Citation Impact
Citing Papers
SuFEx-enabled, agnostic discovery of covalent inhibitors of human neutrophil elastase
2019 StandoutNobel
Hydrazino-Pictet-Spengler Ligation as a Biocompatible Method for the Generation of Stable Protein Conjugates
2013
Diversity oriented clicking delivers β-substituted alkenyl sulfonyl fluorides as covalent human neutrophil elastase inhibitors
2022 StandoutNobel
Soft corrugated channel with synergistic exclusive discrimination gating for CO2 recognition in gas mixture
2023 StandoutNobel
In situ click chemistry generation of cyclooxygenase-2 inhibitors
2017 Standout
An efficient and convenient Cu(OAc)2/air mediated oxidative coupling of azoles via C–H activation
2009
Targeting hypoxia in cancer therapy
2011 Standout
Electrolytic Macrocyclizations: Scalable Synthesis of a Diazonamide‐Based Drug Development Candidate
2015
Cancer nanomedicine: progress, challenges and opportunities
2016 Standout
Antibiotics in the aquatic environment – A review – Part I
2009 Standout
Transition-metal mediated carbon–sulfur bond activation and transformations
2012 Standout
Selective Treatment of Hypoxic Tumor Cells In Vivo: Phosphate Pre‐Prodrugs of Nitro Analogues of the Duocarmycins
2011
Introduction of Fluorine and Fluorine‐Containing Functional Groups
2013 Standout
Brief update on endocytosis of nanomedicines
2019
LYTACs that engage the asialoglycoprotein receptor for targeted protein degradation
2021 StandoutNobel
mRNA vaccines for infectious diseases: principles, delivery and clinical translation
2021 StandoutNobel
Halogen Atoms in the Modern Medicinal Chemistry: Hints for the Drug Design
2010
SuFExable polymers with helical structures derived from thionyl tetrafluoride
2021 StandoutNobel
Antibody–drug conjugates: targeted drug delivery for cancer
2010
Natural products and Pharma 2011: Strategic changes spur new opportunities
2011
Synthesis of Selective Agonists for the α7 Nicotinic Acetylcholine Receptor with In Situ Click-Chemistry on Acetylcholine-Binding Protein Templates
2012 StandoutNobel
Strategic incorporation of fluorine into taxoid anticancer agents for medicinal chemistry and chemical biology studies
2017
Site-specific chemical protein conjugation using genetically encoded aldehyde tags
2012 StandoutNobel
Targeted drug delivery for cancer therapy: the other side of antibodies
2012
Molecular Recognition in Chemical and Biological Systems
2015
Discovery of practical production processes for arylsulfur pentafluorides and their higher homologues, bis- and tris(sulfur pentafluorides): Beginning of a new era of “super-trifluoromethyl” arene chemistry and its industry
2012
Advanced targeted therapies in cancer: Drug nanocarriers, the future of chemotherapy
2015
Transition‐Metal‐Catalyzed Direct Arylation of (Hetero)Arenes by CH Bond Cleavage
2009 Standout
Sulfur(VI) Fluoride Exchange (SuFEx): Another Good Reaction for Click Chemistry
2014 StandoutNobel
1-(3-Aryloxyaryl)benzimidazole sulfones are liver X receptor agonists
2009
Engineered Nanoparticles for Drug Delivery in Cancer Therapy
2014 Standout
Click Chemistry for Drug Development and Diverse Chemical–Biology Applications
2013 Standout
Evaluation of tert‐Butyl Isosteres: Case Studies of Physicochemical and Pharmacokinetic Properties, Efficacies, and Activities
2015
3d Transition Metals for C–H Activation
2018 Standout
SuFEx Click Chemistry Enabled Late-Stage Drug Functionalization
2018 StandoutNobel
Photothermal therapy and photoacoustic imaging via nanotheranostics in fighting cancer
2018 Standout
Bond Formations between Two Nucleophiles: Transition Metal Catalyzed Oxidative Cross-Coupling Reactions
2011 Standout
Fluorine in Pharmaceutical Industry: Fluorine-Containing Drugs Introduced to the Market in the Last Decade (2001–2011)
2013 Standout
Steric and Dynamic Parameters Influencing In Situ Cycloadditions to Form Triazole Inhibitors with Crystalline Acetylcholinesterase
2016 StandoutNobel
Cross‐Coupling Reactions on Azoles with Two and More Heteroatoms
2006
Aptamer–Drug Conjugates
2015
Fluorine and Fluorinated Motifs in the Design and Application of Bioisosteres for Drug Design
2018 Standout
Multidimensional SuFEx Click Chemistry: Sequential Sulfur(VI) Fluoride Exchange Connections of Diverse Modules Launched From An SOF4 Hub
2017 StandoutNobel
New insights into the kinetic target-guided synthesis of protein ligands
2015
Cooperative capture synthesis: yet another playground for copper-free click chemistry
2016 StandoutNobel
The Hitchhiker’s Guide to Flow Chemistry
2017 Standout
Application of the Pentafluorosulfanyl Group as a Bioisosteric Replacement
2017
Synthetic chemistry and biological activity of pentafluorosulphanyl (SF5) organic molecules
2012
The Sonogashira Reaction: A Booming Methodology in Synthetic Organic Chemistry
2007 Standout
Next Generation of Fluorine-Containing Pharmaceuticals, Compounds Currently in Phase II–III Clinical Trials of Major Pharmaceutical Companies: New Structural Trends and Therapeutic Areas
2016 Standout
Copper‐Catalyzed Direct Cross‐Coupling of Compounds Containing Activated C–H/Heteroatom–H Bonds with N‐Tosylhydrazones
2016
Arzneimittelentwicklung: Die Reduzierung von Umweltbelastungen durch gezieltes Moleküldesign
2008
Precise Modulation of CO2 Sorption in Ti8Ce2–Oxo Clusters: Elucidating Lewis Acidity of the Ce Metal Sites and Structural Flexibility
2024 StandoutNobel
Observation of the controlled assembly of preclick components in the in situ click chemistry generation of a chitinase inhibitor
2013 StandoutNobel
Biocompatible SuFEx Click Chemistry: Thionyl Tetrafluoride (SOF4)‐Derived Connective Hubs for Bioconjugation to DNA and Proteins
2019 StandoutNobel
Aryl−Aryl Bond Formation by Transition-Metal-Catalyzed Direct Arylation
2007 Standout
A fluorogenic screening platform enables directed evolution of an alkyne biosynthetic tool
2016 StandoutNobel
Synthesis of kinase inhibitors containing a pentafluorosulfanyl moiety
2017
<i>In Situ</i> Click Chemistry for the Identification of a Potent D-Amino Acid Oxidase Inhibitor
2015 StandoutNobel
Sustainable from the very beginning: rational design of molecules by life cycle engineering as an important approach for green pharmacy and green chemistry
2007
Kinetic Target-Guided Synthesis in Drug Discovery and Chemical Biology: A Comprehensive Facts and Figures Survey
2016
Aerobic Copper-Catalyzed Organic Reactions
2013 Standout
Protein-Catalyzed Capture Agents
2019
Synthetic Organic Electrochemical Methods Since 2000: On the Verge of a Renaissance
2017 Standout
Site-Specific Traceless Coupling of Potent Cytotoxic Drugs to Recombinant Antibodies for Pharmacodelivery
2012
Identification of simple arylfluorosulfates as potent agents against resistant bacteria
2021 StandoutNobel
Alternative Synthetic Methods through New Developments in Catalysis by Gold
2008 Standout
Palladium-Catalyzed C–S Coupling: Access to Thioethers, Benzo[b]thiophenes, and Thieno[3,2-b]thiophenes
2011
Regioselective Functionalization of the Imidazole Ring via Transition Metal‐Catalyzed CN and CC Bond Forming Reactions
2010
Diversity Oriented Clicking (DOC): Divergent Synthesis of SuFExable Pharmacophores from 2‐Substituted‐Alkynyl‐1‐Sulfonyl Fluoride (SASF) Hubs
2020 StandoutNobel
Creation of Customized Bioactivity within a 14-Membered Macrolide Scaffold: Design, Synthesis, and Biological Evaluation Using a Family-18 Chitinase
2015 StandoutNobel
Fluorosulfuryl Isocyanate Enabled SuFEx Ligation of Alcohols and Amines
2021 StandoutNobel
Engineering Folate–Drug Conjugates to Target Cancer: From Chemistry to Clinic
2012
Applications of Palladium-Catalyzed C–N Cross-Coupling Reactions
2016 Standout
The Halogen Bond
2016 Standout
Exploration of Fluorine Chemistry at the Multidisciplinary Interface of Chemistry and Biology
2013
From 2000 to Mid-2010: A Fruitful Decade for the Synthesis of Pyrazoles
2011 Standout
Arylfluorosulfates Inactivate Intracellular Lipid Binding Protein(s) through Chemoselective SuFEx Reaction with a Binding Site Tyr Residue
2016 StandoutNobel
Applications of Fluorine in Medicinal Chemistry
2015 Standout
Synthetic Approaches to the Microtubule-Stabilizing Sponge Alkaloid Ceratamine A and Desbromo Analogues
2009
Reactive oxygen species generating systems meeting challenges of photodynamic cancer therapy
2016 Standout
Sulfur(VI) Fluoride Exchange (SuFEx)-Enabled High-Throughput Medicinal Chemistry
2020 StandoutNobel
Preparation and Utility of Organic Pentafluorosulfanyl-Containing Compounds
2014
In situclick chemistry: from small molecule discovery to synthetic antibodies
2012
Works of Bernhard Stump being referenced
Safe Handling of Cytotoxic Compounds in a Biopharmaceutical Environment
2013
Pentafluorosulfanyl as a Novel Building Block for Enzyme Inhibitors: Trypanothione Reductase Inhibition and Antiprotozoal Activities of Diarylamines
2008
Diaryl sulfide-based inhibitors of trypanothione reductase: inhibition potency, revised binding mode and antiprotozoal activities
2008
Betraying the Parasite’s Redox System: Diaryl Sulfide‐Based Inhibitors of Trypanothione Reductase: Subversive Substrates and Antitrypanosomal Properties
2007
Synthesis, Inhibition Potency, Binding Mode, and Antiprotozoal Activities of Fluorescent Inhibitors of Trypanothione Reductase Based on Mepacrine‐Conjugated Diaryl Sulfide Scaffolds
2009
Structure‐Based Design, Synthesis, and in vitro Evaluation of Nonpeptidic Neprilysin Inhibitors
2004
Generation of Candidate Ligands for Nicotinic Acetylcholine Receptors via in situ Click Chemistry with a Soluble Acetylcholine Binding Protein Template
2012 StandoutNobel
A New Class of Inhibitors for the Metalloprotease Neprilysin Based on a Central Imidazole Scaffold
2005
Antibody−Drug Conjugates: Linking Cytotoxic Payloads to Monoclonal Antibodies
2009