Citation Impact
Citing Papers
Preparation of modified peptides: direct conversion of α-amino acids into β-amino aldehydes
2012
Proteasome inhibitors: from research tools to drug candidates
2001
Two Membrane-Associated Tyrosine Phosphatase Homologs Potentiate C. elegans AKT-1/PKB Signaling
2006 StandoutNobel
Novel cell-penetrating α-keto-amide calpain inhibitors as potential treatment for muscular dystrophy
2005
The ubiquitin‐proteasome pathway and proteasome inhibitors
2001
A series of peptide-based, fluorogenic probes for protein tyrosine phosphatase activity
2007
Proteasome Inhibitors: Complex Tools for a Complex Enzyme
2002
Ocular Drug Delivery
2010 Standout
Optical control of antibacterial activity
2013 StandoutNobel
Structural Basis for Recognizing Phosphoarginine and Evolving Residue-Specific Protein Phosphatases in Gram-Positive Bacteria
2013 StandoutNobel
Aptamers as therapeutics
2010 Standout
Mechanistic Studies on Protein Tyrosine Phosphatases
2003
Fibroblast growth factor signalling: from development to cancer
2010 Standout
Protein degradation and protection against misfolded or damaged proteins
2003 StandoutNature
Pharmaceutical and medicinal significance of sulfur (SVI)-Containing motifs for drug discovery: A critical review
2018 Standout
The Mechanism of Dephosphorylation of Extracellular Signal-regulated Kinase 2 by Mitogen-activated Protein Kinase Phosphatase 3
2001
Copper-catalyzed aerobic oxidative synthesis of α-ketoamides from methyl ketones, amines and NIS at room temperature
2012
The use of spirocyclic scaffolds in drug discovery
2014 Standout
Withaferin A is a potent inhibitor of angiogenesis
2004 Standout
5-Substituted-1H-tetrazoles as carboxylic acid isosteres: medicinal chemistry and synthetic methods
2002 Standout
Exploration of orally available calpain inhibitors. Part 3: Dipeptidyl α-ketoamide derivatives containing pyridine moiety
2006
RNA Molecules That Bind to and Inhibit the Active Site of a Tyrosine Phosphatase
1998
Development of Calpain-specific Inactivators by Screening of Positional Scanning Epoxide Libraries
2007
Protein Tyrosine Phosphatases in the Human Genome
2004 Standout
Proteasome Inhibitors with Photocontrolled Activity
2014 StandoutNobel
De novo design of tyrosine and serine kinase-driven protein switches
2021 StandoutNobel
Synthesis and evaluation of a new series of 1′-cyclobutyl-6-(4-piperidyloxy)spiro[benzopyran-2,4′-piperidine] derivatives as high affinity and selective histamine-3 receptor (H3R) antagonists
2012
Calpain inhibitors based on the quiescent affinity label concept: high rates of calpain inactivation with leaving groups derived from N-hydroxy peptide coupling reagents
2000
Chapter 11 Proteinase families and their inhibitors
2001
Organic Azides: An Exploding Diversity of a Unique Class of Compounds
2005 Standout
Solid-Phase Combinatorial Library of Norstatine-Type Isosters by the Nitroaldol Reaction
2003 StandoutNobel
Serotonin 5-HT6Receptor Antagonists for the Treatment of Cognitive Deficiency in Alzheimer’s Disease
2014
Short, Highly Efficient Syntheses of Protected 3-Azido- and 4-Azidoproline and Their Precursors
2001
A Critical Review on Chagas Disease Chemotherapy
2002 Standout
Fluorine and Fluorinated Motifs in the Design and Application of Bioisosteres for Drug Design
2018 Standout
Cyanogen Bromide Cleavage Generates Fragments Suitable for Expressed Protein and Glycoprotein Ligation
2004 StandoutNobel
Lanthanide Luminescence for Biomedical Analyses and Imaging
2010 Standout
Peptido-organic Diels–Alder reactions on hydrophilic resin: scope for combinatorial chemistry
2001 StandoutNobel
Palladium-Catalyzed Anti-Markovnikov Oxidation of Allylic Amides to Protected β-Amino Aldehydes
2014 StandoutNobel
Calpain inhibitors as potential treatment for stroke and other neurodegenerative diseases: recent trends and developments
1998
Neue Ziele für die Photopharmakologie
2016 StandoutNobel
Combinatorial Library of Peptidotriazoles: Identification of [1,2,3]-Triazole Inhibitors against a RecombinantLeishmaniamexicanaCysteine Protease
2004 StandoutNobel
Occurrence, Biogenesis, and Synthesis of Biologically Active Carbazole Alkaloids
2012 Standout
Versatile Protein Biotinylation Strategies for Potential High-Throughput Proteomics
2004
Protein Tyrosine Phosphatases: Structure and Function, Substrate Specificity, and Inhibitor Development
2002
THE STRUCTURE AND MECHANISM OF PROTEIN PHOSPHATASES: Insights into Catalysis and Regulation
1998
Precise Modulation of CO2 Sorption in Ti8Ce2–Oxo Clusters: Elucidating Lewis Acidity of the Ce Metal Sites and Structural Flexibility
2024 StandoutNobel
The Calpain System
2003 Standout
Solid Phase Combinatorial Library of 1,3‐Azole Containing Peptides for the Discovery of Matrix Metallo Proteinase Inhibitors
2003 StandoutNobel
Combinatorial Library of Serine and Cysteine Protease Inhibitors That Interact with Both the S and S‘ Binding Sites
1999
Design, Synthesis and Evaluation of d-Homophenylalanyl Epoxysuccinate Inhibitors of the Trypanosomal Cysteine Protease Cruzain
2000
Reversible Photocontrol of Biological Systems by the Incorporation of Molecular Photoswitches
2013 StandoutNobel
The Catalytic Asymmetric Aminohydroxylation of Unsaturated Phosphonates
1999 StandoutNobel
Aerobic Copper-Catalyzed Organic Reactions
2013 Standout
The synthesis and crystal structure of alpha-keto tetrazole-based dipeptide mimics
2001
Protease Inhibitors: Current Status and Future Prospects
2000
Solid-Phase Library Synthesis, Screening, and Selection of Tight-Binding Reduced Peptide Bond Inhibitors of a RecombinantLeishmaniamexicanaCysteine Protease B
2002 StandoutNobel
Impact of Natural Products on Developing New Anti-Cancer Agents
2009 Standout
Efficient Synthesis of Maleimides and Carbazoles via Zn(OTf)2-Catalyzed Tandem Annulations of Isonitriles and Allenic Esters
2007
Synthesis and Biological Activity of a Series of Potent Fluoromethyl Ketone Inhibitors of Recombinant Human Calpain I
1997
Investigation into the P3 Binding Domain of m-Calpain Using Photoswitchable Diazo- and Triazene-dipeptide Aldehydes: New Anticataract Agents
2007
Emerging Targets in Photopharmacology
2016 StandoutNobel
Chemistry and Biology Of Multicomponent Reactions
2012 Standout
Photopharmacology: Beyond Proof of Principle
2014 StandoutNobel
Irreversible Inhibitors of Serine, Cysteine, and Threonine Proteases
2002 Standout
Combinatorial Library of Peptide Isosters Based on Diels−Alder Reactions: Identification of Novel Inhibitors against a Recombinant Cysteine Protease fromLeishmania mexicana
2001 StandoutNobel
Copper-catalyzed direct oxidative synthesis of α-ketoamides from aryl methyl ketones, amines, and molecular oxygen
2011
5‐Substituted 1H‐Tetrazoles as Carboxylic Acid Isosteres: Medicinal Chemistry and Synthetic Methods
2003 Standout
Novel Peptidyl Phosphorus Derivatives as Inhibitors of Human Calpain I
1998
Works of Derek Dunn being referenced
Lactam and oxazolidinone derived potent 5-hydroxytryptamine 6 receptor antagonists
2014
P2-proline-derived inhibitors of calpain I
1998
Novel morpholine ketone analogs as potent histamine H3 receptor inverse agonists with wake activity
2012
P2-achiral, P'-extended α-ketoamide inhibitors of calpain I
1999
Identification of pyridazin-3-one derivatives as potent, selective histamine H3 receptor inverse agonists with robust wake activity
2011
Novel poly(ADP-ribose) polymerase-1 inhibitors
2006
4,5-Dihydropyridazin-3-one derivatives as histamine H3 receptor inverse agonists
2011
The Active Site Specificity of the Yersinia Protein-tyrosine Phosphatase
1996
P′-extended α-ketoamide inhibitors of proteasome
1999
Subsite requirements for peptide aldehyde inhibitors of human calpain I
1997
1998