Citation Impact
Citing Papers
Bifluoride Ion Mediated SuFEx Trifluoromethylation of Sulfonyl Fluorides and Iminosulfur Oxydifluorides
2019 StandoutNobel
Tuning the Transcriptional Response to Hypoxia by Inhibiting Hypoxia-inducible Factor (HIF) Prolyl and Asparaginyl Hydroxylases
2016 StandoutNobel
Similarity in drugs: reflections on analogue design
2006
Visible light photoredox catalysis: applications in organic synthesis
2010 Standout
Stereocontrolled routes to β,β′-disubstituted α-amino acids
2009
Recent progress in synthesis and bioactivity studies of indolizines
2011
Insulin Stimulates Hypoxia-inducible Factor 1 through a Phosphatidylinositol 3-Kinase/Target of Rapamycin-dependent Signaling Pathway
2002 StandoutNobel
An Efficient Approach to the Securinega Alkaloids Empowered by Cooperative N‐Heterocyclic Carbene/Lewis Acid Catalysis
2013
Catalysis for fluorination and trifluoromethylation
2011 StandoutNature
Non-heme iron oxygenases
2002
Oxygen sensing by HIF hydroxylases
2004 StandoutNobel
Synthesis, structure and biological activity of copper(II) complexes of 4-(2-pyridylmethyl)-1,7-dimethyl-1,4,7-triazonane-2,6-dione and 4-(2-pyridylethyl)-1,7-dimethyl-1,4,7-triazonane-2,6-dione
2008
Oxidative demethylation by Escherichia coli AlkB directly reverts DNA base damage
2002 StandoutNatureNobel
Nanoporous Carbohydrate Metal–Organic Frameworks
2011 StandoutNobel
Crystal structure of reduced thioredoxin reductase from Escherichia coli: Structural flexibility in the isoalloxazine ring of the flavin adenine dinucleotide cofactor
1999
Hypoxia-inducible Factor (HIF) Asparagine Hydroxylase Is Identical to Factor Inhibiting HIF (FIH) and Is Related to the Cupin Structural Family
2002 StandoutNobel
Asparaginyl Hydroxylation of the Notch Ankyrin Repeat Domain by Factor Inhibiting Hypoxia-inducible Factor
2007 StandoutNobel
Genetic Analysis of the Role of the Asparaginyl Hydroxylase Factor Inhibiting Hypoxia-inducible Factor (HIF) in Regulating HIF Transcriptional Target Genes
2004 StandoutNobel
ERK activation upon hypoxia: involvement in HIF‐1 activation
2000
Highly Efficient and Mild Copper‐Catalyzed N‐ and C‐Arylations with Aryl Bromides and Iodides
2004
A Catalytic Asymmetric 6 π Electrocyclization: Enantioselective Synthesis of 2‐Pyrazolines
2009 StandoutNobel
Asparagine and Aspartate Hydroxylation of the Cytoskeletal Ankyrin Family Is Catalyzed by Factor-inhibiting Hypoxia-inducible Factor
2010 StandoutNobel
DNA‐Based Catalytic Enantioselective Michael Reactions in Water
2007 StandoutNobel
The Hydrogen Bond in the Solid State
2002 Standout
‘Click’ assembly of selective inhibitors for MAO-A
2010
Antiplatelet therapy: in search of the 'magic bullet'
2003
Click Chemistry for Drug Development and Diverse Chemical–Biology Applications
2013 Standout
Monofluorination of Organic Compounds: 10 Years of Innovation
2015 Standout
Copper-Mediated Coupling Reactions and Their Applications in Natural Products and Designed Biomolecules Synthesis
2008 Standout
Synthesis of Celecoxib Analogues Possessing aN-Difluoromethyl-1,2-dihydropyrid-2-one 5-Lipoxygenase Pharmacophore: Biological Evaluation as Dual Inhibitors of Cyclooxygenases and 5-Lipoxygenase with Anti-Inflammatory Activity
2009
Fluorine in Pharmaceutical Industry: Fluorine-Containing Drugs Introduced to the Market in the Last Decade (2001–2011)
2013 Standout
A short and convenient chemoenzymatic synthesis of both enantiomers of 3-phenylGABA and 3-(4-chlorophenyl)GABA (Baclofen)
2005
Crystal Structures of the Bacillus licheniformis BS3 Class A β-Lactamase and of the Acyl−Enzyme Adduct Formed with Cefoxitin,
2002
Copper and Its Complexes in Medicine: A Biochemical Approach
2011
Phenyl−Perfluorophenyl Stacking Interactions: Topochemical [2+2] Photodimerization and Photopolymerization of Olefinic Compounds
1998 StandoutNobel
Hypoxia-inducible factor asparaginyl hydroxylase (FIH-1) catalyses hydroxylation at the β-carbon of asparagine-803
2002
Gold‐Catalyzed Sequential Amination/Annulation Reactions of 2‐Propynyl‐1,3‐dicarbonyl Compounds
2001
The catalytic mechanism of beta-lactamases: NMR titration of an active-site lysine residue of the TEM-1 enzyme.
1996
Stereochemical Control in Organic Synthesis Using Silicon-Containing Compounds
1997
Bis- and Trisindolylmethanes (BIMs and TIMs)
2009 Standout
Asymmetric Construction of Stereogenic Carbon Centers Featuring a Trifluoromethyl Group from Prochiral Trifluoromethylated Substrates
2010
Samarium(II)-Iodide-Mediated Cyclizations in Natural Product Synthesis
2004 Standout
Engineered Biosynthesis of β‐Alkyl Tryptophan Analogues
2018 StandoutNobel
Enantio- and Diastereoselective Michael Reaction of 1,3-Dicarbonyl Compounds to Nitroolefins Catalyzed by a Bifunctional Thiourea
2004
A New Method for the Synthesis of Chiral β-Branched α-Amino Acids
2007
Synthesis and Selective Inhibitory Activity of 1-Acetyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazole Derivatives against Monoamine Oxidase
2004
Synthesis of bromodifluoromethyl substituted pyrazoles and isoxazoles
2009
A New Enantioselective Approach to Total Synthesis of the Securinega Alkaloids: Application to (−)-Norsecurinine and Phyllanthine
2000
Staurosporine and ent-Staurosporine: The First Total Syntheses, Prospects for a Regioselective Approach, and Activity Profiles1
1996
Pyridine Analogues of Nimesulide: Design, Synthesis, and in Vitro and in Vivo Pharmacological Evaluation as Promising Cyclooxygenase 1 and 2 Inhibitors
2009
Next Generation of Fluorine-Containing Pharmaceuticals, Compounds Currently in Phase II–III Clinical Trials of Major Pharmaceutical Companies: New Structural Trends and Therapeutic Areas
2016 Standout
Bacterial Resistance to β-Lactam Antibiotics: Compelling Opportunism, Compelling Opportunity
2005 Standout
Chromone: A Valid Scaffold in Medicinal Chemistry
2014 Standout
Adaptive and Maladaptive Cardiorespiratory Responses to Continuous and Intermittent Hypoxia Mediated by Hypoxia-Inducible Factors 1 and 2
2012 StandoutNobel
Nucleophilic trifluoromethylation
2005
N-Heterocyclic Carbenes in Late Transition Metal Catalysis
2009 Standout
Selected Patented Cross-Coupling Reaction Technologies
2006 Standout
Highly Efficient CuI-Catalyzed Coupling of Aryl Bromides with Oxazolidinones Using Buchwald's Protocol: A Short Route to Linezolid and Toloxatone
2003
Fluorine in Pharmaceuticals: Looking Beyond Intuition
2007 StandoutScience
Stereoselective Cyclopropanation Reactions
2003 Standout
Electrophilic Trifluoromethylation by Use of Hypervalent Iodine Reagents
2014 Standout
Monoamine Oxidase Isoform-Dependent Tautomeric Influence in the Recognition of 3,5-Diaryl Pyrazole Inhibitors
2007
Advances in Catalytic Enantioselective Fluorination, Mono-, Di-, and Trifluoromethylation, and Trifluoromethylthiolation Reactions
2014
A Field Guide to Foldamers
2001 Standout
Recent advances in enantioselective trifluoromethylation reactions
2008
How to Reach Stereogenic Trifluoromethylated Carbon? En Route to the “Grail” of the Asymmetric Trifluoromethylation Reaction
2006
Organocatalytic Reactions Enabled by N-Heterocyclic Carbenes
2015 Standout
Alternative Synthetic Methods through New Developments in Catalysis by Gold
2008 Standout
Catalytic Asymmetric Conjugate Addition and Allylic Alkylation with Grignard Reagents
2008 StandoutNobel
Small-Molecule H-Bond Donors in Asymmetric Catalysis
2007 Standout
Ultrafast Dynamics of Flavins in Five Redox States
2008 StandoutNobel
Total Syntheses of the Securinega Alkaloids (+)-14,15-Dihydronorsecurinine, (−)-Norsecurinine, and Phyllanthine
2000
Acyclic C-nucleosides: synthesis of chiral 1,1-diheteroaryl-alditols and X-ray crystal structure of 2,3,5-tri-O-benzyl-1,1-di-(2′-pyrryl)-1-deoxy-d-arabinitol
1997
Organic Fluorine Hardly Ever Accepts Hydrogen Bonds
1997
Applications of Palladium-Catalyzed C–N Cross-Coupling Reactions
2016 Standout
Aromatic Trifluoromethylation with Metal Complexes
2011 Standout
Advances in Copper Complexes as Anticancer Agents
2013 Standout
Thermal analysis and calorimetric methods in the characterisation of polymorphs and solvates
1995
Remarkable asymmetric induction from remote stereocenters in conjugate addition chemistry for the synthesis of alkyl‐branched α, ω‐diaminoazelates
2001
Palladium-Catalyzed Synthesis of N-Aryloxazolidinones from Aryl Chlorides
2003
Conformationally restricted amino acids: Diastereoselective substitution at the β-position of L-tryptophan
1992
From 2000 to Mid-2010: A Fruitful Decade for the Synthesis of Pyrazoles
2011 Standout
HIF-1 and human disease: one highly involved factor
2000 StandoutNobel
Gold-Catalyzed Organic Reactions
2007 Standout
Application of Rhodium Complexes of Chiral Diphenylphosphino‐Functionalized N‐Heterocyclic Carbenes as Catalysts in Enantioselective Conjugate Additions of Arylboronic Acids
2005
Ultrafast Dynamics and Anionic Active States of the Flavin Cofactor in Cryptochrome and Photolyase
2008 StandoutNobel
Isolation and Synthesis of Biologically Active Carbazole Alkaloids
2002 Standout
Aryl−Aryl Bond Formation One Century after the Discovery of the Ullmann Reaction
2002 Standout
A New Approach Towards the Synthesis of 3-Amino-6-(hetero)arylpyridazines Based on Palladium Catalyzed Cross-coupling Reactions
2000
Stronger Brønsted Acids
2007 Standout
Synopsis of Some Recent Tactical Application of Bioisosteres in Drug Design
2011 Standout
Catalytic Asymmetric Conjugate Addition of Indolizines to α,β‐Unsaturated Ketones
2017 StandoutNobel
Works of F. Durant being referenced
Synthesis and biochemical evaluation of baclofen analogs locked in the baclofen solid-state conformation
1991
Structure and molecular modeling of GABAA receptor antagonists
1992
Terbogrel, a dual-acting agent for thromboxane receptor antagonism and thromboxane synthase inhibition
2000
A Model for the Complex Between the Hypoxia-Inducible Factor-1 (HIF-1) and its Consensus DNA Sequence
2000
Metal-organic compounds: a new approach for drug discovery
2002
A reversible monoamine oxidase a inhibitor, befloxatone: structural approach of its mechanism of action
1999
Structure-affinity relationships of baclofen and 3-heteroaromatic analogues
1995
1-[[4-(Aminoalkoxy)phenyl]sulfonyl]indolizines: a novel class of calcium entry blockers. Relationships between chemical structure, stereoelectronic properties and anticalcic activity
1994
De novo drug design of a new copper chelate molecule acting as HIV-1 protease inhibitor
1998
New COX-2/5-LOX Inhibitors: Apoptosis-Inducing Agents Potentially Useful in Prostate Cancer Chemotherapy
2004
Molecular modeling of the hypoxia-inducible factor-1 (HIF-1)
1999
A reversible monoamine oxidase inhibitor, toloxatone: Structural and electronic properties
1992
A reversible monoamine oxidase inhibitor, toloxatone: spectrophotometric and molecular orbital studies of the interaction with flavin adenine dinucleotide (FAD)
1994
Spectral and Crystallographic Study of Pyridinic Analogues of Nimesulide: Determination of the Active Form of Methanesulfonamides as COX-2 Selective Inhibitors
2002
Étude du Polymorphisme et de L'Intersolubilité de Triglycerides Palmito‐Oleiques par Diffraction RX de Poudres et Analyse Calorimétrique Différentielle
1985
Molecular structure of two gastrokinetic compounds, cisapride and R53757: comparison with dopaminergic D2 antagonists
1989
Reversible inhibition of type B monoamine oxidase. Theoretical study of model diazo heterocylic compound
1997
Stereoselective synthesis of 3-alkylated glutamic acids: application to the synthesis of secokainic acid
1991
Structural characterization of oxidized lumiflavin hydrochloride hydrate: Comparison with the hydrogen bonding at the cofactor of flavoproteins
1994
Rhenium(V) and technetium(V) complexes with N-[2(1H-pyrolylmethyl)]-N′-(4-pentene-3-one-2) ethane-1,2-diaminate (C12H16N3O, MRP 20). X-ray crystal structures of H3MRP 20 and TcO(MRP 20)
1991
Direct n.m.r. evidence for substrate-induced conformational changes in a β-lactamase
1994