Citation Impact
Citing Papers
The 2.6 Angstrom Crystal Structure of a Human A 2A Adenosine Receptor Bound to an Antagonist
2008 StandoutScience
Direct Synthesis of Amides from Alcohols and Amines with Liberation of H 2
2007 StandoutScience
Oxindole Synthesis by Direct Coupling of CH and CH Centers
2009
Palladium‐Catalyzed Cross‐Coupling Reactions in Total Synthesis
2005 Standout
Potent and Selective Triazole-Based Inhibitors of the Hypoxia-Inducible Factor Prolyl-Hydroxylases with Activity in the Murine Brain
2015 StandoutNobel
Catalytic Asymmetric Three‐Component Synthesis of Homoallylic Amines
2013 StandoutNobel
Two novel series of allocolchicinoids with modified seven membered B-rings: design, synthesis, inhibition of tubulin assembly and cytotoxicity
2005
Identification of a Potent and Orally Active Non-peptide C5a Receptor Antagonist
2002
Nucleotide signalling during inflammation
2014 StandoutNature
Rhodium/phosphoramidite-catalyzed asymmetric arylation of aldehydes with arylboronic acids
2006 StandoutNobel
Purinergic Signaling in the Airways
2012
CH Bond Functionalization: Emerging Synthetic Tools for Natural Products and Pharmaceuticals
2012 Standout
Function, structure and therapeutic potential of complement C5a receptors
2007
Adenosine receptors as therapeutic targets
2006 Standout
Integrins Form an Expanding Diffusional Barrier that Coordinates Phagocytosis
2016 StandoutNobel
The tumour microenvironment after radiotherapy: mechanisms of resistance and recurrence
2015 Standout
Purinergic receptors in gastrointestinal inflammation
2007
Understanding and targeting resistance mechanisms in NSCLC
2017
Nonpeptidic ligands for peptide and protein receptors
1999
Palladium(II)‐Catalyzed CH Activation/CC Cross‐Coupling Reactions: Versatility and Practicality
2009 Standout
Pyrrolidinyl‐Spirooxindole Natural Products as Inspirations for the Development of Potential Therapeutic Agents
2007 Standout
International Union of Basic and Clinical Pharmacology. LXXXI. Nomenclature and Classification of Adenosine Receptors—An Update
2011 Standout
Immune attack: the role of inflammation in Alzheimer disease
2015 Standout
Synthesis of Oxindoles by Iron‐Catalyzed Oxidative 1,2‐Alkylarylation of Activated Alkenes with an Aryl C(sp2)H Bond and a C(sp3)H Bond Adjacent to a Heteroatom
2013
Pathophysiology and Therapeutic Potential of Purinergic Signaling
2006
The A3 adenosine receptor: An enigmatic player in cell biology
2007
Targeting apoptosis in cancer therapy
2020 Standout
Introduction to Adenosine Receptors as Therapeutic Targets
2009
Physiology and Pathophysiology of Purinergic Neurotransmission
2007 Standout
Continuous‐Flow Technology—A Tool for the Safe Manufacturing of Active Pharmaceutical Ingredients
2015 Standout
Animal Models of Alzheimer Disease
2012
Adenosine receptors: therapeutic aspects for inflammatory and immune diseases
2008 Standout
Adenosine in the airways: Implications and applications
2006
The Cross‐Dehydrogenative Coupling of CH Bonds: A Versatile Strategy for CC Bond Formations
2013 Standout
Biaryl Phosphane Ligands in Palladium‐Catalyzed Amination
2008 Standout
Exploring the full spectrum of macrophage activation
2008 Standout
Shaping of monocyte and macrophage function by adenosine receptors
2006
Organic Azides: An Exploding Diversity of a Unique Class of Compounds
2005 Standout
Preparation of 2-, 3-, 4- and 7-(2-alkylcarbamoyl-1-alkylvinyl)benzo[b]furans and their BLT1and/or BLT2inhibitory activities
2007
Tonic B cell antigen receptor signals supply an NF-κB substrate for prosurvival BLyS signaling
2008
The case for a role for adenosine in asthma: almost convincing?
2003
Integrated signalling pathways for mast-cell activation
2006 Standout
Iron Catalysis in Organic Synthesis
2015 Standout
Copper-Mediated Coupling Reactions and Their Applications in Natural Products and Designed Biomolecules Synthesis
2008 Standout
Solid phase synthesis of oligomeric guanidiniums
1998
3d Transition Metals for C–H Activation
2018 Standout
Practical Asymmetric Synthesis of an Endothelin Receptor Antagonist
1999
Multicomponent Reactions with Isocyanides
2000 Standout
Chemistry of Polyvalent Iodine
2008 Standout
Focal adhesion proteins connect IgE receptors to the cytoskeleton as revealed by micropatterned ligand arrays
2008
Safe and Reliable Synthesis of Diazoketones and Quinoxalines in a Continuous Flow Reactor
2010
A general and efficient PIFA mediated synthesis of heterocycle-fused quinolinone derivatives
2002
Synthesis of Heterocycles via Electrophilic Cyclization of Alkynes Containing Heteroatom
2011 Standout
Synthesis of Substituted Oxindoles from α-Chloroacetanilides via Palladium-Catalyzed C−H Functionalization
2003
Aryl radical cyclisation onto pyrroles
2002
The Organocatalytic Approach to Enantiopure 2H‐ and 3H‐Pyrroles: Inhibitors of the Hedgehog Signaling Pathway
2016 StandoutNobel
The Long-Term Survival Potential of Mature T Lymphocytes Is Programmed During Development in the Thymus
2011 StandoutNobel
Mandelic acid derived ionic liquids: synthesis, toxicity and biodegradability
2017
What Has Polar Surface Area Ever Done for Drug Discovery?
2011
Nucleophilic Displacement at Benzhydryl Centers: Asymmetric Synthesis of 1,1-Diarylalkyl Derivatives
2003
General and Efficient Approaches to Fused [1,2-a]Pyrroles and [1,2-a]Indoles
1997
Synthesis of Five-, Six-, and Seven-Membered Ring Lactams by Cp*Rh Complex-Catalyzed Oxidative N-Heterocyclization of Amino Alcohols
2004
Chromone: A Valid Scaffold in Medicinal Chemistry
2014 Standout
Stereoselective Enzymatic Synthesis of Heteroatom-Substituted Cyclopropanes
2018 StandoutNobel
Cyclization reactions of N-acryloyl-2-aminobenzaldehyde derivatives: formal total synthesis of martinellic acid
2006
Microwave-Assisted Sequential Amide Bond Formation and Intramolecular Amidation: A Rapid Entry to Functionalized Oxindoles
2005
Synthesis of Sulfotyrosine‐Containing Peptides by Incorporating Fluorosulfated Tyrosine Using an Fmoc‐Based Solid‐Phase Strategy
2015 StandoutNobel
Advances in the Chemistry of Tetrahydroquinolines
2011 Standout
Catalytic Dehydrogenative Cross-Coupling: Forming Carbon−Carbon Bonds by Oxidizing Two Carbon−Hydrogen Bonds
2011 Standout
Aryl−Aryl Bond Formation by Transition-Metal-Catalyzed Direct Arylation
2007 Standout
Facile Synthesis of a Family of H8BINOL-Amine Compounds and Catalytic Asymmetric Arylzinc Addition to Aldehydes
2010
Helicenes: Synthesis and Applications
2011 Standout
Structure-Based Design of β-Site APP Cleaving Enzyme 1 (BACE1) Inhibitors for the Treatment of Alzheimer’s Disease
2013
Asymmetric Synthesis of Isoquinoline Alkaloids
2004 Standout
Green and Sustainable Solvents in Chemical Processes
2018 Standout
Free radicals in the synthesis of medium-sized rings
1999
Enantiospecific, Stereospecific Total Synthesis of the Oxindole Alkaloid Alstonisine
2002
Synthesis of enantiopure mono- and disubstituted tetrahydroisoquinolines by 6-exo radical cyclizations
2001
Inactivation of C5a Anaphylatoxin by a Peptide That Is Complementary to a Region of C5a
2004 StandoutNobel
Targeting Receptor Tyrosine Kinase MET in Cancer: Small Molecule Inhibitors and Clinical Progress
2013
Cyclizations of N-Acyliminium Ions
2004 Standout
An intramolecular cycloaddition approach to pyrrolo[3,2- c ]quinolones
2002
Activation-Enabled Syntheses of Functionalized Pillar[5]arene Derivatives
2015 StandoutNobel
The “Cyclopropyl Fragment” is a Versatile Player that Frequently Appears in Preclinical/Clinical Drug Molecules
2016
The Combinatorial Synthesis of Bicyclic Privileged Structures or Privileged Substructures
2003 Standout
A tandem radical approach to the ABCE-rings of the Aspidosperma and Strychnos alkaloids
2001
Advances in Synthetic Applications of Hypervalent Iodine Compounds
2016 Standout
Palladium-Catalyzed Direct Hydroxymethylation of Aryl Halides and Triflates with Potassium Acetoxymethyltrifluoroborate
2012
Discovery and Characterization of 4‘-(2-Furyl)-N-pyridin-3-yl-4,5‘-bipyrimidin-2‘-amine (LAS38096), a Potent, Selective, and Efficacious A2BAdenosine Receptor Antagonist
2007
Synthesis of Oxindoles by Iron‐Catalyzed Oxidative 1,2‐Alkylarylation of Activated Alkenes with an Aryl C(sp2)H Bond and a C(sp3)H Bond Adjacent to a Heteroatom
2013
Dehydrogenation as a Substrate-Activating Strategy in Homogeneous Transition-Metal Catalysis
2009 Standout
New 4-Point Pharmacophore Method for Molecular Similarity and Diversity Applications: Overview of the Method and Applications, Including a Novel Approach to the Design of Combinatorial Libraries Containing Privileged Substructures
1999
A general solution to the synthesis of 2-azabicyclo[3.3.1]nonane unit of Strychnos alkaloids
1991
Some aspects of reduced quinoline chemistry
1998
Cyclic Carbopalladation. A Versatile Synthetic Methodology for the Construction of Cyclic Organic Compounds
1996 StandoutNobel
Oxindole Synthesis by Direct Coupling of CH and CH Centers
2009
Recent advancements in the homoallylamine chemistry
2002
Macrophage plasticity, polarization, and function in health and disease
2018 Standout
Metal-Free Multicomponent Syntheses of Pyridines
2014 Standout
A New Route to Spirooxindoles
2000
Works of Clive McCarthy being referenced
A Drug Resistance Screen Using a Selective MET Inhibitor Reveals a Spectrum of Mutations That Partially Overlap with Activating Mutations Found in Cancer Patients
2011
A new orally bioavailable dual adenosine A2B/A3 receptor antagonist with therapeutic potential
2005
Potent small molecule inhibitors of spleen tyrosine kinase (Syk)
2003
Discovery and SAR of potent, orally available 2,8-diaryl-quinoxalines as a new class of JAK2 inhibitors
2010
Structure based design, synthesis and SAR of cyclic hydroxyethylamine (HEA) BACE-1 inhibitors
2011
Chiral induction in aryl radical cyclisations
1989
Selective Endothelin A Receptor Antagonists. 3. Discovery and Structure−Activity Relationships of a Series of 4-Phenoxybutanoic Acid Derivatives
1998
Indole alkaloid synthesis; a stereospecific preparation of functionalised cis-hexahydrocarbazoles
1989
Macrocyclic BACE-1 inhibitors acutely reduce Aβ in brain after po application
2009
Intramolecular alkyllithium additions to lactams; a synthesis of 2,3,9,9a-tetrahydro-1H-pyrrolo[1,2-a]indoles (pyrrolo[1,2-a]indolemnes) related to mitomycins
1991
Selective Endothelin A Receptor Antagonists. 4. Discovery and Structure−Activity Relationships of Stilbene Acid and Alcohol Derivatives
1998
Selective ETAAntagonists. 5. Discovery and Structure−Activity Relationships of Phenoxyphenylacetic Acid Derivatives
2000
New non peptidic C5a receptor antagonists
1997
Aryl radical cyclisations: Quinoline, isoquinolone, and 1-benzazepin-2-onerings via 6- and 7-exo cyclisations
1991
Adenosine receptor ligands as potential therapeutics in asthma.
2002