat Dorsal Root Ganglion Neurons Via cAMP-Coupled TTX-Resistant Na+Channels
2001
The Binding Site of Aminergic G Protein–Coupled Receptors: The Transmembrane Segments and Second Extracellular Loop
2002
5-HT2AReceptor-Mediated Regulation of Brain-Derived Neurotrophic Factor mRNA in the Hippocampus and the Neocortex
1997
Trafficking of G Protein–Coupled Receptors
2006 StandoutNobel
Natural compounds boldine and menthol are antagonists of human 5‐HT3 receptors: implications for treating gastrointestinal disorders
2014
5-Chloro-N-(4-methoxy-3-piperazin-1-yl- phenyl)-3-methyl-2-benzothiophenesulfon- amide (SB-271046):  A Potent, Selective, and Orally Bioavailable 5-HT6 Receptor Antagonist
1999
α7-Nicotinic Acetylcholine Receptor Agonists for Cognitive Enhancement in Schizophrenia
2013
The pharmacology and distribution of human 5‐hydroxytryptamine2B (5‐HT2b) receptor gene products: comparison with 5‐HT2a and 5‐HT2c receptors
1995
Serotonin (5-HT) and pain: A reappraisal of its role in the light of receptor multiplicity
1995
Physiology of Microglia
2011 Standout
Hallucinogens
2004 Standout

Works of Frank Boess being referenced

5-HT 6 and 5-HT 7 Receptors: Molecular Biology, Functional Correlates and Possible Therapeutic Indications.
1997
Characterization of Ro 04‐6790 and Ro 63‐0563: potent and selective antagonists at human and rat 5‐HT6 receptors
1998
Functional and Radioligand Binding Characterization of Rat 5-HT 6 Receptors Stably Expressed in HEK293 Cells
1997
Interaction of Tryptamine and Ergoline Compounds with Threonine 196 in the Ligand Binding Site of the 5-Hydroxytryptamine6 Receptor
1997
The 5-Hydroxytryptamine6 Receptor-Selective radioligand [3H]Ro 63–0563 Labels 5-Hydroxytryptamine Receptor Binding Sites in Rat and Porcine Striatum
1998
Analysis of the Ligand Binding Site of the 5-HT 3 Receptor Using Site Directed Mutagenesis: Importance of Glutamate 106
1997
Identification of Residues in Transmembrane Regions III and VI that Contribute to the Ligand Binding Site of the Serotonin 5‐HT6 Receptor
1998
Residues in Transmembrane Regions III and VI Contribute to the 5‐ht6 Receptor Ligand Binding Site
1998
The Putative 5‐ht6 Receptor: Localization and Function
1998
Molecular Properties of 5‐Hydroxytryptamine3 Receptor‐Type Binding Sites Purified from NG1O8‐15 Cells
1992
The Novel α7 Nicotinic Acetylcholine Receptor Agonist N-[(3 R)-1-Azabicyclo[2.2.2]oct-3-yl]-7-[2-(methoxy)phenyl]-1-benzofuran-2-carboxamide Improves Working and Recognition Memory in Rodents
2007
EVP-6124, a novel and selective α7 nicotinic acetylcholine receptor partial agonist, improves memory performance by potentiating the acetylcholine response of α7 nicotinic acetylcholine receptors
2011
AR-R 17779 improves social recognition in rats by activation of nicotinic α7 receptors
2004
Investigation of stretching behaviour induced by the selective 5‐HT6 receptor antagonist, Ro 04–6790, in rats
1999
Inhibition of phosphodiesterase 2 increases neuronal cGMP, synaptic plasticity and memory performance
2004
Ultrastructure of the 5‐Hydroxytryptamine3 Receptor
1995
Involvement of 5‐HT6 receptors in nigro‐striatal function in rodents
1998
Molecular biology of 5-HT receptors
1994
The 5-hydroxytryptamine 6 receptor: localisation and function
1998
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