Citation Impact
Citing Papers
SuFEx-enabled, agnostic discovery of covalent inhibitors of human neutrophil elastase
2019 StandoutNobel
Sulfur [ 18 F]Fluoride Exchange Click Chemistry Enabled Ultrafast Late-Stage Radiosynthesis
2021 StandoutNobel
Diversity oriented clicking delivers β-substituted alkenyl sulfonyl fluorides as covalent human neutrophil elastase inhibitors
2022 StandoutNobel
Retinoic acid receptors: From molecular mechanisms to cancer therapy
2014
SGLT2 inhibitors for primary and secondary prevention of cardiovascular and renal outcomes in type 2 diabetes: a systematic review and meta-analysis of cardiovascular outcome trials
2018 Standout
Dynamic Covalent Chemistry
2002 StandoutNobel
Open Babel: An open chemical toolbox
2011 Standout
Amide bond formation: beyond the myth of coupling reagents
2008 Standout
Signals from the gut microbiota to distant organs in physiology and disease
2016
Standards and guidelines for the interpretation of sequence variants: a joint consensus recommendation of the American College of Medical Genetics and Genomics and the Association for Molecular Pathology
2015 Standout
The road to fully programmable protein catalysis
2022 StandoutNatureNobel
Catalysis for fluorination and trifluoromethylation
2011 StandoutNature
Emil Knoevenagel and the Roots of Aminocatalysis
2010 StandoutNobel
Isoquinolin‐1‐one Inhibitors of the MDM2–p53 Interaction
2008
Design of Flexible Lewis Acidic Sites in Porous Coordination Polymers by using the Viologen Moiety
2012 StandoutNobel
The Catalytic Asymmetric Knoevenagel Condensation
2011 StandoutNobel
Iterative In Situ Click Chemistry Creates Antibody‐like Protein‐Capture Agents
2009 StandoutNobel
Organocatalytic Enantioselective Decarboxylative Aldol Reaction of Malonic Acid Half Thioesters with Aldehydes
2013 StandoutNobel
Canagliflozin and Cardiovascular and Renal Events in Type 2 Diabetes
2017 Standout
Click Chemistry: Diverse Chemical Function from a Few Good Reactions
2001 StandoutNobel
Enterochromaffin Cells Are Gut Chemosensors that Couple to Sensory Neural Pathways
2017 StandoutNobel
Amplification of Dynamic Chiral Crown Ether Complexes During Cyclic Acetal Formation
2003 StandoutNobel
The discovery and optimization of hexahydro-2H-pyrano[3,2-c]quinolines (HHPQs) as potent and selective inhibitors of the mitotic kinesin-5
2010
Thirteen decades of peptide synthesis: key developments in solid phase peptide synthesis and amide bond formation utilized in peptide ligation
2017
Intestinal Crosstalk between Bile Acids and Microbiota and Its Impact on Host Metabolism
2016 Standout
Solid-supported reagents in organic synthesis
1999
Comprehensive survey of chemical libraries yielding enzyme inhibitors, receptor agonists and antagonists, and other biologically active agents: 1992 through 1997
1997
Catalytic CC, CN, and CO Ullmann‐Type Coupling Reactions
2009 Standout
Antibacterial drug discovery in the resistance era
2016 StandoutNature
SGLT-2 inhibitors: Their pleiotropic properties
2016
Strategy for Mitigating DKA Risk in Patients with Type 1 Diabetes on Adjunctive Treatment with SGLT Inhibitors: A STICH Protocol
2018
Click Chemistry for Drug Development and Diverse Chemical–Biology Applications
2013 Standout
Copper-Mediated Coupling Reactions and Their Applications in Natural Products and Designed Biomolecules Synthesis
2008 Standout
SuFEx Click Chemistry Enabled Late-Stage Drug Functionalization
2018 StandoutNobel
Conversion of Imine to Oxazole and Thiazole Linkages in Covalent Organic Frameworks
2018 StandoutNobel
Tandem Catalysis: Three Mechanistically Distinct Reactions from a Single Ruthenium Complex
2000 StandoutNobel
Room-Temperature Ionic Liquids: Solvents for Synthesis and Catalysis. 2
2011 Standout
Methodologies for Generating Solution-Phase Combinatorial Libraries
2000
Environmentally benign metal-free decarboxylative aldol and Mannich reactions
2009
Structure of the STRA6 receptor for retinol uptake
2016 StandoutScienceNobel
Tetrahydroquinoline syntheses induced with catalytic amounts of viologen additives
2009
Oligosaccharide Mimetics Obtained by Novel, Rapid Screening of Carboxylic Acid Encoded Glycopeptide Libraries
1998 StandoutNobel
Multidimensional SuFEx Click Chemistry: Sequential Sulfur(VI) Fluoride Exchange Connections of Diverse Modules Launched From An SOF4 Hub
2017 StandoutNobel
The Catalytic Asymmetric Mukaiyama–Michael Reaction of Silyl Ketene Acetals with α,β‐Unsaturated Methyl Esters
2017 StandoutNobel
Cooperative capture synthesis: yet another playground for copper-free click chemistry
2016 StandoutNobel
Multistep Solid-State Organic Synthesis of Carbamate-Linked Covalent Organic Frameworks
2019 StandoutNobel
Combinatorial Synthesis of Small Organic Molecules
1996
Iminium Catalysis
2007
Palladium-catalyzed coupling of functionalized bromoarenes to a polystyrene-bound aryl tributylstannane
1999
The Current Status of Heterocyclic Combinatorial Libraries
1997
Organizing Principles of Mammalian Nonsense-Mediated mRNA Decay
2013
Copper-Catalyzed Synthesis of Mixed Alkyl Aryl Phosphonates
2014 StandoutNobel
Unlocking Reactivity of TrpB: A General Biocatalytic Platform for Synthesis of Tryptophan Analogues
2017 StandoutNobel
Double-level “orthogonal” dynamic combinatorial libraries on transition metal template
2001
Comprehensive Survey of Combinatorial Library Synthesis: 1999
2000
Comprehensive Survey of Combinatorial Library Synthesis: 2001
2002
Solid-phase organic reactions II: A review of the literature Nov 95–Nov 96
1997
Click Chemistry: Diverse Chemical Function from a Few Good Reactions
2001 StandoutNobel
Comprehensive Survey of Combinatorial Library Synthesis: 2005
2006
Target-Oriented and Diversity-Oriented Organic Synthesis in Drug Discovery
2000 StandoutScience
Identification of simple arylfluorosulfates as potent agents against resistant bacteria
2021 StandoutNobel
Cyclizations of N-Acyliminium Ions
2004 Standout
The Combinatorial Synthesis of Bicyclic Privileged Structures or Privileged Substructures
2003 Standout
Chemomimetic Biocatalysis: Exploiting the Synthetic Potential of Cofactor-Dependent Enzymes To Create New Catalysts
2015 StandoutNobel
Diversity Oriented Clicking (DOC): Divergent Synthesis of SuFExable Pharmacophores from 2‐Substituted‐Alkynyl‐1‐Sulfonyl Fluoride (SASF) Hubs
2020 StandoutNobel
Multi-step organic synthesis using solid-supported reagents and scavengers: a new paradigm in chemical library generation
2000
Asymmetric Catalysis of the Carbonyl-Amine Condensation: Kinetic Resolution of Primary Amines
2017 StandoutNobel
A one-pot multicomponent coupling/cyclization for natural product herbicide (±)-thaxtomin A
2014
Investigation of SAR requirements of SR 142801 through an indexed combinatorial library in solution
1999
Synthesis and Applications of Small Molecule Libraries
1996
Comprehensive Survey of Combinatorial Library Synthesis: 2000
2001
Copper-Mediated Synthesis ofN-Acyl Vinylogous Carbamic Acids and Derivatives: Synthesis of the Antibiotic CJ-15,801
2003
Chemistry and Biology Of Multicomponent Reactions
2012 Standout
The “One-Bead-One-Compound” Combinatorial Library Method
1997
Comprehensive Survey of Combinatorial Library Synthesis: 1998
1999
Katalytische C‐C‐, C‐N‐ und C‐O‐Ullmann‐Kupplungen
2009
Parallel Personal Comments on “Classical” Papers in Combinatorial Chemistry
1998
Polymer-Supported Tetrafluorophenol: A New Activated Resin for Chemical Library Synthesis
2000
Solar Synthesis: Prospects in Visible Light Photocatalysis
2014 StandoutScience
Imine exchange inO-aryl andO-alkyl oximes as a base reaction for aqueous ‘dynamic’ combinatorial libraries. A kinetic and thermodynamic study
1999
Significant facilitation of metal-free aerobic oxidative cyclization of imines with water in synthesis of benzimidazoles
2014
Sulfur(VI) Fluoride Exchange (SuFEx)-Enabled High-Throughput Medicinal Chemistry
2020 StandoutNobel
SPOCC: A Resin for Solid-Phase Organic Chemistry and Enzymatic Reactions on Solid Phase
1999 StandoutNobel
Dapagliflozin and Cardiovascular Outcomes in Type 2 Diabetes
2018 Standout
Challenges of Antibacterial Discovery
2011
Ar−F Reductive Elimination from Palladium(II) Revisited
2007
Synopsis of Some Recent Tactical Application of Bioisosteres in Drug Design
2011 Standout
The role of organometallic copper(iii) complexes in homogeneous catalysis
2013
Works of Benoît Déprez being referenced
Rescue of nonsense mutations by amlexanox in human cells
2012
The Bile Acid Chenodeoxycholic Acid Increases Human Brown Adipose Tissue Activity
2015
Parallel synthesis of a library of 1,4-naphthoquinones and automated screening of potential inhibitors of trypanothione reductase from Trypanosoma cruzi
2000
A library of novel hydroxamic acids targeting the metallo-protease family: Design, parallel synthesis and screening
2006
Automated parallel synthesis of a tetrahydroisoquinolin-based library: Potential prolyl endopeptidase inhibitors
1999
Novel non-carboxylic acid retinoids: 1,2,4-Oxadiazol-5-one derivatives
2008
Synthetic EthR inhibitors boost antituberculous activity of ethionamide
2009
Designing Focused Chemical Libraries Enriched in Protein-Protein Interaction Inhibitors using Machine-Learning Methods
2010
Inhibition of the glucose transporter SGLT2 with dapagliflozin in pancreatic alpha cells triggers glucagon secretion
2015
Versatile Acylation ofN-Nucleophiles Using a New Polymer-Supported 1-Hydroxybenzotriazole Derivative
1997
UFU (‘Ullmann–Finkelstein–Ullmann’): a new multicomponent reaction
2006
Lewis acid-induced reaction of homophthalic anhydride with imines: a convenient synthesis of trans-isoquinolonic acids
1998
Orthogonal Combinatorial Chemical Libraries
1995
Synthesis of five- and six-membered lactams via solvent-free microwave Ugi reaction
2010
Combinatorial chemistry: A rational approach to chemical diversity
1996
Parallel synthesis of polysubstituted tetrahydroquinolines
1998
Kinetic Target-Guided Synthesis in Drug Discovery and Chemical Biology: A Comprehensive Facts and Figures Survey
2016
Monitoring of a three-step solid phase synthesis involving a Heck reaction using magic angle spinning NMR spectroscopy
1996
Parallel synthesis of 1,2,4-oxadiazoles from carboxylic acids using an improved, uronium-based, activation
2001
Novel Selective Inhibitors of the Zinc Plasmodial Aminopeptidase PfA-M1 as Potential Antimalarial Agents
2007
Synthesis of N-(iodophenyl)-amides via an unprecedented Ullmann–Finkelstein tandem reaction
2005
From Hit to Lead. Analyzing Structure−Profile Relationships
2001
Efficient propylphosphonic anhydride (®T3P) mediated synthesis of benzothiazoles, benzoxazoles and benzimidazoles
2012
Hydroxamates: Relationships between Structure and Plasma Stability
2009