Citation Impact
Citing Papers
Bioavailability enhancing activities of natural compounds from medicinal plants.
2009
Corneal Permeation of Ganciclovir: Mechanism of Ganciclovir Permeation Enhancement by Acyl Ester Prodrug Design
2002
Guidelines for the welfare and use of animals in cancer research
2010 Standout
TEER Measurement Techniques for In Vitro Barrier Model Systems
2015 Standout
Effluxing ABC transporters in human corneal epithelium
2009
Incorporation of novel 1-alkylcarbonyloxymethyl prodrugs of 5-fluorouracil into poly(lactide-co-glycolide) nanoparticles
2007
Quinolines and structurally related heterocycles as antimalarials
2010 Standout
The influence of drug-like concepts on decision-making in medicinal chemistry
2007 Standout
Micellar Solubilization of Some Poorly Soluble Antidiabetic Drugs: A Technical Note
2008
Virtual screening of intestinal drug permeability
2000
Controlled release of 5-fluorouridine from radiation-crosslinked poly(ethylene-co-vinyl acetate) films
2006
Predicting Drug Absorption from Molecular Surface Properties Based on Molecular Dynamics Simulations
1998
Permeability of cornea, sclera, and conjunctiva: A literature analysis for drug delivery to the eye
1998
Ocular Drug Delivery
2010 Standout
Amorphous pharmaceutical solids: preparation, characterization and stabilization
2001 Standout
Rapid translocation of nanoparticles from the lung airspaces to the body
2010 StandoutNobel
Assessment of disorder in crystalline powdersâa review of analytical techniques and their application
1999
Dolasetron
1997
Pharmaceutical Applications of Cyclodextrins. 1. Drug Solubilization and Stabilization
1996 Standout
Biomedical applications of biodegradable polymers
2011 Standout
Bioavailability enhancers of herbal origin: An overview
2013 Standout
Biological roles of glycans
2016 Standout
Effect of molecular weight of PGG–paclitaxel conjugates on in vitro and in vivo efficacy
2012
The Endocannabinoid System as an Emerging Target of Pharmacotherapy
2006 Standout
Chemical stability and plasma-catalyzed dealkylation of peptidyl-α-hydroxyglycine derivatives—Intermediates in peptide α-amidation
1991
PEGylation as a strategy for improving nanoparticle-based drug and gene delivery
2015 Standout
Design, synthesis and in vitro drug release investigation of new potential 5-FU prodrugs
2011
How Structural Features Influence the Biomembrane Permeability of Peptides
1996
Correlating Partitioning and Caco-2 Cell Permeability of Structurally Diverse Small Molecular Weight Compounds
1998
Analysis of anticancer drugs: A review
2011 Standout
The effect of a modified β-cyclodextrin, SBE4-β-CD, on the aqueous stability and ocular absorption of pilocarpine
1994
Caco-2 monolayers in experimental and theoretical predictions of drug transport1PII of original article: S0169-409X(96)00415-2. The article was originally published in Advanced Drug Delivery Reviews 22 (1996) 67–84.1
2001
5-Substituted-1H-tetrazoles as carboxylic acid isosteres: medicinal chemistry and synthetic methods
2002 Standout
Phytochemistry of Cannabis sativa L.
2017 Standout
Cannabinoids in the treatment of glaucoma
2002
Mechanisms in photodynamic therapy: part one—photosensitizers, photochemistry and cellular localization
2004 Standout
Indoles as therapeutics of interest in medicinal chemistry: Bird's eye view
2017 Standout
Transcorneal Permeation of l- and d-Aspartate Ester Prodrugs of Acyclovir: Delineation of Passive Diffusion Versus Transporter Involvement
2008
Drug release kinetics and transport mechanisms of non-degradable and degradable polymeric delivery systems
2010 Standout
Engineered Nanoparticles for Drug Delivery in Cancer Therapy
2014 Standout
Functional expression of a sodium dependent nucleoside transporter on rabbit cornea: Role in corneal permeation of acyclovir and idoxuridine
2003
Nitric oxide-donating carbonic anhydrase inhibitors for the treatment of open-angle glaucoma
2009
Synthesis and mechanistic investigations of pH-responsive cationic poly(aminoester)s
2020
Effect of the carriers on the microstructure of mango powder obtained by spray drying and its functional characterization
2005 Standout
Property-Based Design: Optimization of Drug Absorption and Pharmacokinetics
2001
(C) Means to enhance penetration
1992
Lessons Learned from Marketed and Investigational Prodrugs
2004
Molecular Properties That Influence the Oral Bioavailability of Drug Candidates
2002 Standout
Prediction of Drug Absorption Using Multivariate Statistics
2000 Standout
Improvement of oral and rectal bioavailabilities of carmofur by methylated β-cyclodextrin complexations
1987
Derivatives of 5‐Aminolevulinic Acid for Photodynamic Therapy: Enzymatic Conversion into Protoporphyrin
1998
One-Component Multifunctional Sequence-Defined Ionizable Amphiphilic Janus Dendrimer Delivery Systems for mRNA
2021 StandoutNobel
The Medicinal Chemist’s Toolbox: An Analysis of Reactions Used in the Pursuit of Drug Candidates
2011 Standout
Imidazolidin-4-one Derivatives of Primaquine as Novel Transmission-Blocking Antimalarials
2005
Investigation ofN‐[(Acyloxy)alkyl] Ester as a Prodrug Model for Drugs Containing the Phenyltetrazole Moiety
1994
Degradable Controlled-Release Polymers and Polymeric Nanoparticles: Mechanisms of Controlling Drug Release
2016 Standout
Cyclodextrin Drug Carrier Systems
1998 Standout
Caco-2 monolayers in experimental and theoretical predictions of drug transport
1996
Drug Solubility: Importance and Enhancement Techniques
2012 Standout
Ribosomal Synthesis of Dehydroalanine-Containing Peptides
2006 StandoutNobel
Fast Calculation of Molecular Polar Surface Area as a Sum of Fragment-Based Contributions and Its Application to the Prediction of Drug Transport Properties
2000 Standout
Models for polyurethane hydrolysis under moderately acidic conditions: A comparative study of hydrolysis rates of urethanes, ureas, and amides
1989
Mechanisms Whereby Mononuclear Copper Proteins Functionalize Organic Substrates
1996 Standout
N-Glycosylation of Campylobacter jejuni Surface Proteins Promotes Bacterial Fitness
2013
Ocular absorption following topical delivery
1995
?-Azido acids for direct use in solid-phase peptide synthesis
2000 StandoutNobel
Physicochemical and drug-delivery considerations for oral drug bioavailability
1996
Prodrugs for improved ocular drug delivery
1989
5‐Substituted 1H‐Tetrazoles as Carboxylic Acid Isosteres: Medicinal Chemistry and Synthetic Methods
2003 Standout
Multiple Binding Modes of Inhibitors to Carbonic Anhydrases: How to Design Specific Drugs Targeting 15 Different Isoforms?
2012 Standout
Works of Anders Buur being referenced
Prodrugs of Peptides. 18. Synthesis and Evaluation of Various Esters of Desmopressin (dDAVP)
1993
Role of Enzymatic Lability in the Corneal and Conjunctival Penetration of Timolol Ester Prodrugs in the Pigmented Rabbit
1991
Assessment of the combined approach of N-alkylation and salt formation to enhance aqueous solubility of tertiary amines using bupivacaine as a model drug
2004
Prodrugs of 5-Fluorouracil V. 1-Alkoxycarbonyl Derivatives as Potential Prodrug Forms for Improved Rectal or Oral Delivery of 5-Fluorouracil
1986
Prodrugs of propranolol: hydrolysis and intramolecular aminolysis of various propranolol esters and an oxazolidin-2-one derivative
1988
Prodrugs as drug delivery systems. 65. Hydrolysis of α-hydroxy-and α-acyloxy-N-benzoylglycine derivatives and implications for the design of prodrugs of NH-acidic compounds
1987
Prodrugs of 5-fluorouracil. I. Hydrolysis kinetics and physicochemical properties of various N-acyl derivatives of 5-fluorouracil
1984
Permeability of 5-fluorouracil and prodrugs in Caco-2 cell monolayers
1996
Prodrugs of 5-fluorouracil. III. Hydrolysis kinetics in aqueous solution and biological media, lipophilicity and solubility of various 1-carbamoyl derivatives of 5-fluorouracil
1985
Prodrugs of peptides
1988
Prodrugs of 5-fluorouracil. VII. Hydrolysis kinetics and physicochemical properties of N-ethoxy- and N-phenoxycarbonyloxymethyl derivatives of 5-fluorouracil.
1986
Drug Delivery Studies in Caco-2 Monolayers. Synthesis, Hydrolysis, and Transport of O-Cyclopropane Carboxylic Acid Ester Prodrugs of Various β-Blocking Agents
1995
Application of isothermal microcalorimetry in preformulation. I. Hygroscopicity of drug substances
1997
Prodrugs of 5-fluorouracil. IV. Hydrolysis kinetics, bioactivation and physicochemical properties of various N-acyloxymethyl derivatives of 5-fluorouracil
1985
Timolol prodrugs: synthesis, stability and lipophilicity of various alkyl, cycloalkyl and aromatic esters of timolol
1988
Prodrugs of timolol for improved ocular delivery: synthesis, hydrolysis kinetics and lipophilicity of various timolol esters
1986
Low dose O-butyryl timolol improves the therapeutic index of timolol in the pigmented rabbit.
1988
Improved corneal penetration of timolol by prodrugs as a means to reduce systemic drug load.
1987