Citation Impact
Citing Papers
Identification of a Primary Target of Thalidomide Teratogenicity
2010 StandoutScience
Passerini reaction – Amine Deprotection – Acyl Migration (PADAM): a convenient strategy for the solid-phase preparation of peptidomimetic compounds
2003
The Efficient One‐Pot Reaction of up to Eight Components by the Union of Multicomponent Reactions
2009
Catalytic Three‐Component Ugi Reaction
2008 StandoutNobel
Copper‐Catalyzed Synthesis of N‐Sulfonyl‐1,2,3‐triazoles: Controlling Selectivity
2007 StandoutNobel
Azobenzene Photoswitches for Staudinger–Bertozzi Ligation
2013 StandoutNobel
Organoiodine (III) mediated synthesis of 3-aryl/hetryl-5,7-dimethyl-1,2,4-triazolo[4,3-a]pyrimidines as antibacterial agents
2004
A New Structural Motif for Bifunctional Brønsted Acid/Base Organocatalysis
2010 StandoutNobel
The impact of informatics and computational chemistry on synthesis and screening
2001
Halogen Atoms in the Modern Medicinal Chemistry: Hints for the Drug Design
2010
On the industrial applications of MCRs: molecular diversity in drug discovery and generic drug synthesis
2010
In situ click chemistry: probing the binding landscapes of biological molecules
2010
Higher-order multicomponent reactions: beyond four reactants
2013
Phosphoramidites: Privileged Ligands in Asymmetric Catalysis
2010 StandoutNobel
Seven-component reactions by sequential chemoselective Ugi–Mumm/Ugi–Smiles reactions
2010
Protein Structure Similarity as Guiding Principle for Combinatorial Library Design
2003
Development and application of high‐performance affinity beads: Toward chemical biology and drug discovery
2009
Asymmetric Multicomponent Reactions (AMCRs): The New Frontier
2005 Standout
Multicomponent Reaction Design in the Quest for Molecular Complexity and Diversity
2011 Standout
Organic Azides: An Exploding Diversity of a Unique Class of Compounds
2005 Standout
Click Chemistry for Drug Development and Diverse Chemical–Biology Applications
2013 Standout
Regiospecific solid-phase synthesis of substituted 1,2,3-triazoles
2004
Potassium fluoride doped fluorapatite and hydroxyapatite as new catalysts in organic synthesis
2003
Copper-Mediated Coupling Reactions and Their Applications in Natural Products and Designed Biomolecules Synthesis
2008 Standout
3d Transition Metals for C–H Activation
2018 Standout
Bond Formations between Two Nucleophiles: Transition Metal Catalyzed Oxidative Cross-Coupling Reactions
2011 Standout
Cu and Cu-Based Nanoparticles: Synthesis and Applications in Catalysis
2016 Standout
Oxidation of Alcohols with Molecular Oxygen on Solid Catalysts
2004 Standout
Chemistry of Polyvalent Iodine
2008 Standout
Steric and Dynamic Parameters Influencing In Situ Cycloadditions to Form Triazole Inhibitors with Crystalline Acetylcholinesterase
2016 StandoutNobel
Cross‐Coupling Reactions on Azoles with Two and More Heteroatoms
2006
Natural Product Synthesis Using Multicomponent Reaction Strategies
2009 Standout
Investigation of Petasis and Ugi reactions in series in an automated microreactor system
2014
Chemical biology of dynamic combinatorial libraries
2002
Neue Entwicklungen in der asymmetrischen Mehrkomponenten‐Reaktion
2005
Concise synthesis of quinazoline alkaloids, luotonins A and B, and rutaecarpine
2004
Enantio- and diastereoselective synthesis of 2,5-disubstituted pyrrolidines through a multicomponent Ugi reaction and their transformation into bicyclic scaffolds
2004
The Hitchhiker’s Guide to Flow Chemistry
2017 Standout
Application of tandem Ugi reaction/ring-closing metathesis in multicomponent synthesis of unsaturated nine-membered lactams
2003
Comprehensive Survey of Combinatorial Library Synthesis: 2002
2003
The Efficient One‐Pot Reaction of up to Eight Components by the Union of Multicomponent Reactions
2009
Practical Synthesis and Elaboration of Methyl 7-Chloroindole-4-carboxylate
2003
Practical Methodologies for the Synthesis of Indoles
2006 Standout
Parallel synthesis of tandem Ugi/Diels–Alder reaction products on a soluble polymer support directed toward split-pool realization of a small molecule library
2004
Synthesis and Functionalization of Indoles Through Palladium-catalyzed Reactions
2005 Standout
Solid-Phase Synthesis of Indolecarboxylates Using Palladium-Catalyzed Reactions
2003
The Sonogashira Reaction: A Booming Methodology in Synthetic Organic Chemistry
2007 Standout
Next Generation of Fluorine-Containing Pharmaceuticals, Compounds Currently in Phase II–III Clinical Trials of Major Pharmaceutical Companies: New Structural Trends and Therapeutic Areas
2016 Standout
Dynamic Combinatorial Chemistry
2006 Standout
Recent Developments in Isocyanide Based Multicomponent Reactions in Applied Chemistry
2005 Standout
Generation of Candidate Ligands for Nicotinic Acetylcholine Receptors via in situ Click Chemistry with a Soluble Acetylcholine Binding Protein Template
2012 StandoutNobel
Use of Lawesson's Reagent in Organic Syntheses
2007 Standout
Observation of the controlled assembly of preclick components in the in situ click chemistry generation of a chitinase inhibitor
2013 StandoutNobel
Folding of a donor–acceptor polyrotaxane by using noncovalent bonding interactions
2008 StandoutNobel
Selected Patented Cross-Coupling Reaction Technologies
2006 Standout
Catalytic Dehydrogenative Cross-Coupling: Forming Carbon−Carbon Bonds by Oxidizing Two Carbon−Hydrogen Bonds
2011 Standout
Aryl−Aryl Bond Formation by Transition-Metal-Catalyzed Direct Arylation
2007 Standout
1,2,3-Triazole and its derivatives. Development of methods for the formation of the triazole ring
2005
Ugi-Post Functionalization, from a Single Set of Ugi-Adducts to Two Distinct Heterocycles by Microwave-Assisted Palladium-Catalyzed Cyclizations: Tuning the Reaction Pathways by Ligand Switch
2009
Organische Azide – explodierende Vielfalt bei einer einzigartigen Substanzklasse
2005
The Alternative Route to Enantiopure Multicomponent Reaction Products: Biocatalytic or Organocatalytic Enantioselective Production of Inputs for Multicomponent Reactions
2014
Multicomponent reactions: advanced tools for sustainable organic synthesis
2014 Standout
Intramolecular C(sp3)–H amination
2013
Concise Synthesis of 11H-Indolizino- [1,2-b]quinolin-9-one by an Aryl-Aryl Coupling Reaction Using Pd Reagent
2004
Synthesis of Spirocyclopropanated Analogues of Iprodione
2005
Boronic Acids and Esters in the Petasis-Borono Mannich Multicomponent Reaction
2010
Metalated Heterocycles and Their Applications in Synthetic Organic Chemistry
2004
Stereoselective Anhydride Openings
2007
In situclick chemistry: a powerful means for lead discovery
2006 StandoutNobel
The Combinatorial Synthesis of Bicyclic Privileged Structures or Privileged Substructures
2003 Standout
Design of Multi‐Component Reactions: From Libraries of Compounds to Libraries of Reactions
2006
Palladium‐Catalyzed, tert‐Butyllithium‐Mediated Dimerization of Aryl Halides and Its Application in the Atropselective Total Synthesis of Mastigophorene A
2016 StandoutNobel
Large-Scale Applications of Transition Metal-Catalyzed Couplings for the Synthesis of Pharmaceuticals
2011 Standout
Liquid‐phase synthesis of mixture‐based bicyclic β‐lactam libraries
2003
A p-toluenesulfinic acid-catalyzed three-component Ugi-type reaction and its application for the synthesis of α-amino amides and amidines
2013
Regioselective Functionalization of the Imidazole Ring via Transition Metal‐Catalyzed CN and CC Bond Forming Reactions
2010
Advances in Synthetic Applications of Hypervalent Iodine Compounds
2016 Standout
Diversity Oriented Clicking (DOC): Divergent Synthesis of SuFExable Pharmacophores from 2‐Substituted‐Alkynyl‐1‐Sulfonyl Fluoride (SASF) Hubs
2020 StandoutNobel
Synthesis of Conformationally Constrained Peptidomimetics using Multicomponent Reactions
2008
Rapid Assembly of Polyfunctional Structures Using a One‐Pot Five‐ and Six‐Component Sequential Groebke–Blackburn/Ugi/Passerini Process
2010
Applications of Palladium-Catalyzed C–N Cross-Coupling Reactions
2016 Standout
Asymmetric Catalysis of the Carbonyl-Amine Condensation: Kinetic Resolution of Primary Amines
2017 StandoutNobel
The Halogen Bond
2016 Standout
A convergent synthesis of enantiopure bicyclic scaffolds through multicomponent Ugi reaction
2007
Comprehensive Survey of Combinatorial Library Synthesis: 2000
2001
Transition Metal-Catalyzed C–H Amination: Scope, Mechanism, and Applications
2017 Standout
Chemistry and Biology Of Multicomponent Reactions
2012 Standout
Direct C−H Transformation via Iron Catalysis
2010 Standout
Cu-Catalyzed Azide−Alkyne Cycloaddition
2008 StandoutNobel
New method for the preparation of solid-phase bound isocyanocarboxylic acids and Ugi reactions therewith
2003
Solar Synthesis: Prospects in Visible Light Photocatalysis
2014 StandoutScience
Synthesis and Applications of tert-Butanesulfinamide
2010
Sulfur(VI) Fluoride Exchange (SuFEx)-Enabled High-Throughput Medicinal Chemistry
2020 StandoutNobel
Aryl−Aryl Bond Formation One Century after the Discovery of the Ullmann Reaction
2002 Standout
Works of David E. Portlock being referenced
Lead compounds discovered from libraries: Part 2
2003
Lead compounds discovered from libraries
2001
Parallel synthesis and evaluation of N-(1-phenylethyl)-5-phenyl-imidazole-2-amines as Na+/K+ ATPase inhibitors
2000
Petasis boronic acid–Mannich reactions of substituted hydrazines: synthesis of α-hydrazinocarboxylic acids
2002
Multi-Component Synthesis of Imidazo[1,2-a] Annulated Heterocycles on α-Isocyano Resin Esters
2001
Novel Petasis boronic acid–Mannich reactions with tertiary aromatic amines
2003
Solid-phase synthesis of five-dimensional libraries via a tandem Petasis–Ugi multi-component condensation reaction
2003
Solid-phase synthesis of functionalized 1,2,4-triazin-6-ones
2002
Solid-Supported Synthesis of Putative Peptide β-Turn Mimetics via Ugi Reaction for Diketopiperazine Formation
2002
The solid-phase Nenitzescu indole synthesis
2000
A tandem Petasis–Ugi multi component condensation reaction: solution phase synthesis of six dimensional libraries
2003
Hydroxylamines and sulfinamide as amine components in the Petasis boronic acid–Mannich reaction: synthesis of N-hydroxy or alkoxy-α-aminocarboxylicacids and N-(tert-butyl sulfinyl)-α-amino carboxylicacids
2003
A facile, selective KF/Al2O3 mediated method for the deprotection of aryl silyl ethers and preparation of aryl SEM ethers
2001
Benzylic halogenation of methylquinones
1972
The synthesis of aza-β-lactams via tandem Petasis–Ugi multi-component condensation and 1,3-diisopropylcarbodiimide (DIC) condensation reaction
2003
A facile KF/Al2O3 mediated method for the synthesis of substituted oxazolidinones
1999
Combination of enzymatic procedures with multicomponent condensations
2003
Dimetalated heterocycles as synthetic intermediates. V. Dianions derived from certain 2-hydroxy-4-methylpyrimidines, 2-amino-4-methylpyrimidines, and related compounds
1974
Solid-phase synthesis of functionalized 1,2,3-triazoles
2002