Adrian Glas

Expansive discovery of chemically diverse structured macrocyclic oligoamides

Accurate de novo design of heterochiral protein–protein interactions

Targeted Protein Degradation: from Chemical Biology to Drug Discovery

Discovery and optimization of peptide macrocycles

Coronavirus envelope protein: current knowledge

Anchor extension: a structure-guided approach to design cyclic peptides targeting enzyme active sites

Synthetic Peptides as Protein Mimics

End-to-end design of wearable sensors

Naturally Occurring Oxazole-Containing Peptides

Rational Tuning of Fluorobenzene Probes for Cysteine‐Selective Protein Modification

CPProtectides: Rapid uptake of well‐folded β‐hairpin peptides with enhanced resistance to intracellular degradation

Natural Products as Sources of New Drugs over the Nearly Four Decades from 01/1981 to 09/2019

Hydrocarbon Stapled Peptides as Modulators of Biological Function

Hydrogen Bond Surrogate Stabilization of β-Hairpins

Diversity Oriented Clicking (DOC): Divergent Synthesis of SuFExable Pharmacophores from 2‐Substituted‐Alkynyl‐1‐Sulfonyl Fluoride (SASF) Hubs

Rational Tuning of Fluorobenzene Probes for Cysteine‐Selective Protein Modification

Catalytic Asymmetric Synthesis of Unprotected β²-Amino Acids

Diversity Oriented Clicking (DOC): Divergent Synthesis of SuFExable Pharmacophores from 2‐Substituted‐Alkynyl‐1‐Sulfonyl Fluoride (SASF) Hubs

Rapid biocompatible macrocyclization of peptides with decafluoro-diphenylsulfone

Strategies for the Diversity-Oriented Synthesis of Macrocycles

Natural Products as Sources of New Drugs from 1981 to 2014

Chemical Inhibition of ENL/AF9 YEATS Domains in Acute Leukemia

Stapled β-Hairpins Featuring 4-Mercaptoproline

Differential Effects of β³‐ versus β²‐Amino Acid Residues on the Helicity and Recognition Properties of Bim BH3‐Derived α/β‐Peptides

Modulators of Protein–Protein Interactions

Structure‐Based Design of Inhibitors of Protein–Protein Interactions: Mimicking Peptide Binding Epitopes

Adapting free energy perturbation simulations for large macrocyclic ligands: how to dissect contributions from direct binding and free ligand flexibility

Strukturbasierte Entwicklung von Protein‐Protein‐Interaktionsinhibitoren: Stabilisierung und Nachahmung von Peptidliganden

Constraining an Irregular Peptide Secondary Structure through Ring‐Closing Alkyne Metathesis

Constrained Peptides with Target‐Adapted Cross‐Links as Inhibitors of a Pathogenic Protein–Protein Interaction