Citation Impact
Citing Papers
SuFEx-enabled, agnostic discovery of covalent inhibitors of human neutrophil elastase
2019 StandoutNobel
Diversity oriented clicking delivers β-substituted alkenyl sulfonyl fluorides as covalent human neutrophil elastase inhibitors
2022 StandoutNobel
Unified Synthesis of Polycyclic Alkaloids by Complementary Carbonyl Activation**
2021 StandoutNobel
A Porous Crystalline Nitrone‐Linked Covalent Organic Framework**
2023 StandoutNobel
Triphenylphosphine-catalysed amide bond formation between carboxylic acids and amines
2014
Expansive discovery of chemically diverse structured macrocyclic oligoamides
2024 StandoutScienceNobel
Bioconjugated lanthanide luminescent helicates as multilabels for lab-on-a-chip detection of cancer biomarkers
2009
Immobilization of Ferrocene-Modified SNAP-Fusion Proteins
2013
Iron‐Catalyzed CH and CC Bond Cleavage: A Direct Approach to Amides from Simple Hydrocarbons
2011
Metal–organic framework composites
2014 Standout
Iron-catalysed oxidative amidation of alcohols with amines
2013
Rethinking amide bond synthesis
2011 StandoutNature
Microreactors for peptide synthesis: looking through the eyes of twenty first century !!!
2014
Macrocyclic peptide-based inhibition and imaging of hepatocyte growth factor
2019
In-solution enrichment identifies peptide inhibitors of protein–protein interactions
2019
Atmospheric pressure aminocarbonylation of aryl iodides using palladium nanoparticles supported on MOF-5
2011
Iron‐Catalyzed Oxidative Amidation of Tertiary Amines with Aldehydes
2012
The road to fully programmable protein catalysis
2022 StandoutNatureNobel
Umpolung reactivity in amide and peptide synthesis
2010 Nature
Bayer’s in silico ADMET platform: a journey of machine learning over the past two decades
2020
Scalable, Continuous Evolution of Genes at Mutation Rates above Genomic Error Thresholds
2018
Molecular monolayers on silicon as substrates for biosensors
2010
Anchor extension: a structure-guided approach to design cyclic peptides targeting enzyme active sites
2021 StandoutNobel
Efficient Amide Bond Formation through a Rapid and Strong Activation of Carboxylic Acids in a Microflow Reactor
2013
Enantioselective Total Synthesis of (−)‐Lansai B and (+)‐Nocardioazines A and B
2014
Thirteen decades of peptide synthesis: key developments in solid phase peptide synthesis and amide bond formation utilized in peptide ligation
2017
Delivery of Oligonucleotides to the Liver with GalNAc: From Research to Registered Therapeutic Drug
2020
Chiral amides via copper-catalysed enantioselective conjugate addition
2013 StandoutNobel
A biomolecule-compatible visible-light-induced azide reduction from a DNA-encoded reaction-discovery system
2011
Rhodium‐Catalyzed Synthesis of Amides from Aldehydes and Azides by Chelation‐Assisted CH Bond Activation
2013
Metal-catalysed approaches to amide bond formation
2011 Standout
Combining UV Lithography and an Imprinting Technique for Patterning Metal‐Organic Frameworks
2013 StandoutNobel
Trends in peptide drug discovery
2021
Peptide Fragment Coupling Using a Continuous‐Flow Photochemical Rearrangement of Nitrones
2013
Recent advances in Sonogashira reactions
2011 Standout
Catalytic Acylation of Amines with Aldehydes or Aldoximes
2010
The Unexpected Importance of the Primary Structure of the Hydrophobic Part of One-Component Ionizable Amphiphilic Janus Dendrimers in Targeted mRNA Delivery Activity
2022 StandoutNobel
Monofluorination of Organic Compounds: 10 Years of Innovation
2015 Standout
Ru(II)-catalyzed ortho-amidation and decarboxylation of aromatic acids: a versatile route to meta-substituted N-aryl benzamides
2015
Iron Catalysis in Organic Synthesis
2015 Standout
Amide Bond Formation through Iron-Catalyzed Oxidative Amidation of Tertiary Amines with Anhydrides
2013
Artificial Photosynthesis: Molecular Systems for Catalytic Water Oxidation
2014
Peptide Coupling Reagents, More than a Letter Soup
2011
Diacetoxyiodobenzene Mediated One-Pot Synthesis of Diverse Carboxamides from Aldehydes
2012
Macrocycles in Drug Discovery─Learning from the Past for the Future
2023
Transamidation of Carboxamides Catalyzed by Fe(III) and Water
2014
Iron‐Catalyzed Efficient Synthesis of Amides from Aldehydes and Amine Hydrochloride Salts
2012
Organic Photoredox Catalysis
2016 Standout
Magnetic CuFe2O4 nanoparticles: a retrievable catalyst for oxidative amidation of aldehydes with amine hydrochloride salts
2014
Cost efficient synthesis of amides from oximes with indium or zinc catalysts
2010
Lanthanide Luminescence for Biomedical Analyses and Imaging
2010 Standout
State of the Art and Prospects in Metal–Organic Framework (MOF)-Based and MOF-Derived Nanocatalysis
2019 Standout
The Hitchhiker’s Guide to Flow Chemistry
2017 Standout
Adapting free energy perturbation simulations for large macrocyclic ligands: how to dissect contributions from direct binding and free ligand flexibility
2020
Recyclable Hypervalent Iodine(III) Reagent Iodosodilactone as an Efficient Coupling Reagent for Direct Esterification, Amidation, and Peptide Coupling
2012
Macrocyclic Peptides as Drug Candidates: Recent Progress and Remaining Challenges
2019
Cucurbituril-Based Molecular Recognition
2015 Standout
Mild and Selective Heterogeneous Catalytic Hydration of Nitriles to Amides by Flowing through Manganese Dioxide
2014
Multistep Solid-State Organic Synthesis of Carbamate-Linked Covalent Organic Frameworks
2019 StandoutNobel
Phosphine Organocatalysis
2018 Standout
Degradable Controlled-Release Polymers and Polymeric Nanoparticles: Mechanisms of Controlling Drug Release
2016 Standout
Deep Eutectic Solvents (DESs) and Their Applications
2014 Standout
Chromone: A Valid Scaffold in Medicinal Chemistry
2014 Standout
Applications of Acceptorless Dehydrogenation and Related Transformations in Chemical Synthesis
2013 StandoutScience
Sulfur–Fluoride Exchange (SuFEx)‐Mediated Synthesis of Sterically Hindered and Electron‐Deficient Secondary and Tertiary Amides via Acyl Fluoride Intermediates
2017
Metal-Catalyzed Decarboxylative C–H Functionalization
2017 Standout
Trypsin‐Immobilized Metal–Organic Framework as a Biocatalyst In Proteomics Analysis
2012
Computational Study on the Catalytic Role of Pincer Ruthenium(II)-PNN Complex in Directly Synthesizing Amide from Alcohol and Amine: The Origin of Selectivity of Amide over Ester and Imine
2011
Applications of metal–organic frameworks in heterogeneous supramolecular catalysis
2014 Standout
Electrochemical synthesis of amides: direct transformation of methyl ketones with formamides
2013
Recent Advances in the Catalytic Asymmetric Synthesis of β2‐ and β2,2‐Amino Acids
2019
Polystyrene‐supported palladium(II) ethylenediamine complex: A highly active and recyclable catalyst for the synthesis of 2‐benzylimidazo[2,1‐b]pyridines through heteroannulation of acetylenic compounds
2009
RNA Display Methods for the Discovery of Bioactive Macrocycles
2018
Synthetic Organic Electrochemical Methods Since 2000: On the Verge of a Renaissance
2017 Standout
Iron(II)-Catalyzed Amidation of Aldehydes with Iminoiodinanes at Room Temperature and under Microwave-Assisted Conditions
2011
Direct Amide Synthesis from Either Alcohols or Aldehydes with Amines: Activity of Ru(II) Hydride and Ru(0) Complexes
2010
Rhodium(III)-Catalyzed Intermolecular Direct Amidation of Aldehyde C–H Bonds withN-Chloroamines at Room Temperature
2013
Water solubilization of xanthene dyes by post-synthetic sulfonation in organic media
2010
Lipids and Lipid Derivatives for RNA Delivery
2021
Catalytic Asymmetric Synthesis of Unprotected β2-Amino Acids
2021 StandoutNobel
Modular Functionalization of Electrodes by Cross‐Coupling Reactions at Their Surfaces
2011 StandoutNobel
Extending the application of biocatalysis to meet the challenges of drug development
2018
Reactive Oxygen Species (ROS)-Based Nanomedicine
2019 Standout
A Phage-Assisted Continuous Selection Approach for Deep Mutational Scanning of Protein–Protein Interactions
2019
Pseudo-Five-Component Reaction between 3-Formylchromones, Meldrum’s Acid, Isocyanides and Primary Arylamines: Diversity-Oriented Synthesis of Novel Chromone-Containing Peptidomimetics
2011
Advances in Synthetic Applications of Hypervalent Iodine Compounds
2016 Standout
The thermal and boron-catalysed direct amide formation reactions: mechanistically understudied yet important processes
2010
Diversity Oriented Clicking (DOC): Divergent Synthesis of SuFExable Pharmacophores from 2‐Substituted‐Alkynyl‐1‐Sulfonyl Fluoride (SASF) Hubs
2020 StandoutNobel
A Panel of TrpB Biocatalysts Derived from Tryptophan Synthase through the Transfer of Mutations that Mimic Allosteric Activation
2016 StandoutNobel
Recent advances towards sulfur (VI) fluoride exchange (SuFEx) click chemistry
2018
Redox-responsive polymers for drug delivery: from molecular design to applications
2013
Enantioselective Total Synthesis of (−)‐Lansai B and (+)‐Nocardioazines A and B
2014
ADMETlab 2.0: an integrated online platform for accurate and comprehensive predictions of ADMET properties
2021 Standout
Metal–organic frameworks meet metal nanoparticles: synergistic effect for enhanced catalysis
2017 Standout
Thio FCMA Intermediates as Strong Acyl Donors: A General Solution to the Formation of Complex Amide Bonds
2009
De Novo Carborane-Containing Macrocyclic Peptides Targeting Human Epidermal Growth Factor Receptor
2019 StandoutNobel
Synthesis of Primary Amides via Copper-Catalyzed Aerobic Decarboxylative Ammoxidation of Phenylacetic Acids and α-Hydroxyphenylacetic Acids with Ammonia in Water
2014
Cocatalysts for Selective Photoreduction of CO2into Solar Fuels
2019 Standout
Choline chloride based eutectic solvent: an efficient and reusable solvent system for the synthesis of primary amides from aldehydes and from nitriles
2013
Scalable mRNA and siRNA Lipid Nanoparticle Production Using a Parallelized Microfluidic Device
2021 StandoutNobel
Visible Light Photoredox Catalysis with Transition Metal Complexes: Applications in Organic Synthesis
2013 Standout
Recent Progress in Cobalt‐Based Heterogeneous Catalysts for Electrochemical Water Splitting
2015 Standout
Visible‐Light Photocatalysis: Does It Make a Difference in Organic Synthesis?
2018 Standout
Selective radical amination of aldehydic C(sp2)–H bonds with fluoroaryl azides via Co(ii )-based metalloradical catalysis: synthesis of N-fluoroaryl amides from aldehydes under neutral and nonoxidative conditions
2014
Transition Metal-Catalyzed C–H Amination: Scope, Mechanism, and Applications
2017 Standout
N-Heterocyclic Carbene-Mediated Microfluidic Oxidative Electrosynthesis of Amides from Aldehydes
2016
Solar Synthesis: Prospects in Visible Light Photocatalysis
2014 StandoutScience
Metal-free oxidative amide formation with N-hydroxysuccinimide and hypervalent iodine reagents
2012
Conformational Strain of Macrocyclic Peptides in Ligand–Receptor Complexes Based on Advanced Refinement of Bound-State Conformers
2021
Iron‐Catalyzed Amidation of Aldehydes with N‐Chloroamines
2012
Differential Effects of β3‐ versus β2‐Amino Acid Residues on the Helicity and Recognition Properties of Bim BH3‐Derived α/β‐Peptides
2018
Cyclic Tetrapeptides from Nature and Design: A Review of Synthetic Methodologies, Structure, and Function
2019
Design Strategies for Water-Soluble Small Molecular Chromogenic and Fluorogenic Probes
2013 Standout
Approach to Comparing the Functional Group Tolerance of Reactions
2017
Accurate proteome-wide missense variant effect prediction with AlphaMissense
2023 StandoutScienceNobel
Phenazinium Salt-Catalyzed Aerobic Oxidative Amidation of Aromatic Aldehydes
2014
Well-Defined N-Heterocyclic Carbene Based Ruthenium Catalysts for Direct Amide Synthesis from Alcohols and Amines
2010
Works of Eric Valeur being referenced
PS-IIDQ: an efficient polymer-supported amide coupling reagent
2005
Directing evolution: the next revolution in drug discovery?
2017
Amide bond formation: beyond the myth of coupling reagents
2008 Standout
Therapeutic Potential of Foldamers: From Chemical Biology Tools To Drug Candidates?
2016
New Modalities, Technologies, and Partnerships in Probe and Lead Generation: Enabling a Mode-of-Action Centric Paradigm
2018
Macrocyclic Modalities Combining Peptide Epitopes and Natural Product Fragments
2020
Inhibition of low-density lipoprotein receptor degradation with a cyclic peptide that disrupts the homodimerization of IDOL E3 ubiquitin ligase
2018
New Modalities for Challenging Targets in Drug Discovery
2017
Emerging modes-of-action in drug discovery
2019
PS-IIDQ: a supported coupling reagent for efficient and general amide bond formation
2007
Targeted delivery of antisense oligonucleotides to pancreatic β-cells
2018