Citation Impact
Citing Papers
Transaminases for the synthesis of enantiopure beta-amino acids
2012
Characterization of a thermostable methylaspartate ammonia lyase from Carboxydothermus hydrogenoformans
2011 StandoutNobel
Organic base-catalyzed stereodivergent synthesis of (R)- and (S)-3-amino-4,4,4-trifluorobutanoic acids
2012
Catalytic Asymmetric Three‐Component Synthesis of Homoallylic Amines
2013 StandoutNobel
Stress-Activated NRF2-MDM2 Cascade Controls Neoplastic Progression in Pancreas
2017
Recent advances in the catalytic asymmetric synthesis of β-amino acids
2010 StandoutNobel
Donor–Acceptor Oligorotaxanes Made to Order
2011 StandoutNobel
‘100 years of peptide synthesis’: ligation methods for peptide and protein synthesis with applications to β‐peptide assemblies*
2005
Synthetic Routes towards Enantiomerically Pure β‐Amino Acids
2003
Enzymatic Synthesis of Enantiopure α‐ and β‐Amino Acids by Phenylalanine Aminomutase‐Catalysed Amination of Cinnamic Acid Derivatives
2009 StandoutNobel
Small-molecule MDM2/X inhibitors and PROTAC degraders for cancer therapy: advances and perspectives
2020
Synthesis and Conformation of Fluorinated β‐Peptidic Compounds
2012
Asymmetric synthesis of 2-alkyl- and 2-aryl-3-aminopropionic acids (β2-amino acids) from (S)-N-acryloyl-5,5-dimethyloxazolidin-2-one SuperQuat derivatives
2004
Engineering of an enantioselective tyrosine aminomutase by mutation of a single active site residue in phenylalanine aminomutase
2010 StandoutNobel
Aminomutases: mechanistic diversity, biotechnological applications and future perspectives
2011 StandoutNobel
Introduction of Fluorine and Fluorine‐Containing Functional Groups
2013 Standout
The C–F bond as a conformational tool in organic and biological chemistry
2010
Stereoselective Fluorination Alters the Geometry of a Cyclic Peptide: Exploration of Backbone‐Fluorinated Analogues of Unguisin A
2014
Evolving Strategies for Protein Synthesis Converge on Native Chemical Ligation
2006 StandoutNobel
Conversion of biomass to selected chemical products
2011 Standout
Biological Functions of Autophagy Genes: A Disease Perspective
2019 Standout
Indolizidine and quinolizidine alkaloids
2005
Foldamers as versatile frameworks for the design and evolution of function
2007
Helices and other secondary structures of β‐ and γ‐peptides
2005
The vicinal F–C–C–F moiety as a tool for influencing peptide conformation
2005
Enantiomerically pure β-phenylalanine analogues from α–β-phenylalanine mixtures in a single reactive extraction step
2009 StandoutNobel
The World of β‐ and γ‐Peptides Comprised of Homologated Proteinogenic Amino Acids and Other Components
2004
Mechanism‐Inspired Engineering of Phenylalanine Aminomutase for Enhanced β‐Regioselective Asymmetric Amination of Cinnamates
2011 StandoutNobel
PROTAC targeted protein degraders: the past is prologue
2022 Standout
In Vitro and In Vivo Enzymatic Formation of Supramolecular Hydrogels Based on Self‐Assembled Nanofibers of a β‐Amino Acid Derivative
2007
N-Linked Glycosylatedβ-Peptides Are Resistant to Degradation by Glycoamidase A
2005
β-Amino acid-containing hybrid peptides—new opportunities in peptidomimetics
2007
Bacterial β-peptidyl aminopeptidases: on the hydrolytic degradation of β-peptides
2007
Solid phase synthesis of peptides containing backbone-fluorinated amino acids
2012
Synthesis and Conformational Analysis of α,β‐Difluoro‐γ‐amino Acid Derivatives
2011
Insight into the mechanism of aminomutase reaction: A case study of phenylalanine aminomutase by computational approach
2013
Engineered Nanoparticles for Drug Delivery in Cancer Therapy
2014 Standout
NF-κB, inflammation, immunity and cancer: coming of age
2018 Standout
β2‐amino acids—syntheses, occurrence in natural products, and components of β‐peptides1,2
2004
Enantioselective synthesis of β2-amino acids using rhodium-catalyzed hydrogenation
2006 StandoutNobel
Ring Expansion Induced by DAST: Synthesis of Substituted 3‐Fluoropiperidines from Prolinols and 3‐Fluoroazepanes from 2‐Hydroxymethylpiperidines
2007
Physiology and Pathophysiology of Carnosine
2013 Standout
Click Chemistry for Drug Development and Diverse Chemical–Biology Applications
2013 Standout
Monofluorination of Organic Compounds: 10 Years of Innovation
2015 Standout
Practical Synthesis of Fluorine-Containing α- and β-Amino Acids: Recipes from Kiev, Ukraine
2009
3d Transition Metals for C–H Activation
2018 Standout
Sequential Deoxyfluorination Approach for the Synthesis of Protected α,β,γ-Trifluoro-δ-amino Acids
2013
Fluorine in Pharmaceutical Industry: Fluorine-Containing Drugs Introduced to the Market in the Last Decade (2001–2011)
2013 Standout
Fluorine and Fluorinated Motifs in the Design and Application of Bioisosteres for Drug Design
2018 Standout
Supramolecular Hydrogelators and Hydrogels: From Soft Matter to Molecular Biomaterials
2015 Standout
Phenylalanine Aminomutase-Catalyzed Addition of Ammonia to Substituted Cinnamic Acids: a Route to Enantiopure α- and β-Amino Acids
2009 StandoutNobel
Hydroamination: Direct Addition of Amines to Alkenes and Alkynes
2008 Standout
Chemical Routes for the Transformation of Biomass into Chemicals
2007 Standout
Efficient Tandem Biocatalytic Process for the Kinetic Resolution of Aromatic β‐Amino Acids
2010 StandoutNobel
Palladium-Catalyzed Anti-Markovnikov Oxidation of Allylic Amides to Protected β-Amino Aldehydes
2014 StandoutNobel
Synthesis of Gly-ψ[(Z)CF═CH]-Phe, a Fluoroalkene Dipeptide Isostere, and Its Incorporation into a Leu-enkephalin Peptidomimetic
2016
Next Generation of Fluorine-Containing Pharmaceuticals, Compounds Currently in Phase II–III Clinical Trials of Major Pharmaceutical Companies: New Structural Trends and Therapeutic Areas
2016 Standout
Folding of Oligoviologens Induced by Radical–Radical Interactions
2014 StandoutNobel
Titanium Enolate Chemistry at the Beginning of the 21st Century
2016
Enantioselective Synthesis of α-Fluoro-β3-amino Esters: Synthesis of Enantiopure, Orthogonally Protected α-Fluoro-β3-lysine
2010
Collagen Structure and Stability
2009 Standout
Free radical fluoroalkylation of terminal alkenes and alkynes with iododifluoromethanesulfonamides
2011
β-Peptidic Peptidomimetics
2008
Electrophilic Trifluoromethylation by Use of Hypervalent Iodine Reagents
2014 Standout
Recent Advances in Stereoselective Synthesis and Application of β-Amino Acids
2009
Functional π-Gelators and Their Applications
2014 Standout
An enantioselective synthesis of β2-amino acid derivatives
2005
Fluorine in Peptides: The Synthesis of α‐Fluoro‐β‐Amino Dipeptides by Direct Deoxofluorination/Rearrangement of N‐Seryl Dipeptides
2012
Biochemical Properties and Crystal Structure of a β-Phenylalanine Aminotransferase from Variovorax paradoxus
2012 StandoutNobel
Supramolecular Helical Systems: Helical Assemblies of Small Molecules, Foldamers, and Polymers with Chiral Amplification and Their Functions
2016 Standout
Synthesis of Optically Active Bifunctional Building Blocks through Enantioselective Copper-Catalyzed Allylic Alkylation Using Grignard Reagents
2007 StandoutNobel
Recent Progress in the in situ Detrifluoroacetylative Generation of Fluoro Enolates and Their Reactions with Electrophiles
2015
Note: Helix or No Helix of β‐Peptides Containing β3hAla(αF) Residues?
2011
Enantioselective Synthesis of α-Fluorinated β2-Amino Acids
2008
Catalytic Asymmetric Synthesis of Unprotected β2-Amino Acids
2021 StandoutNobel
Asymmetric Allylic Alkylation in Combination with Ring-Closing Metathesis for the Preparation of Chiral N-Heterocycles
2010 StandoutNobel
Helical Polymers: Synthesis, Structures, and Functions
2009 Standout
Structural Investigations into the Stereochemistry and Activity of a Phenylalanine-2,3-aminomutase from Taxus chinensis
2014 StandoutNobel
Enantioselective Rhodium Enolate Protonations. A New Methodology for the Synthesis of β2-Amino Acids
2005
Electrophilic S‐Trifluoromethylation of Cysteine Side Chains in α‐ and β‐Peptides: Isolation of Trifluoro‐methylated Sandostatin® (Octreotide) Derivatives
2008
The Path Forward for Biofuels and Biomaterials
2006 StandoutScience
Disulfonimide-Catalyzed Asymmetric Synthesis of β3-Amino Esters Directly from N-Boc-Amino Sulfones
2013 StandoutNobel
Chiral Phosphoric Acid Catalyzed Enantioselective Synthesis of β-Amino-α,α-difluoro Carbonyl Compounds
2011
Organocatalytic Asymmetric Transferhydrogenation of β-Nitroacrylates: Accessing β2-Amino Acids
2008 StandoutNobel
Direct Catalytic Asymmetric Mannich-Type Reaction of α- and β-Fluorinated Amides
2015
Complete Field Guide to Asymmetric BINOL-Phosphate Derived Brønsted Acid and Metal Catalysis: History and Classification by Mode of Activation; Brønsted Acidity, Hydrogen Bonding, Ion Pairing, and Metal Phosphates
2014 Standout
Highly enantioselective rhodium-catalyzed conjugate addition of arylboronic acids to enones at room temperature
2005 StandoutNobel
β-Amino Acid and Amino-Alcohol Conjugation of a Nonsteroidal Anti-Inflammatory Drug (NSAID) Imparts Hydrogelation Displaying Remarkable Biostability, Biocompatibility, and Anti-Inflammatory Properties
2013
Reciprocity of Steric and Stereoelectronic Effects in the Collagen Triple Helix
2006
Exploration of Fluorine Chemistry at the Multidisciplinary Interface of Chemistry and Biology
2013
How we drifted into peptide chemistry and where we have arrived at
2004
Unsaturated O- and N-Heterocycles from Carbohydrate Feedstocks
2002
Applications of Fluorine in Medicinal Chemistry
2015 Standout
CF2H, a Hydrogen Bond Donor
2017 Standout
Aldehyde Selective Wacker Oxidations of Phthalimide Protected Allylic Amines: A New Catalytic Route to β3-Amino Acids
2009 StandoutNobel
Incorporation of fluoroprolines to proctolin: Study on the effect of a fluorine atom toward peptidic conformation
2008
Structural Chemistry of Peptides Containing Backbone Expanded Amino Acid Residues: Conformational Features of β, γ, and Hybrid Peptides
2010
Operationally convenient asymmetric synthesis of (S)- and (R)-3-amino-4,4,4-trifluorobutanoic acid
2006
Stereoselective Fluorination Alters the Geometry of a Cyclic Peptide: Exploration of Backbone‐Fluorinated Analogues of Unguisin A
2014
Synopsis of Some Recent Tactical Application of Bioisosteres in Drug Design
2011 Standout
Can a C–H···O Interaction Be a Determinant of Conformation?
2012
Synthesis, Biological Activity, and Molecular Modeling Studies of 1H-1,2,3-Triazole Derivatives of Carbohydrates as α-Glucosidases Inhibitors
2010
Works of F. Gessier being referenced
Carbohydrate transition state mimics: synthesis of imidazolo-Pyrrolidinoses as potential nectrisine surrogates
2003
Discovery of dihydroisoquinolinone derivatives as novel inhibitors of the p53–MDM2 interaction with a distinct binding mode
2015
Probing the Proteolytic Stability of β‐Peptides Containing α‐Fluoro‐ and α‐Hydroxy‐β‐Amino Acids
2004
Stereoisomeric Imidazolo-Pentoses − Synthesis, Chiroptical Properties, and Evaluation as Glycosidase Inhibitors
2001
The Effect of Backbone-Heteroatom Substitution on the Folding of Peptides - A Single Fluorine Substituent Prevents a?-Heptapeptide from Folding into a314-Helix (NMR Analysis)
2005
Stereocontrolled synthesis of imidazolo[1,5]hexopiperidinoses and imidazol-4(5)-yl-C-glycosides
2003
Preparation ofβ2-Amino Acid Derivatives (β2hThr,β2hTrp,β2hMet,β2hPro,β2hLys, Pyrrolidine-3-carboxylic Acid) by Using DIOZ as Chiral Auxiliary
2005
Discovery of a Dihydroisoquinolinone Derivative (NVP-CGM097): A Highly Potent and Selective MDM2 Inhibitor Undergoing Phase 1 Clinical Trials in p53wt Tumors
2015
Stereoselective Preparation of 3‐Amino‐2‐fluoro Carboxylic Acid Derivatives, and Their Incorporation in Tetrahydropyrimidin‐4(1H)‐ones, and in Open‐Chain and Cyclic β‐Peptides
2011
Enantioselective Preparation of 2‐Aminomethyl Carboxylic Acid Derivatives: Solving the β2‐Amino Acid Problem with the Chiral Auxiliary 4‐Isopropyl‐5,5‐diphenyloxazolidin‐2‐one (DIOZ). Preliminary Communication
2003
Abstract 1798: Mechanistic study of NVP-CGM097: a potent, selective and species specific inhibitor of p53-Mdm2
2014
Synthesis and CD Spectra of Fluoro‐ and Hydroxy‐Substituted β‐Peptides
2003