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Recent Development and Application of Chiral Phase-Transfer Catalysts
2007
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Copper in cross-coupling reactions
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Chemistry and Biology of the Zaragozic Acids (Squalestatins)
1996
Selectivity in the cycloadditions of carbonyl ylides with glyoxylates: an approach to the zaragozic acids—squalestatins
2000
5‐(Pyrrolidine‐2‐yl)tetrazole: Rationale for the Increased Reactivity of the Tetrazole Analogue of Proline in Organocatalyzed Aldol Reactions
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Ruthenium-Catalyzed Reactions for Organic Synthesis
1998
The biology , function , and biomedical applications of exosomes
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Direct organocatalytic asymmetric epoxidation of α,β-unsaturated aldehydes
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Confined acids catalyze asymmetric single aldolizations of acetaldehyde enolates
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Anion−π and π−π Cooperative Interactions Regulating the Self-Assembly of Nitrate−Triazine−Triazine Complexes
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Green chemistry by nano-catalysis
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Anion‐π‐Wechselwirkungen ins rechte Licht gerückt
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Der Stand der Totalsynthese zu Beginn des 21. Jahrhunderts
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Selective Anion Encapsulation by a Metalated Cryptophane with a π-Acidic Interior
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Synthetic Applications of Nonmetal Catalysts for Homogeneous Oxidations
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Anion−π Interactions in Crystal Structures: Commonplace or Extraordinary?
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2005
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Structural Criteria for the Design of Anion Receptors: The Interaction of Halides with Electron-Deficient Arenes
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Activation of olefins via asymmetric Brønsted acid catalysis
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Nano-organocatalyst: magnetically retrievable ferrite-anchored glutathione for microwave-assisted Paal–Knorr reaction, aza-Michael addition, and pyrazole synthesis
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Cu-Catalyzed Azide−Alkyne Cycloaddition
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Effect of the Metal‐Assisted Assembling Mode on the Redox States of Hexaazatriphenylene Hexacarbonitrile
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Dynamic Control of Chiral Space in a Catalytic Asymmetric Reaction Using a Molecular Motor
2011 StandoutScienceNobel
Applying Flow Chemistry: Methods, Materials, and Multistep Synthesis
2013
Organocatalytic Asymmetric Epoxidation of Olefins by Chiral Ketones
2004
Asymmetric Enamine Catalysis
2007 StandoutNobel
Iminomalonate as a Convenient Electrophilic Amination Reagent for Grignard Reagents
2002
Asymmetric α‐Amination of Aldehydes Catalyzed by PS‐Diphenylprolinol Silyl Ethers: Remediation of Catalyst Deactivation for Continuous Flow Operation
2012
A Unified Total Synthesis of the Immunomodulators (−)-Rapamycin and (−)-27-Demethoxyrapamycin: Construction of the C(21−42) Perimeters
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Totalsynthese der CP-Verbindungen CP-263,114 und CP 225,917 – Teil 1: Synthese von Schlüsselintermediaten und neue präparative Erkenntnisse
1999
The Art of Innovation in Organic Chemistry: Synthetic Efforts toward the Phomoidrides
2003
Total Synthesis of the Squalene Synthase Inhibitor Zaragozic Acid C
2005
Anion−π Interactions in a Carousel Copper(II)−Triazine Complex
2004
Magnetically Driven Agitation in a Tube Mixer Affords Clog-Resistant Fast Mixing Independent of Linear Velocity
2011
“Inverse Drug Discovery” Strategy To Identify Proteins That Are Targeted by Latent Electrophiles As Exemplified by Aryl Fluorosulfates
2017 StandoutNobel
A monolithic 5-(pyrrolidin-2-yl)tetrazole flow microreactor for the asymmetric aldol reaction in water–ethanol solvent
2015
Asymmetrische Katalyse durch chirale Wasserstoffbrückendonoren
2006
Are Oxazolidinones Really Unproductive, Parasitic Species in Proline Catalysis? – Thoughts and Experiments Pointing to an Alternative View
2007
Synthesis of a Precursor to Sacubitril Using Enabling Technologies
2015
Wechselwirkungen mit aromatischen Ringen in chemischen und biologischen Erkennungsprozessen
2003
Enantioselective organocatalytic epoxidation using hypervalent iodine reagents
2006
Novel Process Windows for Enabling, Accelerating, and Uplifting Flow Chemistry
2013
Asymmetric Organocatalysis in Continuous Flow: Opportunities for Impacting Industrial Catalysis
2015
Works of Alan Armstrong being referenced
The Flow’s the Thing…Or Is It? Assessing the Merits of Homogeneous Reactions in Flask and Flow
2010
Kinetic Template‐Guided Tethering of Fragments
2012
Kinetic and mechanistic studies of proline-mediated direct intermolecular aldol reactions
2009
Thermodynamic control of asymmetric amplification in amino acid catalysis
2006 Nature
A mechanistic rationalization of unusual kinetic behavior in proline-mediated C–O and C–N bond-forming reactions
2006
Rationalization and Prediction of Solution Enantiomeric Excess in Ternary Phase Systems
2006
Kinetic Rationalization of Nonlinear Effects in Asymmetric Catalysis Based on Phase Behavior
2006
Amine‐Catalyzed Epoxidation of Alkenes: A New Mechanism for the Activation of Oxone
2004
Direct Azole Amination: CH Functionalization as a New Approach to Biologically Important Heterocycles
2010
Water in Organocatalytic Processes: Debunking the Myths
2007
Der Fluss ist das Ding … oder ist er es? Ein Vergleich homogener Reaktionen in Reaktionskolben und Durchflussreaktoren
2010
A highly convergent total synthesis of the spiroacetal macrolide (+)-milbemycinβ1
1989
Enantioselective cation binding with a functionalized podand ionophore
1992
Catalytic enantioselective epoxidation of alkenes with a tropinone-derived chiral ketone
1998
Wasser in organokatalytischen Prozessen: ein Mythos wird entschleiert
2007
Asymmetric epoxidation catalyzed by esters of α-hydroxy-8-oxabicyclo[3.2.1]octan-3-one
2001
Synthetic studies on CP-225,917 and CP-263,114: concise synthesis of the bicyclic core using an intramolecular Mukaiyama aldol reactionElectronic supplementary information (ESI) available: crystal data for 13a. See http://www.rsc.org/suppdata/p1/b2/b202752f/
2002
Aminkatalysierte Epoxidierung von Alkenen: ein neuer Mechanismus zur Aktivierung von Oxone
2004
Highly stereoselective intramolecular epoxidation in unsaturated oxaziridines
1999
Approaches to the γ-lactone unit of CP-225,917 and CP-263,114
2002
Unusual Reversal of Enantioselectivity in the Proline-Mediated α-Amination of Aldehydes Induced by Tertiary Amine Additives
2010
Total Synthesis of Avermectin B1a: Planning of the Synthesis and Preparation of the C1-C10 "Southern" Hydrobenzofuran Fragment
1990
Total synthesis of (+)-zaragozic acid C
1998
Enamine Carboxylates as Stereodetermining Intermediates in Prolinate Catalysis
2011
Pyrrolidine-Derived Iminium Salts as Catalysts for Alkene Epoxidation by Oxone®
1997
Total Synthesis of (+)-Zaragozic Acid C
2000
Alkene epoxidation catalyzed by bicyclo[3.2.1]octan-3-ones: effects of structural modifications on catalyst efficiency and epoxidation enantioselectivity
2000
Kinetic Rationalization of Nonlinear Effects in Asymmetric Catalysis Based on Phase Behavior
2006
Rationalization and Prediction of Solution Enantiomeric Excess in Ternary Phase Systems
2006
Recent synthetic studies on the zaragozic acids (squalestatins)
2002
Electrophilic amination of carbanions by N-carboxamido oxaziridines
2000
Intramolecular Epoxidation of Unsaturated Oxaziridines
1998
Enantioselective Epoxidation of Alkenes Catalyzed by 2-Fluoro-N-Carbethoxytropinone and Related Tropinone Derivatives
2002
Synthesis of the Bicyclo[4.4.1]decenone Core of CP-225,917 and CP-263,114
1998
Exocyclic iminium salts as catalysts for alkene epoxidation by Oxone®
1999
Stereocontrolled Synthesis of 3-(trans-2-Aminocyclopropyl)alanine, a Key Component of Belactosin A
2003
Direkte Azolaminierung: C‐H‐Funktionalisierung zur Herstellung biologisch wichtiger Heterocyclen
2010
Emergence of Solution-Phase Homochirality via Crystal Engineering of Amino Acids
2007
Curtin–Hammett Paradigm for Stereocontrol in Organocatalysis by Diarylprolinol Ether Catalysts
2012
A one-step synthesis of tetrahydropyranopyranones from carbonyl compounds
2001
Total Synthesis of Avermectin B1a: Final Coupling Reactions and the Total Synthesis of Avermectin B1a Aglycone
1990
Anion−Aromatic Bonding: A Case for Anion Recognition by π-Acidic Rings
2002
Probing the Active Catalyst in Product-Accelerated Proline-Mediated Reactions
2004
Transition State Stereoelectronics in Alkene Epoxidations by Fluorinated Dioxiranes
2000
Clarification of the Role of Water in Proline-Mediated Aldol Reactions
2007
Kinetic Profiling of Prolinate-Catalyzed α-Amination of Aldehydes
2011
Total synthesis of the anthelmintic macrolide avermectin B1a
1991
α-Functionalised ketones as promoters of alkene epoxidation by Oxone®
1999
Mechanistic Rationalization of Organocatalyzed Conjugate Addition of Linear Aldehydes to Nitro-olefins
2011
Total synthesis of (+)-milbemycin β1
1989
Asymmetric electrophilic amination of enolates by a chiral N-alkoxycarbonyloxaziridine
2001
Synthetic studies on amphidinolides C and F: synthesis of the C18–C29 segment of amphidinolide F
2009
Synthesis of the Bicyclic Core of the Zaragozic Acids (Squalestatins)
1995